Compile Data Set for Download or QSAR
Report error Found 28 Enz. Inhib. hit(s) with all data for entry = 50003842
TargetGlutamate receptor ionotropic, NMDA 1/2A(Human)
Chiba University

Curated by ChEMBL
LigandPNGBDBM50476423(CHEMBL228435)
Affinity DataIC50: 72nMAssay Description:Antagonist activity at recombinant NR1/NR2A receptor expressed in Xenopus laevis oocytesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1/2A(Human)
Chiba University

Curated by ChEMBL
LigandPNGBDBM50476427(CHEMBL228436)
Affinity DataIC50: 78nMAssay Description:Antagonist activity at recombinant NR1/NR2A receptor expressed in Xenopus laevis oocytesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1/2B(Human)
Chiba University

Curated by ChEMBL
LigandPNGBDBM50476433(CHEMBL228486)
Affinity DataIC50: 83nMAssay Description:Antagonist activity at recombinant NR1/NR2B receptor expressed in Xenopus laevis oocytesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1/2B(Human)
Chiba University

Curated by ChEMBL
LigandPNGBDBM50476427(CHEMBL228436)
Affinity DataIC50: 108nMAssay Description:Antagonist activity at recombinant NR1/NR2B receptor expressed in Xenopus laevis oocytesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1/2B(Human)
Chiba University

Curated by ChEMBL
LigandPNGBDBM50476432(CHEMBL228437)
Affinity DataIC50: 108nMAssay Description:Antagonist activity at recombinant NR1/NR2B receptor expressed in Xenopus laevis oocytesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1/2A(Human)
Chiba University

Curated by ChEMBL
LigandPNGBDBM50476430(CHEMBL388315)
Affinity DataIC50: 111nMAssay Description:Antagonist activity at recombinant NR1/NR2A receptor expressed in Xenopus laevis oocytesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1/2A(Human)
Chiba University

Curated by ChEMBL
LigandPNGBDBM50476424(CHEMBL228380)
Affinity DataIC50: 117nMAssay Description:Antagonist activity at recombinant NR1/NR2A receptor expressed in Xenopus laevis oocytesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1/2A(Human)
Chiba University

Curated by ChEMBL
LigandPNGBDBM50476432(CHEMBL228437)
Affinity DataIC50: 127nMAssay Description:Antagonist activity at recombinant NR1/NR2A receptor expressed in Xenopus laevis oocytesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1/2B(Human)
Chiba University

Curated by ChEMBL
LigandPNGBDBM50476423(CHEMBL228435)
Affinity DataIC50: 142nMAssay Description:Antagonist activity at recombinant NR1/NR2B receptor expressed in Xenopus laevis oocytesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1/2A(Human)
Chiba University

Curated by ChEMBL
LigandPNGBDBM50476433(CHEMBL228486)
Affinity DataIC50: 145nMAssay Description:Antagonist activity at recombinant NR1/NR2A receptor expressed in Xenopus laevis oocytesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1/2B(Human)
Chiba University

Curated by ChEMBL
LigandPNGBDBM50476430(CHEMBL388315)
Affinity DataIC50: 166nMAssay Description:Antagonist activity at recombinant NR1/NR2B receptor expressed in Xenopus laevis oocytesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1/2B(Human)
Chiba University

Curated by ChEMBL
LigandPNGBDBM50476431(CHEMBL390521)
Affinity DataIC50: 189nMAssay Description:Antagonist activity at recombinant NR1/NR2B receptor expressed in Xenopus laevis oocytesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1/2A(Human)
Chiba University

Curated by ChEMBL
LigandPNGBDBM50476425(CHEMBL228325)
Affinity DataIC50: 198nMAssay Description:Antagonist activity at recombinant NR1/NR2A receptor expressed in Xenopus laevis oocytesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1/2B(Human)
Chiba University

Curated by ChEMBL
LigandPNGBDBM50476422(CHEMBL390304)
Affinity DataIC50: 199nMAssay Description:Antagonist activity at recombinant NR1/NR2B receptor expressed in Xenopus laevis oocytesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1/2A(Human)
Chiba University

