Compile Data Set for Download or QSAR
Report error Found 11 Enz. Inhib. hit(s) with all data for entry = 50020854
TargetCannabinoid receptor 2(Human)
Taisho Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50218270((Z)-N-(5-tert-butyl-3-(cyclopropylmethyl)-4-methyl...)
Affinity DataEC50:  7.20nMAssay Description:Agonist activity at human CB2 receptor expressed in CHO cells by [35S]GTP-gamma-S binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
Taisho Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM5035(CHEMBL235747 | N-[(2Z)-5-tert-butyl-3,4-dimethyl-2...)
Affinity DataEC50:  110nMAssay Description:Agonist activity at human CB2 receptor expressed in CHO cells by [35S]GTP-gamma-S binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
Taisho Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50218270((Z)-N-(5-tert-butyl-3-(cyclopropylmethyl)-4-methyl...)
Affinity DataIC50: 16nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
Taisho Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50218272((Z)-N-(5-tert-butyl-3-(cyclopropylmethyl)-4-methyl...)
Affinity DataIC50: 65nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
Taisho Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50218271((Z)-N-(3-allyl-5-tert-butyl-4-methylthiazol-2(3H)-...)
Affinity DataIC50: 75nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
Taisho Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50218273((Z)-N-(5-tert-butyl-4-methyl-3-(3-methylbut-2-enyl...)
Affinity DataIC50: 170nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
Taisho Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50218274((Z)-N-(5-tert-butyl-4-methyl-3-(prop-2-ynyl)thiazo...)
Affinity DataIC50: 210nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
Taisho Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM5035(CHEMBL235747 | N-[(2Z)-5-tert-butyl-3,4-dimethyl-2...)
Affinity DataIC50: 340nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
Taisho Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50218275((Z)-N-(5-tert-butyl-3-(cyclopropylmethyl)-4-methyl...)
Affinity DataIC50: 490nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1(Human)
Taisho Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50218270((Z)-N-(5-tert-butyl-3-(cyclopropylmethyl)-4-methyl...)
Affinity DataIC50: 1.70E+3nMAssay Description:Displacement of [3H]CP-55940 from human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1(Human)
Taisho Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM5035(CHEMBL235747 | N-[(2Z)-5-tert-butyl-3,4-dimethyl-2...)
Affinity DataIC50: 5.00E+4nMAssay Description:Displacement of [3H]CP-55940 from human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed