Compile Data Set for Download or QSAR
Report error Found 64 Enz. Inhib. hit(s) with all data for entry = 50020613
TargetMAP kinase-activated protein kinase 2(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50215481(5-methoxy-9,12-diazatetracyclo[10.2.1.0^{2,10}.0^{...)
Affinity DataIC50: 290nMAssay Description:Inhibition of MK2More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMAP kinase-activated protein kinase 2(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50215517(6-methoxy-2-methyl-2,3,4,9-tetrahydro-1H-pyrido[3,...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of MK2More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMAP kinase-activated protein kinase 2(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50215501(6-(2-oxo-2-phenyl-ethoxy)-2,3,4,9-tetrahydro-1H-be...)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of MK2More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMAP kinase-activated protein kinase 2(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50215503(4-ethyl-6-methoxy-2,3,4,9-tetrahydro-1H-pyrido[3,4...)
Affinity DataIC50: 2.20E+3nMAssay Description:Inhibition of MK2More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMAP kinase-activated protein kinase 2(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50215502(6-methoxy-4-methyl-2,3,4,9-tetrahydro-1H-pyrido[3,...)
Affinity DataIC50: 2.20E+3nMAssay Description:Inhibition of MK2More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMAP kinase-activated protein kinase 2(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50215483(6-methoxy-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indol...)
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition of MK2More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMAP kinase-activated protein kinase 2(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50215510(3-(hydroxymethyl)-6-methoxy-2,3,4,9-tetrahydro-1H-...)
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of MK2More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMAP kinase-activated protein kinase 2(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50215506(prop-2-en-1-yl 5-methoxy-9,12-diazatetracyclo[10.2...)
Affinity DataIC50: 3.27E+3nMAssay Description:Inhibition of MK2More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMAP kinase-activated protein kinase 2(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50215489(6-hydroxy-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indol...)
Affinity DataIC50: 4.50E+3nMAssay Description:Inhibition of MK2More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMAP kinase-activated protein kinase 2(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50215497(5-methoxy-9,12-diazatetracyclo[10.3.1.0^{2,10}.0^{...)
Affinity DataIC50: 5.10E+3nMAssay Description:Inhibition of MK2More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMAP kinase-activated protein kinase 2(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50215508(2-ethyl-6-methoxy-2,3,4,9-tetrahydro-1H-pyrido[3,4...)
Affinity DataIC50: 5.80E+3nMAssay Description:Inhibition of MK2More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMAP kinase-activated protein kinase 2(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50215523(3-(aminomethyl)-6-methoxy-2,3,4,9-tetrahydro-1H-py...)
Affinity DataIC50: 5.90E+3nMAssay Description:Inhibition of MK2More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMAP kinase-activated protein kinase 2(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50215520(6-(methoxycarbonyl)-2,3,4,9-tetrahydro-1H-pyrido[3...)
Affinity DataIC50: 6.60E+3nMAssay Description:Inhibition of MK2More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMAP kinase-activated protein kinase 2(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50215485(benzyl 5-methoxy-9,12-diazatetracyclo[10.2.1.0^{2,...)
Affinity DataIC50: 7.09E+3nMAssay Description:Inhibition of MK2More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMAP kinase-activated protein kinase 2(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50215482(6-methoxy-3-methyl-2,3,4,9-tetrahydro-1H-pyrido[3,...)
Affinity DataIC50: 7.10E+3nMAssay Description:Inhibition of MK2More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMAP kinase-activated protein kinase 2(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50215504(propyl 5-methoxy-9,12-diazatetracyclo[10.2.1.0^{2,...)
Affinity DataIC50: 1.01E+4nMAssay Description:Inhibition of MK2More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMAP kinase-activated protein kinase 2(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50215513(6-(benzyloxy)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]i...)
Affinity DataIC50: 1.20E+4nMAssay Description:Inhibition of MK2More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMAP kinase-activated protein kinase 2(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50215488(1-phenylethyl 5-methoxy-9,12-diazatetracyclo[10.2....)
Affinity DataIC50: 1.30E+4nMAssay Description:Inhibition of MK2More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMAP kinase-activated protein kinase 2(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50215524(4-benzyl-6-methoxy-2,3,4,9-tetrahydro-1H-pyrido[3,...)
Affinity DataIC50: 1.60E+4nMAssay Description:Inhibition of MK2More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMAP kinase-activated protein kinase 2(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50215511(6-chloro-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole...)
Affinity DataIC50: 1.90E+4nMAssay Description:Inhibition of MK2More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMAP kinase-activated protein kinase 5(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50215483(6-methoxy-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indol...)
Affinity DataIC50: 1.90E+4nMAssay Description:Inhibition of PRAKMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMAP kinase-activated protein kinase 5(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50215481(5-methoxy-9,12-diazatetracyclo[10.2.1.0^{2,10}.0^{...)
Affinity DataIC50: 2.40E+4nMAssay Description:Inhibition of PRAKMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMAP kinase-activated protein kinase 5(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50215497(5-methoxy-9,12-diazatetracyclo[10.3.1.0^{2,10}.0^{...)
Affinity DataIC50: 2.50E+4nMAssay Description:Inhibition of PRAKMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMAP kinase-activated protein kinase 2(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50215512(6-fluoro-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole...)
Affinity DataIC50: 2.60E+4nMAssay Description:Inhibition of MK2More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMAP kinase-activated protein kinase 2(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50215491(6-carbamoyl-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]ind...)
