Compile Data Set for Download or QSAR
Report error Found 66 Enz. Inhib. hit(s) with all data for entry = 50020362
TargetFatty acid-binding protein, adipocyte(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM60927(ANS | BDBM50126831 | 1-anilinonaphthalene-8-sulfon...)
Affinity DataKd:  150nMAssay Description:Binding affinity to aFABPMore data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
TargetFatty acid-binding protein, adipocyte(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50212876(2,3-bis[(2,4-dichlorobenzyl)oxy]benzoic acid | CHE...)
Affinity DataKd:  21nMAssay Description:Binding affinity to aFABPMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetFatty acid-binding protein 5(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50212876(2,3-bis[(2,4-dichlorobenzyl)oxy]benzoic acid | CHE...)
Affinity DataKi:  2nMAssay Description:Displacement of 1,8-ANS from eFABP by fluorescence based-assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetFatty acid-binding protein, adipocyte(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50212876(2,3-bis[(2,4-dichlorobenzyl)oxy]benzoic acid | CHE...)
Affinity DataKi:  2nMAssay Description:Displacement of 1,8-ANS from aFABP by fluorescence based-assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetFatty acid-binding protein, adipocyte(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50212885([2'-(1-methyl-4,5-diphenyl-1H-imidazol-2-yl)-biphe...)
Affinity DataKi:  2.70nMAssay Description:Displacement of 1,8-ANS from aFABP by fluorescence based-assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetFatty acid-binding protein, adipocyte(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50212884([2'-(1-ethyl-4,5-diphenyl-1H-imidazol-2-yl)-biphen...)
Affinity DataKi:  3.30nMAssay Description:Displacement of [3H]2,3-bis[(2,4-dichlorobenzyl)oxy]benzoic acid from aFABPMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetFatty acid-binding protein, adipocyte(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50212877([2'-(1-ethyl-4,5-diphenyl-1H-imidazol-2-yl)-biphen...)
Affinity DataKi:  3.40nMAssay Description:Displacement of 1,8-ANS from aFABP by fluorescence based-assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetFatty acid-binding protein, adipocyte(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50212886([2'-(3-ethyl-4,5-diphenyl-furan-2-yl)-biphenyl-3-y...)
Affinity DataKi:  3.5nMAssay Description:Displacement of 1,8-ANS from aFABP by fluorescence based-assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetFatty acid-binding protein, heart(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50212876(2,3-bis[(2,4-dichlorobenzyl)oxy]benzoic acid | CHE...)
Affinity DataKi:  4nMAssay Description:Displacement of 1,8-ANS from mFABP by fluorescence based-assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetFatty acid-binding protein, adipocyte(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50029969([2'-(4,5-Diphenyl-oxazol-2-yl)-biphenyl-3-yloxy]-a...)
Affinity DataKi:  6nMAssay Description:Displacement of 1,8-ANS from aFABP by fluorescence based-assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetFatty acid-binding protein, adipocyte(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50212873(((2'-(5-ETHYL-3,4-DIPHENYL-1H-PYRAZOL-1-YL)-3-BIPH...)
Affinity DataKi:  7.40nMAssay Description:Displacement of [3H]2,3-bis[(2,4-dichlorobenzyl)oxy]benzoic acid from aFABPMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetFatty acid-binding protein, adipocyte(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50212883({2'-[1-(2-fluoro-ethyl)-4,5-diphenyl-1H-imidazol-2...)
Affinity DataKi:  8.70nMAssay Description:Displacement of [3H]2,3-bis[(2,4-dichlorobenzyl)oxy]benzoic acid from aFABPMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetFatty acid-binding protein, adipocyte(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50212879([2'-(4,5-diphenyl-1H-imidazol-2-yl)-biphenyl-3-ylo...)
Affinity DataKi:  9.30nMAssay Description:Displacement of 1,8-ANS from aFABP by fluorescence based-assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetFatty acid-binding protein, adipocyte(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50212887([2'-(4,5-diphenyl-1H-pyrrol-2-yl)-biphenyl-3-yloxy...)
Affinity DataKi:  12nMAssay Description:Displacement of 1,8-ANS from aFABP by fluorescence based-assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetFatty acid-binding protein, adipocyte(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50212877([2'-(1-ethyl-4,5-diphenyl-1H-imidazol-2-yl)-biphen...)
Affinity DataKi:  13nMAssay Description:Displacement of [3H]2,3-bis[(2,4-dichlorobenzyl)oxy]benzoic acid from aFABPMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetFatty acid-binding protein, adipocyte(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50212881([2'-(1-methyl-4,5-diphenyl-1H-imidazol-2-yl)-biphe...)
