Compile Data Set for Download or QSAR
Report error Found 10 Enz. Inhib. hit(s) with all data for entry = 3580
TargetEstrogen receptor(Human)
University of New Mexico Health Sciences Center

LigandPNGBDBM17292([2,4,6,7-3H]-17beta-estradiol | [3H]-estradiol | 1...)
Affinity DataKi:  0.650nMAssay Description:Competitive binding of estrogen to GPR30 and ER alpha were conducted using COS-7 cells transfected with GPR30-GFP or ER alpha-GFP and fluorescent est...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/18/2011
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
University of New Mexico Health Sciences Center

LigandPNGBDBM36492(E2-NMe3+)
Affinity DataKi:  1.40nMAssay Description:Competitive binding of estrogen to GPR30 and ER alpha were conducted using COS-7 cells transfected with GPR30-GFP or ER alpha-GFP and fluorescent est...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/18/2011
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
University of New Mexico Health Sciences Center

LigandPNGBDBM36491(E2-COO-)
Affinity DataKi:  2nMAssay Description:Competitive binding of estrogen to GPR30 and ER alpha were conducted using COS-7 cells transfected with GPR30-GFP or ER alpha-GFP and fluorescent est...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/18/2011
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
University of New Mexico Health Sciences Center

LigandPNGBDBM36493(E2-NB)
Affinity DataKi:  2.70nMAssay Description:Competitive binding of estrogen to GPR30 and ER alpha were conducted using COS-7 cells transfected with GPR30-GFP or ER alpha-GFP and fluorescent est...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/18/2011
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
University of New Mexico Health Sciences Center

LigandPNGBDBM36490(E2-NH3+)
Affinity DataKi:  4.10nMAssay Description:Competitive binding of estrogen to GPR30 and ER alpha were conducted using COS-7 cells transfected with GPR30-GFP or ER alpha-GFP and fluorescent est...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/18/2011
Entry Details Article
PubMed
TargetG-protein coupled estrogen receptor 1(Human)
University of New Mexico Health Sciences Center

LigandPNGBDBM17292([2,4,6,7-3H]-17beta-estradiol | [3H]-estradiol | 1...)
Affinity DataKi:  9nMAssay Description:Competitive binding of estrogen to GPR30 and ER alpha were conducted using COS-7 cells transfected with GPR30-GFP or ER alpha-GFP and fluorescent est...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/18/2011
Entry Details Article
PubMed
TargetG-protein coupled estrogen receptor 1(Human)
University of New Mexico Health Sciences Center

LigandPNGBDBM36493(E2-NB)
Affinity DataKi:  16nMAssay Description:Competitive binding of estrogen to GPR30 and ER alpha were conducted using COS-7 cells transfected with GPR30-GFP or ER alpha-GFP and fluorescent est...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/18/2011
Entry Details Article
PubMed
TargetG-protein coupled estrogen receptor 1(Human)
University of New Mexico Health Sciences Center

LigandPNGBDBM36492(E2-NMe3+)
Affinity DataKi:  17nMAssay Description:Competitive binding of estrogen to GPR30 and ER alpha were conducted using COS-7 cells transfected with GPR30-GFP or ER alpha-GFP and fluorescent est...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/18/2011
Entry Details Article
PubMed
TargetG-protein coupled estrogen receptor 1(Human)
University of New Mexico Health Sciences Center

LigandPNGBDBM36490(E2-NH3+)
Affinity DataKi:  25nMAssay Description:Competitive binding of estrogen to GPR30 and ER alpha were conducted using COS-7 cells transfected with GPR30-GFP or ER alpha-GFP and fluorescent est...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/18/2011
Entry Details Article
PubMed
TargetG-protein coupled estrogen receptor 1(Human)
University of New Mexico Health Sciences Center

LigandPNGBDBM36491(E2-COO-)
Affinity DataKi:  30nMAssay Description:Competitive binding of estrogen to GPR30 and ER alpha were conducted using COS-7 cells transfected with GPR30-GFP or ER alpha-GFP and fluorescent est...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/18/2011
Entry Details Article
PubMed