Curated by ChEMBL
LigandPNGBDBM50476422(CHEMBL390304)
Affinity DataIC50: 203nMAssay Description:Antagonist activity at recombinant NR1/NR2A receptor expressed in Xenopus laevis oocytesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1/2A(Human)
Chiba University

Curated by ChEMBL
LigandPNGBDBM50476431(CHEMBL390521)
Affinity DataIC50: 211nMAssay Description:Antagonist activity at recombinant NR1/NR2A receptor expressed in Xenopus laevis oocytesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1/2A(Human)
Chiba University

Curated by ChEMBL
LigandPNGBDBM50476426(CHEMBL390305)
Affinity DataIC50: 215nMAssay Description:Antagonist activity at recombinant NR1/NR2A receptor expressed in Xenopus laevis oocytesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1/2A(Human)
Chiba University

Curated by ChEMBL
LigandPNGBDBM50476421(CHEMBL228378)
Affinity DataIC50: 240nMAssay Description:Antagonist activity at recombinant NR1/NR2A receptor expressed in Xenopus laevis oocytesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1/2B(Human)
Chiba University

Curated by ChEMBL
LigandPNGBDBM50476424(CHEMBL228380)
Affinity DataIC50: 270nMAssay Description:Antagonist activity at recombinant NR1/NR2B receptor expressed in Xenopus laevis oocytesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1/2B(Human)
Chiba University

Curated by ChEMBL
LigandPNGBDBM50476421(CHEMBL228378)
Affinity DataIC50: 293nMAssay Description:Antagonist activity at recombinant NR1/NR2B receptor expressed in Xenopus laevis oocytesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1/2B(Human)
Chiba University

Curated by ChEMBL
LigandPNGBDBM50476425(CHEMBL228325)
Affinity DataIC50: 335nMAssay Description:Antagonist activity at recombinant NR1/NR2B receptor expressed in Xenopus laevis oocytesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1/2B(Human)
Chiba University

Curated by ChEMBL
LigandPNGBDBM50476426(CHEMBL390305)
Affinity DataIC50: 348nMAssay Description:Antagonist activity at recombinant NR1/NR2B receptor expressed in Xenopus laevis oocytesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1/2A(Human)
Chiba University

Curated by ChEMBL
LigandPNGBDBM50476428(CHEMBL228324)
Affinity DataIC50: 392nMAssay Description:Antagonist activity at recombinant NR1/NR2A receptor expressed in Xenopus laevis oocytesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1/2B(Human)
Chiba University

Curated by ChEMBL
LigandPNGBDBM50476429(CHEMBL228379)
Affinity DataIC50: 442nMAssay Description:Antagonist activity at recombinant NR1/NR2B receptor expressed in Xenopus laevis oocytesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1/2B(Human)
Chiba University

Curated by ChEMBL
LigandPNGBDBM50476428(CHEMBL228324)
Affinity DataIC50: 491nMAssay Description:Antagonist activity at recombinant NR1/NR2B receptor expressed in Xenopus laevis oocytesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1/2A(Human)
Chiba University

Curated by ChEMBL
LigandPNGBDBM50062599(CHEMBL807 | Namenda | 3,5-Dimethyl-adamantan-1-yla...)
Affinity DataIC50: 911nMAssay Description:Antagonist activity at recombinant NR1/NR2A receptor expressed in Xenopus laevis oocytesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1/2A(Human)
Chiba University

Curated by ChEMBL
LigandPNGBDBM50476429(CHEMBL228379)
Affinity DataIC50: 958nMAssay Description:Antagonist activity at recombinant NR1/NR2A receptor expressed in Xenopus laevis oocytesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1/2B(Human)
Chiba University

Curated by ChEMBL
LigandPNGBDBM50062599(CHEMBL807 | Namenda | 3,5-Dimethyl-adamantan-1-yla...)
Affinity DataIC50: 1.02E+3nMAssay Description:Antagonist activity at recombinant NR1/NR2B receptor expressed in Xenopus laevis oocytesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed