Compile Data Set for Download or QSAR
Report error Found 6 Enz. Inhib. hit(s) with all data for entry = 50037955
TargetP2X purinoceptor 3(Human)
Institute of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50219120(LVVYPWT | CHEMBL395493)
Affinity DataIC50: 0.00830nMAssay Description:Antagonist activity at human P2X3 receptor expressed in Xenopus oocytes assessed as inhibition of ATP-induced ion current by two electrode voltage cl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetP2X purinoceptor 3(Human)
Institute of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50219120(LVVYPWT | CHEMBL395493)
Affinity DataIC50: 0.0481nMAssay Description:Antagonist activity at human recombinant P2X3 receptor expressed in Xenopus oocytes assessed as inhibition of ATP-induced ion current in presence of ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetP2X purinoceptor 3(Human)
Institute of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50219121(AVVYPWT | CHEMBL238310)
Affinity DataIC50: 14.3nMAssay Description:Antagonist activity at human P2X3 receptor expressed in Xenopus oocytes assessed as inhibition of ATP-induced ion current by two electrode voltage cl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetP2X purinoceptor 3(Human)
Institute of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50219123(LAVYPWT | CHEMBL395723)
Affinity DataIC50: 32.4nMAssay Description:Antagonist activity at human P2X3 receptor expressed in Xenopus oocytes assessed as inhibition of ATP-induced ion current by two electrode voltage cl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetP2X purinoceptor 3(Human)
Institute of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50219122(cyclic LVVYPWT | CHEMBL397926)
Affinity DataIC50: 82.4nMAssay Description:Antagonist activity at human P2X3 receptor expressed in Xenopus oocytes assessed as inhibition of ATP-induced ion current by two electrode voltage cl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetP2X purinoceptor 3(Human)
Institute of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50064800(2-(4-Formyl-5-hydroxy-6-methyl-3-phosphonooxymethy...)
Affinity DataIC50: 108nMAssay Description:Antagonist activity at human P2X3 receptor expressed in Xenopus oocytes assessed as inhibition of ATP-induced ion current by two electrode voltage cl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed