Compile Data Set for Download or QSAR
Report error Found 101 Enz. Inhib. hit(s) with all data for entry = 50041920
TargetEpidermal growth factor receptor(Human)
Korea Institute of Science and Technology

Curated by ChEMBL
LigandPNGBDBM3639(N-(3-bromophenyl)-6-(morpholin-4-ylmethyl)-8H-pyrr...)
Affinity DataIC50: 9.55nMAssay Description:Inhibition autophosphorylation of EGFR in human DiFi cells after 2 hrs by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEpidermal growth factor receptor(Human)
Korea Institute of Science and Technology

Curated by ChEMBL
LigandPNGBDBM3641(5-[(3-Bromophenyl)amino]-3-[[N-(carboxymethyl)-N-m...)
Affinity DataIC50: 9.55nMAssay Description:Inhibition autophosphorylation of EGFR in human DiFi cells after 2 hrs by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEpidermal growth factor receptor(Human)
Korea Institute of Science and Technology

Curated by ChEMBL
LigandPNGBDBM3638(N-(3-bromophenyl)-6-[(dimethylamino)methyl]-8H-pyr...)
Affinity DataIC50: 9.77nMAssay Description:Inhibition autophosphorylation of EGFR in human DiFi cells after 2 hrs by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEpidermal growth factor receptor(Human)
Korea Institute of Science and Technology

Curated by ChEMBL
LigandPNGBDBM3624(N-(3-bromophenyl)-1-methyl-1H-pyrazolo[4,3-g]quina...)
Affinity DataIC50: 12.9nMAssay Description:Inhibition autophosphorylation of EGFR in human DiFi cells after 2 hrs by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEpidermal growth factor receptor(Human)
Korea Institute of Science and Technology

Curated by ChEMBL
LigandPNGBDBM3634(5-[(3-Bromophenyl)amino]-1-[2-(4-morpholino)ethyl]...)
Affinity DataIC50: 15.8nMAssay Description:Inhibition autophosphorylation of EGFR in human DiFi cells after 2 hrs by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEpidermal growth factor receptor(Human)
Korea Institute of Science and Technology

Curated by ChEMBL
LigandPNGBDBM3582(N-(3-bromophenyl)-1H-pyrazolo[4,3-g]quinazolin-5-a...)
Affinity DataIC50: 19.9nMAssay Description:Inhibition autophosphorylation of EGFR in human DiFi cells after 2 hrs by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEpidermal growth factor receptor(Human)
Korea Institute of Science and Technology

Curated by ChEMBL
LigandPNGBDBM3583(Pyrroloquinazoline deriv. 3a | Anilinopyrimidine d...)
Affinity DataIC50: 21.9nMAssay Description:Inhibition autophosphorylation of EGFR in human DiFi cells after 2 hrs by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEpidermal growth factor receptor(Human)
Korea Institute of Science and Technology

Curated by ChEMBL
LigandPNGBDBM3630(N-(3-bromophenyl)-8-methyl-8H-pyrrolo[3,2-g]quinaz...)
Affinity DataIC50: 21.9nMAssay Description:Inhibition autophosphorylation of EGFR in human DiFi cells after 2 hrs by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEpidermal growth factor receptor(Human)
Korea Institute of Science and Technology

Curated by ChEMBL
LigandPNGBDBM3631(5-[(3-Bromophenyl)amino]-1-(2,3-dihydroxypropyl)-p...)
Affinity DataIC50: 49.0nMAssay Description:Inhibition autophosphorylation of EGFR in human DiFi cells after 2 hrs by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEpidermal growth factor receptor(Human)
Korea Institute of Science and Technology

Curated by ChEMBL
LigandPNGBDBM3032(CHEMBL29197 | N-(3-bromophenyl)-6,7-dimethoxyquina...)
Affinity DataIC50: 70.8nMAssay Description:Inhibition autophosphorylation of EGFR in human DiFi cells after 2 hrs by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEpidermal growth factor receptor(Human)
Korea Institute of Science and Technology

Curated by ChEMBL
LigandPNGBDBM3635(N-(3-bromophenyl)-8-[3-(morpholin-4-yl)propyl]-8H-...)
Affinity DataIC50: 77.6nMAssay Description:Inhibition autophosphorylation of EGFR in human DiFi cells after 2 hrs by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEpidermal growth factor receptor(Human)
Korea Institute of Science and Technology

