Compile Data Set for Download or QSAR
Report error Found 33 Enz. Inhib. hit(s) with all data for entry = 3048
TargetOxysterols receptor LXR-alpha(Human)
Tanabe Research Laboratories Usa

LigandPNGBDBM27264(tert-butyl 2-[4-(2-cyanoethyl)phenyl]-1H-indole-1-...)
Affinity DataEC50:  1.19E+3nMpH: 7.5 T: 2°CAssay Description:Polyhistidine-tagged human LXR ligand-binding domain was mixed with the test compound, biotin-SRC1 peptide, streptavidin-allophycocyanin, and europiu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/8/2009
Entry Details Article
PubMed
TargetOxysterols receptor LXR-beta(Human)
Tanabe Research Laboratories Usa

LigandPNGBDBM27268(tert-butyl 2-[4-(2-carbamoylethyl)phenyl]-1H-indol...)
Affinity DataEC50:  57nMpH: 7.5 T: 2°CAssay Description:Polyhistidine-tagged human LXR ligand-binding domain was mixed with the test compound, biotin-SRC1 peptide, streptavidin-allophycocyanin, and europiu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/8/2009
Entry Details Article
PubMed
TargetOxysterols receptor LXR-beta(Human)
Tanabe Research Laboratories Usa

LigandPNGBDBM27269(tert-butyl 2-{4-[(1E)-2-carbamoyleth-1-en-1-yl]phe...)
Affinity DataEC50:  4.90E+3nMpH: 7.5 T: 2°CAssay Description:Polyhistidine-tagged human LXR ligand-binding domain was mixed with the test compound, biotin-SRC1 peptide, streptavidin-allophycocyanin, and europiu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/8/2009
Entry Details Article
PubMed
TargetOxysterols receptor LXR-beta(Human)
Tanabe Research Laboratories Usa

LigandPNGBDBM27270(tert-butyl 2-{4-[2-(methylcarbamoyl)ethyl]phenyl}-...)
Affinity DataEC50:  490nMpH: 7.5 T: 2°CAssay Description:Polyhistidine-tagged human LXR ligand-binding domain was mixed with the test compound, biotin-SRC1 peptide, streptavidin-allophycocyanin, and europiu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/8/2009
Entry Details Article
PubMed
TargetOxysterols receptor LXR-beta(Human)
Tanabe Research Laboratories Usa

LigandPNGBDBM27271(tert-butyl 2-(4-{2-[(2-methylpropyl)carbamoyl]ethy...)
Affinity DataEC50:  1.51E+3nMpH: 7.5 T: 2°CAssay Description:Polyhistidine-tagged human LXR ligand-binding domain was mixed with the test compound, biotin-SRC1 peptide, streptavidin-allophycocyanin, and europiu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/8/2009
Entry Details Article
PubMed
TargetOxysterols receptor LXR-beta(Human)
Tanabe Research Laboratories Usa

LigandPNGBDBM27272(tert-butyl 2-{4-[2-(phenylcarbamoyl)ethyl]phenyl}-...)
Affinity DataEC50:  1.78E+3nMpH: 7.5 T: 2°CAssay Description:Polyhistidine-tagged human LXR ligand-binding domain was mixed with the test compound, biotin-SRC1 peptide, streptavidin-allophycocyanin, and europiu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/8/2009
Entry Details Article
PubMed
TargetOxysterols receptor LXR-beta(Human)
Tanabe Research Laboratories Usa

LigandPNGBDBM27273(3-[4-(1-benzoyl-1H-indol-2-yl)phenyl]propanenitril...)
Affinity DataEC50:  12nMpH: 7.5 T: 2°CAssay Description:Polyhistidine-tagged human LXR ligand-binding domain was mixed with the test compound, biotin-SRC1 peptide, streptavidin-allophycocyanin, and europiu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/8/2009
Entry Details Article
PubMed
TargetOxysterols receptor LXR-beta(Human)
Tanabe Research Laboratories Usa

LigandPNGBDBM27274(N-{2-[4-(1-benzoyl-1H-indol-2-yl)phenyl]ethyl}benz...)
Affinity DataEC50:  1.78E+3nMpH: 7.5 T: 2°CAssay Description:Polyhistidine-tagged human LXR ligand-binding domain was mixed with the test compound, biotin-SRC1 peptide, streptavidin-allophycocyanin, and europiu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/8/2009
Entry Details Article
PubMed
TargetOxysterols receptor LXR-alpha(Human)
Tanabe Research Laboratories Usa

LigandPNGBDBM27251(tert-butyl 2-(2-benzenesulfonamido-2,3-dihydro-1H-...)
Affinity DataEC50:  1.50E+3nMpH: 7.5 T: 2°CAssay Description:Polyhistidine-tagged human LXR ligand-binding domain was mixed with the test compound, biotin-SRC1 peptide, streptavidin-allophycocyanin, and europiu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/8/2009
Entry Details Article
PubMed
TargetOxysterols receptor LXR-beta(Human)
Tanabe Research Laboratories Usa

LigandPNGBDBM27267(3-(4-{1-[(tert-butoxy)carbonyl]-1H-indol-2-yl}phen...)
Affinity DataEC50:  220nMpH: 7.5 T: 2°CAssay Description:Polyhistidine-tagged human LXR ligand-binding domain was mixed with the test compound, biotin-SRC1 peptide, streptavidin-allophycocyanin, and europiu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/8/2009
Entry Details Article
PubMed
TargetOxysterols receptor LXR-alpha(Human)
Tanabe Research Laboratories Usa

LigandPNGBDBM27267(3-(4-{1-[(tert-butoxy)carbonyl]-1H-indol-2-yl}phen...)
Affinity DataEC50:  1.15E+3nMpH: 7.5 T: 2°CAssay Description:Polyhistidine-tagged human LXR ligand-binding domain was mixed with the test compound, biotin-SRC1 peptide, streptavidin-allophycocyanin, and europiu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/8/2009
Entry Details Article
PubMed
TargetOxysterols receptor LXR-alpha(Human)
Tanabe Research Laboratories Usa

LigandPNGBDBM27268(tert-butyl 2-[4-(2-carbamoylethyl)phenyl]-1H-indol...)
Affinity DataEC50:  1.11E+3nMpH: 7.5 T: 2°CAssay Description:Polyhistidine-tagged human LXR ligand-binding domain was mixed with the test compound, biotin-SRC1 peptide, streptavidin-allophycocyanin, and europiu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/8/2009
Entry Details Article
PubMed
TargetOxysterols receptor LXR-alpha(Human)
Tanabe Research Laboratories Usa

LigandPNGBDBM27273(3-[4-(1-benzoyl-1H-indol-2-yl)phenyl]propanenitril...)
Affinity DataEC50:  220nMpH: 7.5 T: 2°CAssay Description:Polyhistidine-tagged human LXR ligand-binding domain was mixed with the test compound, biotin-SRC1 peptide, streptavidin-allophycocyanin, and europiu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/8/2009
Entry Details Article
PubMed
TargetOxysterols receptor LXR-alpha(Human)
Tanabe Research Laboratories Usa

LigandPNGBDBM19992(2-{3-[3-({[2-chloro-3-(trifluoromethyl)phenyl]meth...)
Affinity DataEC50:  367nMAssay Description:Polyhistidine-tagged human LXR ligand-binding domain was mixed with the test compound, biotin-SRC1 peptide, streptavidin-allophycocyanin, and europiu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/8/2009
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetOxysterols receptor LXR-alpha(Human)
Tanabe Research Laboratories Usa

LigandPNGBDBM19993(CHEMBL62136 | [3H]T0901317 | T 0901317 | N-[4-(1,1...)
Affinity DataEC50:  40nMAssay Description:Polyhistidine-tagged human LXR ligand-binding domain was mixed with the test compound, biotin-SRC1 peptide, streptavidin-allophycocyanin, and europiu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/8/2009
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetOxysterols receptor LXR-beta(Human)
Tanabe Research Laboratories Usa

LigandPNGBDBM19992(2-{3-[3-({[2-chloro-3-(trifluoromethyl)phenyl]meth...)
Affinity DataEC50:  35nMAssay Description:Polyhistidine-tagged human LXR ligand-binding domain was mixed with the test compound, biotin-SRC1 peptide, streptavidin-allophycocyanin, and europiu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/8/2009
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetOxysterols receptor LXR-beta(Human)
Tanabe Research Laboratories Usa