Affinity DataKi:  13nMAssay Description:Displacement of [3H]2,3-bis[(2,4-dichlorobenzyl)oxy]benzoic acid from aFABPMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetFatty acid-binding protein, adipocyte(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50212874([2'-(4,5-diphenyl-1H-imidazol-2-yl)-biphenyl-3-yla...)
Affinity DataKi:  18nMAssay Description:Displacement of 1,8-ANS from aFABP by fluorescence based-assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetFatty acid-binding protein, adipocyte(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50212882([2'-(5-ethyl-3,4-diphenyl-pyrazol-1-yl)-biphenyl-3...)
Affinity DataKi:  28nMAssay Description:Displacement of 1,8-ANS from aFABP by fluorescence based-assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetFatty acid-binding protein, adipocyte(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50212886([2'-(3-ethyl-4,5-diphenyl-furan-2-yl)-biphenyl-3-y...)
Affinity DataKi:  32nMAssay Description:Displacement of [3H]2,3-bis[(2,4-dichlorobenzyl)oxy]benzoic acid from aFABPMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetFatty acid-binding protein, heart(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50002838(5-[2-(4,5-Diphenyl-oxazol-2-yl)-phenoxy]-pentanoic...)
Affinity DataKi:  32nMAssay Description:Displacement of 1,8-ANS from mFABP by fluorescence based-assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetFatty acid-binding protein, adipocyte(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50212878([2'-(4,5-diphenyl-furan-2-yl)-biphenyl-3-yloxy]-ac...)
Affinity DataKi:  36nMAssay Description:Displacement of 1,8-ANS from aFABP by fluorescence based-assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetFatty acid-binding protein, adipocyte(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50212885([2'-(1-methyl-4,5-diphenyl-1H-imidazol-2-yl)-biphe...)
Affinity DataKi:  48nMAssay Description:Displacement of [3H]2,3-bis[(2,4-dichlorobenzyl)oxy]benzoic acid from aFABPMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetFatty acid-binding protein, adipocyte(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50002838(5-[2-(4,5-Diphenyl-oxazol-2-yl)-phenoxy]-pentanoic...)
Affinity DataKi:  58nMAssay Description:Displacement of 1,8-ANS from aFABP by fluorescence based-assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetFatty acid-binding protein, adipocyte(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50029969([2'-(4,5-Diphenyl-oxazol-2-yl)-biphenyl-3-yloxy]-a...)
Affinity DataKi:  95nMAssay Description:Displacement of [3H]2,3-bis[(2,4-dichlorobenzyl)oxy]benzoic acid from aFABPMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetFatty acid-binding protein, heart(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50212875(2'-(5-ethyl-3,4-diphenyl-pyrazol-1-yl)-biphenyl-3-...)
Affinity DataKi:  110nMAssay Description:Displacement of 1,8-ANS from mFABP by fluorescence based-assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetFatty acid-binding protein, adipocyte(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50212880([2'-(1-isobutyl-4,5-diphenyl-1H-imidazol-2-yl)-bip...)
Affinity DataKi:  130nMAssay Description:Displacement of 1,8-ANS from aFABP by fluorescence based-assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetFatty acid-binding protein, adipocyte(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50150484(CHEMBL8659 | oleaic acid | Octadec-9-enoic acid | ...)
Affinity DataKi:  185nMAssay Description:Displacement of 1,8-ANS from aFABP by fluorescence based-assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
TargetFatty acid-binding protein, heart(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50212886([2'-(3-ethyl-4,5-diphenyl-furan-2-yl)-biphenyl-3-y...)
Affinity DataKi:  220nMAssay Description:Displacement of 1,8-ANS from mFABP by fluorescence based-assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetFatty acid-binding protein 5(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50212875(2'-(5-ethyl-3,4-diphenyl-pyrazol-1-yl)-biphenyl-3-...)
Affinity DataKi:  240nMAssay Description:Displacement of 1,8-ANS from eFABP by fluorescence based-assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetFatty acid-binding protein 5(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50150484(CHEMBL8659 | oleaic acid | Octadec-9-enoic acid | ...)
Affinity DataKi:  248nMAssay Description:Displacement of 1,8-ANS from eFABP by fluorescence based-assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetFatty acid-binding protein, heart(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50212873(((2'-(5-ETHYL-3,4-DIPHENYL-1H-PYRAZOL-1-YL)-3-BIPH...)
Affinity DataKi:  250nMAssay Description:Displacement of 1,8-ANS from mFABP by fluorescence based-assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetFatty acid-binding protein 5(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50212886([2'-(3-ethyl-4,5-diphenyl-furan-2-yl)-biphenyl-3-y...)
Affinity DataKi:  290nMAssay Description:Displacement of 1,8-ANS from eFABP by fluorescence based-assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetFatty acid-binding protein, adipocyte(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50212874([2'-(4,5-diphenyl-1H-imidazol-2-yl)-biphenyl-3-yla...)
Affinity DataKi:  300nMAssay Description:Displacement of [3H]2,3-bis[(2,4-dichlorobenzyl)oxy]benzoic acid from aFABPMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetFatty acid-binding protein, adipocyte(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50152850(1-HEXYLDECANOIC ACID | Hexadecanoic acid anion | H...)
Affinity DataKi:  336nMAssay Description:Displacement of 1,8-ANS from aFABP by fluorescence based-assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetFatty acid-binding protein 5(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50212873(((2'-(5-ETHYL-3,4-DIPHENYL-1H-PYRAZOL-1-YL)-3-BIPH...)
Affinity DataKi:  350nMAssay Description:Displacement of 1,8-ANS from eFABP by fluorescence based-assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetFatty acid-binding protein, heart(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50212882([2'-(5-ethyl-3,4-diphenyl-pyrazol-1-yl)-biphenyl-3...)
Affinity DataKi:  360nMAssay Description:Displacement of 1,8-ANS from mFABP by fluorescence based-assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetFatty acid-binding protein 5(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50212882([2'-(5-ethyl-3,4-diphenyl-pyrazol-1-yl)-biphenyl-3...)
Affinity DataKi:  550nMAssay Description:Displacement of 1,8-ANS from eFABP by fluorescence based-assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetFatty acid-binding protein, adipocyte(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50212875(2'-(5-ethyl-3,4-diphenyl-pyrazol-1-yl)-biphenyl-3-...)
Affinity DataKi:  650nMAssay Description:Displacement of 1,8-ANS from aFABP by fluorescence based-assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetFatty acid-binding protein 5(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50152850(1-HEXYLDECANOIC ACID | Hexadecanoic acid anion | H...)
Affinity DataKi:  802nMAssay Description:Displacement of 1,8-ANS from eFABP by fluorescence based-assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetFatty acid-binding protein 5(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50212884([2'-(1-ethyl-4,5-diphenyl-1H-imidazol-2-yl)-biphen...)
Affinity DataKi:  830nMAssay Description:Displacement of 1,8-ANS from eFABP by fluorescence based-assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetFatty acid-binding protein 5(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50212881([2'-(1-methyl-4,5-diphenyl-1H-imidazol-2-yl)-biphe...)
Affinity DataKi:  830nMAssay Description:Displacement of 1,8-ANS from eFABP by fluorescence based-assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetFatty acid-binding protein, heart(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50212881([2'-(1-methyl-4,5-diphenyl-1H-imidazol-2-yl)-biphe...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of 1,8-ANS from mFABP by fluorescence based-assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetFatty acid-binding protein, heart(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50212874([2'-(4,5-diphenyl-1H-imidazol-2-yl)-biphenyl-3-yla...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of 1,8-ANS from mFABP by fluorescence based-assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetFatty acid-binding protein, heart(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50212878([2'-(4,5-diphenyl-furan-2-yl)-biphenyl-3-yloxy]-ac...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of 1,8-ANS from mFABP by fluorescence based-assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetFatty acid-binding protein, heart(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50212887([2'-(4,5-diphenyl-1H-pyrrol-2-yl)-biphenyl-3-yloxy...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of 1,8-ANS from mFABP by fluorescence based-assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetFatty acid-binding protein, heart(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50212884([2'-(1-ethyl-4,5-diphenyl-1H-imidazol-2-yl)-biphen...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of 1,8-ANS from mFABP by fluorescence based-assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetFatty acid-binding protein, heart(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50212885([2'-(1-methyl-4,5-diphenyl-1H-imidazol-2-yl)-biphe...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of 1,8-ANS from mFABP by fluorescence based-assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetFatty acid-binding protein, heart(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50212879([2'-(4,5-diphenyl-1H-imidazol-2-yl)-biphenyl-3-ylo...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of 1,8-ANS from mFABP by fluorescence based-assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetFatty acid-binding protein, heart(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50212877([2'-(1-ethyl-4,5-diphenyl-1H-imidazol-2-yl)-biphen...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of 1,8-ANS from mFABP by fluorescence based-assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetFatty acid-binding protein, heart(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50212872([2'-(1-carboxymethyl-4,5-diphenyl-1H-imidazol-2-yl...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of 1,8-ANS from mFABP by fluorescence based-assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
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