Compile Data Set for Download or QSAR
Report error Found 53 Enz. Inhib. hit(s) with all data for entry = 50021386
TargetCannabinoid receptor 2(Human)
Université

Curated by ChEMBL
LigandPNGBDBM50224081(N3-(1-(3,5-dimethyl)adamantyl)-7-chloro-4-oxo-1-pe...)
Affinity DataKi:  5.30nMAssay Description:Inhibition of human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
Université

Curated by ChEMBL
LigandPNGBDBM50224046((-)-N3-(1-(1-adamantyl)ethyl)-4-oxo-1-pentyl-1,4-d...)
Affinity DataKi:  14nMAssay Description:Inhibition of human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
Université

Curated by ChEMBL
LigandPNGBDBM50224077(N3-(1-(3,5-dimethyl)adamantyl)-1-pentyl-4-thioxo-1...)
Affinity DataKi:  18.2nMAssay Description:Inhibition of human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
Université

Curated by ChEMBL
LigandPNGBDBM50224059(N3-(1-(3,5-dimethyl)adamantyl)-4-oxo-1-pentyl-1,4-...)
Affinity DataKi:  23.5nMAssay Description:Inhibition of human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
Université

Curated by ChEMBL
LigandPNGBDBM50224052(adamantane-1-carboxylic Acid (4-Oxo-1-pentyl-1,4-d...)
Affinity DataKi:  25.5nMAssay Description:Inhibition of human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
Université

Curated by ChEMBL
LigandPNGBDBM50224051((-)-N3-(1-(1-adamantyl)ethyl)-7-chloro-4-oxo-1-pen...)
Affinity DataKi:  26.1nMAssay Description:Inhibition of human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
Université

Curated by ChEMBL
LigandPNGBDBM50224063(N3-(1-(3,5-dimethyl)adamantyl)-8-chloro-4-oxo-1-pe...)
Affinity DataKi:  27.4nMAssay Description:Inhibition of human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
Université

Curated by ChEMBL
LigandPNGBDBM50224061(N3-(1-(3,5-dimethyl)adamantyl)-4-oxo-1-pentyl-1,4-...)
Affinity DataKi:  30.9nMAssay Description:Inhibition of human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
Université

Curated by ChEMBL
LigandPNGBDBM50224062(N3-((1-adamantyl)methyl)-4-oxo-1-pentyl-1,4-dihydr...)
Affinity DataKi:  50.6nMAssay Description:Inhibition of human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
Université

Curated by ChEMBL
LigandPNGBDBM50224064(N3-(1-(3,5-dimethyl)adamantyl)-6-chloro-4-oxo-1-pe...)
Affinity DataKi:  54.6nMAssay Description:Inhibition of human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
Université

Curated by ChEMBL
LigandPNGBDBM50224083(N3-(1-(3,5-dimethyl)adamantyl)-4-oxo-1-(4-fluorobe...)
Affinity DataKi:  83.4nMAssay Description:Inhibition of human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
Université

Curated by ChEMBL
LigandPNGBDBM50224068(N3-(1-(3,5-dimethyl)adamantyl)-4-oxo-1-pentyl-1,4-...)
Affinity DataKi:  93nMAssay Description:Inhibition of human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
Université

Curated by ChEMBL
LigandPNGBDBM50224050(N3-(1-(3,5-dimethyl)adamantyl)-4-oxo-2-phenyl-1-pe...)
Affinity DataKi:  119nMAssay Description:Inhibition of human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
Université

Curated by ChEMBL
LigandPNGBDBM50224074((+)-N3-(1-(1,2,3,4-tetrahydronaphthyl))-6-chloro-4...)
Affinity DataKi:  121nMAssay Description:Inhibition of human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
Université

Curated by ChEMBL
LigandPNGBDBM50224074((+)-N3-(1-(1,2,3,4-tetrahydronaphthyl))-6-chloro-4...)
Affinity DataKi:  121nMAssay Description:Inhibition of human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
Université

Curated by ChEMBL
LigandPNGBDBM50224045((-)-N3-(1-(1-adamantyl)ethyl)-6-chloro-4-oxo-1-pen...)
Affinity DataKi:  144nMAssay Description:Inhibition of human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
Université

Curated by ChEMBL
LigandPNGBDBM50224045((-)-N3-(1-(1-adamantyl)ethyl)-6-chloro-4-oxo-1-pen...)
Affinity DataKi:  144nMAssay Description:Inhibition of human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
Université

Curated by ChEMBL
LigandPNGBDBM50224045((-)-N3-(1-(1-adamantyl)ethyl)-6-chloro-4-oxo-1-pen...)
Affinity DataKi:  144nMAssay Description:Inhibition of human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
Université

Curated by ChEMBL
LigandPNGBDBM50224054(N3-(1-adamantyl)-4-oxo-1-(2-(morpholin-4-yl)ethyl)...)
Affinity DataKi:  152nMAssay Description:Inhibition of human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
Université

Curated by ChEMBL
LigandPNGBDBM50224072(3-(naphthalene-1-carbonyl)-1-pentyl-1,4-dihydroqui...)
Affinity DataKi:  154nMAssay Description:Inhibition of human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
Université

Curated by ChEMBL
LigandPNGBDBM50224069(N3-(1-(3,5-dimethyl)adamantyl)-4-oxo-1-(3-phenylpr...)
Affinity DataKi:  160nMAssay Description:Inhibition of human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
Université

Curated by ChEMBL
LigandPNGBDBM50224082(N3-(1-(3,5-dimethyl)adamantyl)-2-methyl-4-oxo-1-pe...)
Affinity DataKi:  200nMAssay Description:Inhibition of human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
Université

Curated by ChEMBL
LigandPNGBDBM50224046((-)-N3-(1-(1-adamantyl)ethyl)-4-oxo-1-pentyl-1,4-d...)
Affinity DataKi:  202nMAssay Description:Inhibition of human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
Université

Curated by ChEMBL
LigandPNGBDBM50224046((-)-N3-(1-(1-adamantyl)ethyl)-4-oxo-1-pentyl-1,4-d...)
Affinity DataKi:  202nMAssay Description:Inhibition of human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
Université

Curated by ChEMBL
LigandPNGBDBM50224056(N3-(1-(3,5-dimethyl)adamantyl)-4-oxo-1-(2-(morphol...)
Affinity DataKi:  221nMAssay Description:Inhibition of human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
Université

Curated by ChEMBL
LigandPNGBDBM50224047(1-(4-fluorobenzyl)-3-(naphthalene-1-carbonyl)-1,4-...)
Affinity DataKi:  225nMAssay Description:Inhibition of human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
Université

Curated by ChEMBL
LigandPNGBDBM50224057(N3-(1-(3,5-dimethyl)adamantyl)-4-oxo-1-pentyl-1,4-...)
Affinity DataKi:  259nMAssay Description:Inhibition of human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
Université

Curated by ChEMBL
LigandPNGBDBM50224078(naphthalene-1-carboxylic acid (4-xo-1-pentyl-1,4-d...)
Affinity DataKi:  265nMAssay Description:Inhibition of human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
Université

Curated by ChEMBL
LigandPNGBDBM50224051((-)-N3-(1-(1-adamantyl)ethyl)-7-chloro-4-oxo-1-pen...)
Affinity DataKi:  265nMAssay Description:Inhibition of human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
Université

Curated by ChEMBL
LigandPNGBDBM50224051((-)-N3-(1-(1-adamantyl)ethyl)-7-chloro-4-oxo-1-pen...)
Affinity DataKi:  265nMAssay Description:Inhibition of human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
Université

Curated by ChEMBL
LigandPNGBDBM50224070(N3-(1-(3,5-dimethyl)adamantyl)-4-oxo-1-(2-phenylet...)
Affinity DataKi:  333nMAssay Description:Inhibition of human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
Université

Curated by ChEMBL
LigandPNGBDBM50224055(N3-(1-adamantyl)-4-oxo-1-pentyl-2-phenyl-1,4-dihyd...)
Affinity DataKi:  338nMAssay Description:Inhibition of human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
Université

Curated by ChEMBL
LigandPNGBDBM50224060(3-benzoyl-1-pentyl-1,4-dihydroquinolin-4-one | CHE...)
Affinity DataKi:  446nMAssay Description:Inhibition of human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
Université

Curated by ChEMBL
LigandPNGBDBM50224087(1-hexyl-3-(naphthalene-1-carbonyl)-1,4-dihydroquin...)
Affinity DataKi:  582nMAssay Description:Inhibition of human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
Université

Curated by ChEMBL
LigandPNGBDBM50224085(1-benzyl-3-(naphthalene-1-carbonyl)-1,4-dihydroqui...)
Affinity DataKi:  656nMAssay Description:Inhibition of human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
Université

Curated by ChEMBL
LigandPNGBDBM50224075((-)-N3-(1-phenylethyl)-2-methyl-4-oxo-1-pentyl-1,4...)
Affinity DataKi:  663nMAssay Description:Inhibition of human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
Université

Curated by ChEMBL
LigandPNGBDBM50224065(1-(4-bromobenzyl)-3-(naphthalene-1-carbonyl)-1,4-d...)
Affinity DataKi:  966nMAssay Description:Inhibition of human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
Université

Curated by ChEMBL
LigandPNGBDBM50180028((RS)-N3-(1-(1,2,3,4-tetrahydronaphthyl))-4-oxo-1-p...)
Affinity DataKi:  1.01E+3nMAssay Description:Inhibition of human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
Université

Curated by ChEMBL
LigandPNGBDBM50180028((RS)-N3-(1-(1,2,3,4-tetrahydronaphthyl))-4-oxo-1-p...)
Affinity DataKi:  1.01E+3nMAssay Description:Inhibition of human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
Université

Curated by ChEMBL
LigandPNGBDBM50224067(1-(4-chlorobenzyl)-3-(naphthalene-1-carbonyl)-1,4-...)
Affinity DataKi:  1.12E+3nMAssay Description:Inhibition of human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
Université

Curated by ChEMBL
LigandPNGBDBM50224073(N-(4-oxo-1-pentyl-1,4-dihydroquinolin-3-yl)-3-phen...)
Affinity DataKi:  1.13E+3nMAssay Description:Inhibition of human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
Université

Curated by ChEMBL
LigandPNGBDBM50224066(3-(naphthalene-2-carbonyl)-1-pentyl-1,4-dihydroqui...)
Affinity DataKi:  1.29E+3nMAssay Description:Inhibition of human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
Université

Curated by ChEMBL
LigandPNGBDBM50224071(3-(anthracene-9-carbonyl)-1-pentyl-1,4-dihydroquin...)
Affinity DataKi:  1.50E+3nMAssay Description:Inhibition of human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
Université

Curated by ChEMBL
LigandPNGBDBM50224049(1-butyl-3-(naphthalene-1-carbonyl)-1,4-dihydroquin...)
Affinity DataKi:  1.55E+3nMAssay Description:Inhibition of human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
Université

Curated by ChEMBL
LigandPNGBDBM50224084(3-((1-adamantyl)aminomethyl)-1-pentyl-1H-quinolin-...)
Affinity DataKi:  1.67E+3nMAssay Description:Inhibition of human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
Université

Curated by ChEMBL
LigandPNGBDBM50224088(3-(naphthalene-1-carbonyl)-1-(2-(cyclohexyl)ethyl)...)
Affinity DataKi:  1.67E+3nMAssay Description:Inhibition of human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
Université

Curated by ChEMBL
LigandPNGBDBM50224058(3-(benzo[1,3]dioxole-5-carbonyl)-1-pentyl-1,4-dihy...)
Affinity DataKi: >2.00E+3nMAssay Description:Inhibition of human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
Université

Curated by ChEMBL
LigandPNGBDBM50224053(1-hexyl-3-(4-methoxybenzoyl)-1,4-dihydroquinolin-4...)
Affinity DataKi: >2.00E+3nMAssay Description:Inhibition of human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
Université

Curated by ChEMBL
LigandPNGBDBM50224048((-)-N3-(1-(2-naphthyl)ethyl)-2-methyl-4-oxo-1-pent...)
Affinity DataKi: >2.00E+3nMAssay Description:Inhibition of human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
Université

Curated by ChEMBL
LigandPNGBDBM50224086(3-(naphthalene-1-carbonyl)-1-phenylpropyl-1,4-dihy...)
Affinity DataKi: >2.00E+3nMAssay Description:Inhibition of human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
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