LigandPNGBDBM19993(CHEMBL62136 | [3H]T0901317 | T 0901317 | N-[4-(1,1...)
Affinity DataEC50:  15nMAssay Description:Polyhistidine-tagged human LXR ligand-binding domain was mixed with the test compound, biotin-SRC1 peptide, streptavidin-allophycocyanin, and europiu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/8/2009
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetOxysterols receptor LXR-beta(Human)
Tanabe Research Laboratories Usa

LigandPNGBDBM27251(tert-butyl 2-(2-benzenesulfonamido-2,3-dihydro-1H-...)
Affinity DataEC50:  190nMpH: 7.5 T: 2°CAssay Description:Polyhistidine-tagged human LXR ligand-binding domain was mixed with the test compound, biotin-SRC1 peptide, streptavidin-allophycocyanin, and europiu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/8/2009
Entry Details Article
PubMed
TargetOxysterols receptor LXR-beta(Human)
Tanabe Research Laboratories Usa

LigandPNGBDBM27266(tert-butyl 2-[4-(2-hydroxyethoxy)phenyl]-1H-indole...)
Affinity DataEC50:  420nMpH: 7.5 T: 2°CAssay Description:Polyhistidine-tagged human LXR ligand-binding domain was mixed with the test compound, biotin-SRC1 peptide, streptavidin-allophycocyanin, and europiu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/8/2009
Entry Details Article
PubMed
TargetOxysterols receptor LXR-beta(Human)
Tanabe Research Laboratories Usa

LigandPNGBDBM27265(tert-butyl 2-[4-(3-hydroxypropyl)phenyl]-1H-indole...)
Affinity DataEC50:  380nMpH: 7.5 T: 2°CAssay Description:Polyhistidine-tagged human LXR ligand-binding domain was mixed with the test compound, biotin-SRC1 peptide, streptavidin-allophycocyanin, and europiu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/8/2009
Entry Details Article
PubMed
TargetOxysterols receptor LXR-beta(Human)
Tanabe Research Laboratories Usa

LigandPNGBDBM27264(tert-butyl 2-[4-(2-cyanoethyl)phenyl]-1H-indole-1-...)
Affinity DataEC50:  130nMpH: 7.5 T: 2°CAssay Description:Polyhistidine-tagged human LXR ligand-binding domain was mixed with the test compound, biotin-SRC1 peptide, streptavidin-allophycocyanin, and europiu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/8/2009
Entry Details Article
PubMed
TargetOxysterols receptor LXR-beta(Human)
Tanabe Research Laboratories Usa

LigandPNGBDBM27263(tert-butyl 2-[4-(cyanomethyl)phenyl]-1H-indole-1-c...)
Affinity DataEC50:  300nMpH: 7.5 T: 2°CAssay Description:Polyhistidine-tagged human LXR ligand-binding domain was mixed with the test compound, biotin-SRC1 peptide, streptavidin-allophycocyanin, and europiu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/8/2009
Entry Details Article
PubMed
TargetOxysterols receptor LXR-beta(Human)
Tanabe Research Laboratories Usa

LigandPNGBDBM27262(tert-butyl 2-[4-(aminomethyl)phenyl]-1H-indole-1-c...)
Affinity DataEC50:  5.60E+3nMpH: 7.5 T: 2°CAssay Description:Polyhistidine-tagged human LXR ligand-binding domain was mixed with the test compound, biotin-SRC1 peptide, streptavidin-allophycocyanin, and europiu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/8/2009
Entry Details Article
PubMed
TargetOxysterols receptor LXR-beta(Human)
Tanabe Research Laboratories Usa

LigandPNGBDBM27261(tert-butyl 2-{4-[3-(phenylformamido)propyl]phenyl}...)
Affinity DataEC50:  360nMpH: 7.5 T: 2°CAssay Description:Polyhistidine-tagged human LXR ligand-binding domain was mixed with the test compound, biotin-SRC1 peptide, streptavidin-allophycocyanin, and europiu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/8/2009
Entry Details Article
PubMed
TargetOxysterols receptor LXR-beta(Human)
Tanabe Research Laboratories Usa

LigandPNGBDBM27260(tert-butyl 2-{4-[2-(phenylformamido)ethyl]phenyl}-...)
Affinity DataEC50:  1.75E+3nMpH: 7.5 T: 2°CAssay Description:Polyhistidine-tagged human LXR ligand-binding domain was mixed with the test compound, biotin-SRC1 peptide, streptavidin-allophycocyanin, and europiu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/8/2009
Entry Details Article
PubMed
TargetOxysterols receptor LXR-beta(Human)
Tanabe Research Laboratories Usa

LigandPNGBDBM27259(tert-butyl 2-{4-[(phenylformamido)methyl]phenyl}-1...)
Affinity DataEC50:  1.80E+3nMpH: 7.5 T: 2°CAssay Description:Polyhistidine-tagged human LXR ligand-binding domain was mixed with the test compound, biotin-SRC1 peptide, streptavidin-allophycocyanin, and europiu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/8/2009
Entry Details Article
PubMed
TargetOxysterols receptor LXR-beta(Human)
Tanabe Research Laboratories Usa

LigandPNGBDBM27258(tert-butyl 2-[4-(2-{[5-(pyridin-2-yl)thiophene-2-]...)
Affinity DataEC50:  230nMpH: 7.5 T: 2°CAssay Description:Polyhistidine-tagged human LXR ligand-binding domain was mixed with the test compound, biotin-SRC1 peptide, streptavidin-allophycocyanin, and europiu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/8/2009
Entry Details Article
PubMed
TargetOxysterols receptor LXR-beta(Human)
Tanabe Research Laboratories Usa

LigandPNGBDBM27257(tert-butyl 2-{4-[2-(thiophene-2-sulfonamido)ethyl]...)
Affinity DataEC50:  58nMpH: 7.5 T: 2°CAssay Description:Polyhistidine-tagged human LXR ligand-binding domain was mixed with the test compound, biotin-SRC1 peptide, streptavidin-allophycocyanin, and europiu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/8/2009
Entry Details Article
PubMed
TargetOxysterols receptor LXR-beta(Human)
Tanabe Research Laboratories Usa

LigandPNGBDBM27256(tert-butyl 2-(4-benzenesulfonamidophenyl)-1H-indol...)
Affinity DataEC50:  1.32E+3nMpH: 7.5 T: 2°CAssay Description:Polyhistidine-tagged human LXR ligand-binding domain was mixed with the test compound, biotin-SRC1 peptide, streptavidin-allophycocyanin, and europiu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/8/2009
Entry Details Article
PubMed
TargetOxysterols receptor LXR-beta(Human)
Tanabe Research Laboratories Usa

LigandPNGBDBM27255(tert-butyl 2-[4-(3-benzenesulfonamidopropyl)phenyl...)
Affinity DataEC50:  350nMpH: 7.5 T: 2°CAssay Description:Polyhistidine-tagged human LXR ligand-binding domain was mixed with the test compound, biotin-SRC1 peptide, streptavidin-allophycocyanin, and europiu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/8/2009
Entry Details Article
PubMed
TargetOxysterols receptor LXR-beta(Human)
Tanabe Research Laboratories Usa

LigandPNGBDBM27254(tert-butyl 2-[4-(benzenesulfonamidomethyl)phenyl]-...)
Affinity DataEC50:  220nMpH: 7.5 T: 2°CAssay Description:Polyhistidine-tagged human LXR ligand-binding domain was mixed with the test compound, biotin-SRC1 peptide, streptavidin-allophycocyanin, and europiu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/8/2009
Entry Details Article
PubMed
TargetOxysterols receptor LXR-beta(Human)
Tanabe Research Laboratories Usa

LigandPNGBDBM27253(tert-butyl 2-[4-(2-benzenesulfonamidoethyl)phenyl]...)
Affinity DataEC50:  120nMpH: 7.5 T: 2°CAssay Description:Polyhistidine-tagged human LXR ligand-binding domain was mixed with the test compound, biotin-SRC1 peptide, streptavidin-allophycocyanin, and europiu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/8/2009
Entry Details Article
PubMed
TargetOxysterols receptor LXR-beta(Human)
Tanabe Research Laboratories Usa

LigandPNGBDBM27252(tert-butyl 2-[3-(2-benzenesulfonamidoethyl)phenyl]...)
Affinity DataEC50:  420nMpH: 7.5 T: 2°CAssay Description:Polyhistidine-tagged human LXR ligand-binding domain was mixed with the test compound, biotin-SRC1 peptide, streptavidin-allophycocyanin, and europiu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/8/2009
Entry Details Article
PubMed