Affinity DataIC50: 2.80E+4nMAssay Description:Inhibition of MK2More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMAP kinase-activated protein kinase 2(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50215492(ethyl 5-methoxy-9,12-diazatetracyclo[10.2.1.0^{2,1...)
Affinity DataIC50: 2.93E+4nMAssay Description:Inhibition of MK2More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMAP kinase-activated protein kinase 2(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50215522(5-methoxy-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indol...)
Affinity DataIC50: 4.20E+4nMAssay Description:Inhibition of MK2More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMAP kinase-activated protein kinase 2(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50215498(methyl 6-methoxy-2,3,4,9-tetrahydro-1H-pyrido[3,4-...)
Affinity DataIC50: 4.70E+4nMAssay Description:Inhibition of MK2More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMAP kinase-activated protein kinase 2(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50215525(7-hydroxy-6-methoxy-2,3,4,9-tetrahydro-1H-pyrido[3...)
Affinity DataIC50: 5.30E+4nMAssay Description:Inhibition of MK2More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMAP kinase-activated protein kinase 2(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50215528(3-ethyl-6-methoxy-2,3,4,9-tetrahydro-1H-pyrido[3,4...)
Affinity DataIC50: 6.40E+4nMAssay Description:Inhibition of MK2More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMAP kinase-activated protein kinase 2(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50215516(2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-1-carbox...)
Affinity DataIC50: 8.70E+4nMAssay Description:Inhibition of MK2More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMAP kinase-activated protein kinase 2(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50215499(N-hydroxy-6-methoxy-2,3,4,9-tetrahydro-1H-pyrido[3...)
Affinity DataIC50: 8.80E+4nMAssay Description:Inhibition of MK2More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMAP kinase-activated protein kinase 3(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50215481(5-methoxy-9,12-diazatetracyclo[10.2.1.0^{2,10}.0^{...)
Affinity DataIC50: 9.00E+4nMAssay Description:Inhibition of MK3More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50215481(5-methoxy-9,12-diazatetracyclo[10.2.1.0^{2,10}.0^{...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMitogen-activated protein kinase 1(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50215483(6-methoxy-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indol...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of ERK2More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50215483(6-methoxy-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indol...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMAP kinase-activated protein kinase 2(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50215521(6-methoxy-1-(2H-tetrazol-5-yl)-2,3,4,9-tetrahydro-...)
Affinity DataIC50: 1.30E+5nMAssay Description:Inhibition of MK2More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMAP kinase-activated protein kinase 2(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50215484(2-benzyl-6-methoxy-2,3,4,9-tetrahydro-1H-pyrido[3,...)
Affinity DataIC50: 1.30E+5nMAssay Description:Inhibition of MK2More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMAP kinase-activated protein kinase 3(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50215497(5-methoxy-9,12-diazatetracyclo[10.3.1.0^{2,10}.0^{...)
Affinity DataIC50: 1.60E+5nMAssay Description:Inhibition of MK3More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMAP kinase-activated protein kinase 2(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50215527(2-isopropyl-6-methoxy-2,3,4,9-tetrahydro-1H-pyrido...)
Affinity DataIC50: 1.70E+5nMAssay Description:Inhibition of MK2More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMAP kinase-activated protein kinase 2(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50215515(6-acetoxy-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indol...)
Affinity DataIC50: 1.70E+5nMAssay Description:Inhibition of MK2More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMAP kinase-activated protein kinase 2(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50215509(6-methoxy-1,3,4,9-tetrahydropyrano[3,4-b]indole-1-...)
Affinity DataIC50: 2.00E+5nMAssay Description:Inhibition of MK2More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRibosomal protein S6 kinase alpha-5(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50215481(5-methoxy-9,12-diazatetracyclo[10.2.1.0^{2,10}.0^{...)
Affinity DataIC50: 2.00E+5nMAssay Description:Inhibition of MSK1More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMitogen-activated protein kinase 9(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50215483(6-methoxy-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indol...)
Affinity DataIC50: 2.00E+5nMAssay Description:Inhibition of JNK2More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMitogen-activated protein kinase 9(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50215481(5-methoxy-9,12-diazatetracyclo[10.2.1.0^{2,10}.0^{...)
Affinity DataIC50: 2.00E+5nMAssay Description:Inhibition of JNK2More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMAP kinase-activated protein kinase 2(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50215526(6-methoxy-1-methyl-2,3,4,9-tetrahydro-1H-pyrido[3,...)
Affinity DataIC50: 2.00E+5nMAssay Description:Inhibition of MK2More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMAP kinase-activated protein kinase 2(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50215486((6-methoxy-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indo...)
Affinity DataIC50: 2.00E+5nMAssay Description:Inhibition of MK2More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRibosomal protein S6 kinase alpha-5(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50215483(6-methoxy-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indol...)
Affinity DataIC50: 2.00E+5nMAssay Description:Inhibition of MSK1More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMAP kinase-activated protein kinase 2(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50215495(6-methoxy-3-(trifluoromethyl)-2,3,4,9-tetrahydro-1...)
Affinity DataIC50: 2.00E+5nMAssay Description:Inhibition of MK2More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMAP kinase-activated protein kinase 2(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50215518(methyl 6-methoxy-9H-pyrido[3,4-b]indole-1-carboxyl...)
Affinity DataIC50: 2.00E+5nMAssay Description:Inhibition of MK2More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
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