Curated by ChEMBL
LigandPNGBDBM31090((E)-N-[4-(3-chloro-4-fluoroanilino)-3-cyano-7-etho...)
Affinity DataIC50: 79.4nMAssay Description:Inhibition autophosphorylation of EGFR in human DiFi cells after 2 hrs by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEpidermal growth factor receptor(Human)
Korea Institute of Science and Technology

Curated by ChEMBL
LigandPNGBDBM3640(5-[(3-Bromophenyl)amino]-3-[(N,N,N-trimethylethyle...)
Affinity DataIC50: 81.3nMAssay Description:Inhibition autophosphorylation of EGFR in human DiFi cells after 2 hrs by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEpidermal growth factor receptor(Human)
Korea Institute of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50122578(4-Dimethylamino-but-2-ynoic acid [4-(3-bromo-pheny...)
Affinity DataIC50: 89.1nMAssay Description:Inhibition autophosphorylation of EGFR in human DiFi cells after 2 hrs by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEpidermal growth factor receptor(Human)
Korea Institute of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50122565(4-Dipropylamino-but-2-ynoic acid [4-(3-bromo-pheny...)
Affinity DataIC50: 129nMAssay Description:Inhibition autophosphorylation of EGFR in human DiFi cells after 2 hrs by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEpidermal growth factor receptor(Human)
Korea Institute of Science and Technology

Curated by ChEMBL
LigandPNGBDBM3637(5-[(3-Bromophenyl)amino]-3-[[N,N-bis(2-hydroxyethy...)
Affinity DataIC50: 135nMAssay Description:Inhibition autophosphorylation of EGFR in human DiFi cells after 2 hrs by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEpidermal growth factor receptor(Human)
Korea Institute of Science and Technology

Curated by ChEMBL
LigandPNGBDBM3632(5-[(3-Bromophenyl)amino]-1-[2-(N,N-dimethylamino)-...)
Affinity DataIC50: 145nMAssay Description:Inhibition autophosphorylation of EGFR in human DiFi cells after 2 hrs by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEpidermal growth factor receptor(Human)
Korea Institute of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50122570((2S)4-(2-Methoxymethyl-pyrrolidin-1-yl)-but-2-ynoi...)
Affinity DataIC50: 151nMAssay Description:Inhibition autophosphorylation of EGFR in human DiFi cells after 2 hrs by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEpidermal growth factor receptor(Human)
Korea Institute of Science and Technology

Curated by ChEMBL
LigandPNGBDBM4473(4-(4-Fluoro-3-trifluoromethylphenylamino)-6,7-dime...)
Affinity DataIC50: 158nMAssay Description:Inhibition autophosphorylation of EGFR in human DiFi cells after 2 hrs by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEpidermal growth factor receptor(Human)
Korea Institute of Science and Technology

Curated by ChEMBL
LigandPNGBDBM4446(4-[(3-chlorophenyl)amino]-6,7-dimethoxyquinoline-3...)
Affinity DataIC50: 182nMAssay Description:Inhibition autophosphorylation of EGFR in human DiFi cells after 2 hrs by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEpidermal growth factor receptor(Human)
Korea Institute of Science and Technology

Curated by ChEMBL
LigandPNGBDBM4445(4-[(3-bromophenyl)amino]-6,7-dimethoxyquinoline-3-...)
Affinity DataIC50: 191nMAssay Description:Inhibition autophosphorylation of EGFR in human DiFi cells after 2 hrs by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEpidermal growth factor receptor(Human)
Korea Institute of Science and Technology

Curated by ChEMBL
LigandPNGBDBM3627(5-[(3-Bromophenyl)amino]-1-[2-(4-morpholino)ethyl]...)
Affinity DataIC50: 191nMAssay Description:Inhibition autophosphorylation of EGFR in human DiFi cells after 2 hrs by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEpidermal growth factor receptor(Human)
Korea Institute of Science and Technology

Curated by ChEMBL
LigandPNGBDBM3633(N-(3-bromophenyl)-8-[3-(dimethylamino)propyl]-8H-p...)
Affinity DataIC50: 229nMAssay Description:Inhibition autophosphorylation of EGFR in human DiFi cells after 2 hrs by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEpidermal growth factor receptor(Human)
Korea Institute of Science and Technology

Curated by ChEMBL
LigandPNGBDBM4468(4-(4-Isopropylphenylamino)-6,7-dimethoxyquinoline-...)
Affinity DataIC50: 229nMAssay Description:Inhibition autophosphorylation of EGFR in human DiFi cells after 2 hrs by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEpidermal growth factor receptor(Human)
Korea Institute of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50418616(CHEMBL1797541)
Affinity DataIC50: 251nMAssay Description:Inhibition autophosphorylation of EGFR in human DiFi cells after 2 hrs by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEpidermal growth factor receptor(Human)
Korea Institute of Science and Technology

Curated by ChEMBL
LigandPNGBDBM3626(N-(3-bromophenyl)-1-[2-(dimethylamino)ethyl]-1H-py...)
Affinity DataIC50: 263nMAssay Description:Inhibition autophosphorylation of EGFR in human DiFi cells after 2 hrs by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEpidermal growth factor receptor(Human)
Korea Institute of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50122567((E)-4-Dimethylamino-but-2-enoic acid [4-(3-bromo-p...)
Affinity DataIC50: 309nMAssay Description:Inhibition autophosphorylation of EGFR in human DiFi cells after 2 hrs by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEpidermal growth factor receptor(Human)
Korea Institute of Science and Technology

Curated by ChEMBL
LigandPNGBDBM3625(3-{5-[(3-bromophenyl)amino]-1H-pyrazolo[4,3-g]quin...)
Affinity DataIC50: 316nMAssay Description:Inhibition autophosphorylation of EGFR in human DiFi cells after 2 hrs by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEpidermal growth factor receptor(Human)
Korea Institute of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50148234(3-Methoxymethoxy-propynoic acid [4-(3-bromo-phenyl...)
Affinity DataIC50: 331nMAssay Description:Inhibition autophosphorylation of EGFR in human DiFi cells after 2 hrs by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEpidermal growth factor receptor(Human)
Korea Institute of Science and Technology

Curated by ChEMBL
LigandPNGBDBM4485(4-[(3-bromophenyl)amino]-6,7-dihydroxyquinoline-3-...)
Affinity DataIC50: 347nMAssay Description:Inhibition autophosphorylation of EGFR in human DiFi cells after 2 hrs by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEpidermal growth factor receptor(Human)
Korea Institute of Science and Technology

Curated by ChEMBL
LigandPNGBDBM4469(6,7-dimethoxy-4-{[2-(propan-2-yl)phenyl]amino}quin...)
Affinity DataIC50: 363nMAssay Description:Inhibition autophosphorylation of EGFR in human DiFi cells after 2 hrs by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEpidermal growth factor receptor(Human)
Korea Institute of Science and Technology

Curated by ChEMBL
LigandPNGBDBM4443(4-[(3-bromophenyl)amino]-6,7-diethoxyquinoline-3-c...)
Affinity DataIC50: 417nMAssay Description:Inhibition autophosphorylation of EGFR in human DiFi cells after 2 hrs by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEpidermal growth factor receptor(Human)
Korea Institute of Science and Technology

Curated by ChEMBL
LigandPNGBDBM4456(4-(3-Chloro-4-fluorophenylamino)-6,7-dimethoxyquin...)
Affinity DataIC50: 537nMAssay Description:Inhibition autophosphorylation of EGFR in human DiFi cells after 2 hrs by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEpidermal growth factor receptor(Human)
Korea Institute of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50122577(4-Thiomorpholin-4-yl-but-2-ynoic acid [4-(3-bromo-...)
Affinity DataIC50: 550nMAssay Description:Inhibition autophosphorylation of EGFR in human DiFi cells after 2 hrs by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEpidermal growth factor receptor(Human)
Korea Institute of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50122579(N-[4-(3-Chloro-4-fluoro-phenylamino)-3-cyano-7-eth...)
Affinity DataIC50: 562nMAssay Description:Inhibition autophosphorylation of EGFR in human DiFi cells after 2 hrs by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEpidermal growth factor receptor(Human)
Korea Institute of Science and Technology

Curated by ChEMBL
LigandPNGBDBM3642(5-[(3-bromophenyl)amino]-3-[[N-(carboxymethyl)-N-m...)
Affinity DataIC50: 589nMAssay Description:Inhibition autophosphorylation of EGFR in human DiFi cells after 2 hrs by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEpidermal growth factor receptor(Human)
Korea Institute of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50122562(N-[4-(3-Bromo-phenylamino)-3-cyano-quinolin-6-yl]-...)
Affinity DataIC50: 589nMAssay Description:Inhibition autophosphorylation of EGFR in human DiFi cells after 2 hrs by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEpidermal growth factor receptor(Human)
Korea Institute of Science and Technology

Curated by ChEMBL
LigandPNGBDBM4475(4-[(4-bromo-3-methylphenyl)amino]-6,7-dimethoxyqui...)
Affinity DataIC50: 617nMAssay Description:Inhibition autophosphorylation of EGFR in human DiFi cells after 2 hrs by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEpidermal growth factor receptor(Human)
Korea Institute of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50122563((E)-4-Dimethylamino-but-2-enoic acid [4-(3-chloro-...)
Affinity DataIC50: 646nMAssay Description:Inhibition autophosphorylation of EGFR in human DiFi cells after 2 hrs by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEpidermal growth factor receptor(Human)
Korea Institute of Science and Technology

Curated by ChEMBL
LigandPNGBDBM4449(4-[(3-fluorophenyl)amino]-6,7-dimethoxyquinoline-3...)
Affinity DataIC50: 741nMAssay Description:Inhibition autophosphorylation of EGFR in human DiFi cells after 2 hrs by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEpidermal growth factor receptor(Human)
Korea Institute of Science and Technology

Curated by ChEMBL
LigandPNGBDBM4465(6,7-Dimethoxy-4-(3-methylthiophenylamino)quinoline...)
Affinity DataIC50: 759nMAssay Description:Inhibition autophosphorylation of EGFR in human DiFi cells after 2 hrs by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEpidermal growth factor receptor(Human)
Korea Institute of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50122588(4-Methoxy-but-2-ynoic acid [4-(3-bromo-phenylamino...)
Affinity DataIC50: 794nMAssay Description:Inhibition autophosphorylation of EGFR in human DiFi cells after 2 hrs by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEpidermal growth factor receptor(Human)
Korea Institute of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50122560(4-Dimethylamino-but-2-enoic acid [4-(3-bromo-pheny...)
Affinity DataIC50: 794nMAssay Description:Inhibition autophosphorylation of EGFR in human DiFi cells after 2 hrs by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEpidermal growth factor receptor(Human)
Korea Institute of Science and Technology

Curated by ChEMBL
LigandPNGBDBM4453(4-(3-Aminophenylamino)-6,7-dimethoxyquinoline-3-ca...)
Affinity DataIC50: 813nMAssay Description:Inhibition autophosphorylation of EGFR in human DiFi cells after 2 hrs by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEpidermal growth factor receptor(Human)
Korea Institute of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50122583(N-[4-(3-Bromo-phenylamino)-3-cyano-7-methoxy-quino...)
Affinity DataIC50: 813nMAssay Description:Inhibition autophosphorylation of EGFR in human DiFi cells after 2 hrs by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEpidermal growth factor receptor(Human)
Korea Institute of Science and Technology

Curated by ChEMBL
LigandPNGBDBM4474(4-[(3-bromo-2-methylphenyl)amino]-6,7-dimethoxyqui...)
Affinity DataIC50: 832nMAssay Description:Inhibition autophosphorylation of EGFR in human DiFi cells after 2 hrs by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEpidermal growth factor receptor(Human)
Korea Institute of Science and Technology

Curated by ChEMBL
LigandPNGBDBM4454(4-{[3-(dimethylamino)phenyl]amino}-6,7-dimethoxyqu...)
Affinity DataIC50: 851nMAssay Description:Inhibition autophosphorylation of EGFR in human DiFi cells after 2 hrs by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEpidermal growth factor receptor(Human)
Korea Institute of Science and Technology

Curated by ChEMBL
LigandPNGBDBM4455(6,7-dimethoxy-4-[(3-nitrophenyl)amino]quinoline-3-...)
Affinity DataIC50: 871nMAssay Description:Inhibition autophosphorylation of EGFR in human DiFi cells after 2 hrs by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEpidermal growth factor receptor(Human)
Korea Institute of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50122572(But-2-ynoic acid [4-(3-bromo-phenylamino)-3-cyano-...)
Affinity DataIC50: 912nMAssay Description:Inhibition autophosphorylation of EGFR in human DiFi cells after 2 hrs by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEpidermal growth factor receptor(Human)
Korea Institute of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50122573(But-2-ynoic acid [4-(3-bromo-phenylamino)-3-cyano-...)
Affinity DataIC50: 933nMAssay Description:Inhibition autophosphorylation of EGFR in human DiFi cells after 2 hrs by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
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