Compile Data Set for Download or QSAR
Report error Found 11 Enz. Inhib. hit(s) with all data for entry = 50037944
TargetSodium-dependent dopamine transporter(Rat)
University of Sassari

Curated by ChEMBL
LigandPNGBDBM50094751(3-{2-[Bis-(4-fluoro-phenyl)-methoxy]-ethyl}-8-(1H-...)
Affinity DataIC50: 40nMAssay Description:Inhibition of [3H]dopamine uptake at DAT in Sprague-Dawley rat striatum synaptosomeMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
University of Sassari

Curated by ChEMBL
LigandPNGBDBM50209498(3-{2-[bis-(4-fluorophenyl)methoxy]ethyl}-6-[(1Hind...)
Affinity DataKi:  5.5nMAssay Description:Inhibition of [3H]dopamine uptake at DAT in Sprague-Dawley rat striatum synaptosomeMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
University of Sassari

Curated by ChEMBL
LigandPNGBDBM50209493(3-{2-[bis-(4-fluorophenyl)methoxy]ethyl}-6-[3-(2-m...)
Affinity DataKi:  6.30nMAssay Description:Inhibition of [3H]dopamine uptake at DAT in Sprague-Dawley rat striatum synaptosomeMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
University of Sassari

Curated by ChEMBL
LigandPNGBDBM50209495(3-{2-[bis-(4-fluorophenyl)methoxy]ethyl}-6-[(1Hind...)
Affinity DataKi:  6.5nMAssay Description:Inhibition of [3H]dopamine uptake at DAT in Sprague-Dawley rat striatum synaptosomeMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
University of Sassari

Curated by ChEMBL
LigandPNGBDBM50209497(3-{2-[bis-(4-fluorophenyl)methoxy]ethyl}-6-[(E)-3-...)
Affinity DataKi:  8.80nMAssay Description:Inhibition of [3H]dopamine uptake at DAT in Sprague-Dawley rat striatum synaptosomeMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
University of Sassari

Curated by ChEMBL
LigandPNGBDBM50209491(3-{2-[bis-(4-fluorophenyl)methoxy]ethyl}-6-cinnamy...)
Affinity DataKi:  9.10nMAssay Description:Inhibition of [3H]dopamine uptake at DAT in Sprague-Dawley rat striatum synaptosomeMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
University of Sassari

Curated by ChEMBL
LigandPNGBDBM50209490(3-{2-[bis-(4-fluorophenyl)methoxy]ethyl}-6-[(E)-3-...)
Affinity DataKi:  13nMAssay Description:Inhibition of [3H]dopamine uptake at DAT in Sprague-Dawley rat striatum synaptosomeMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
University of Sassari

Curated by ChEMBL
LigandPNGBDBM50209496(6-[(benzo[b]thiophen-2-yl)methyl]-3-{2-[bis-(4-flu...)
Affinity DataKi:  35nMAssay Description:Inhibition of [3H]dopamine uptake at DAT in Sprague-Dawley rat striatum synaptosomeMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
University of Sassari

Curated by ChEMBL
LigandPNGBDBM50209494(6-[(benzofuran-2-yl)methyl]-3-{2-[bis-(4-fluorophe...)
Affinity DataKi:  38nMAssay Description:Inhibition of [3H]dopamine uptake at DAT in Sprague-Dawley rat striatum synaptosomeMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
University of Sassari

Curated by ChEMBL
LigandPNGBDBM50209492(3-{2-[bis-(4-fluorophenyl)methoxy]ethyl}-6-[(E)-3-...)
Affinity DataKi:  46nMAssay Description:Inhibition of [3H]dopamine uptake at DAT in Sprague-Dawley rat striatum synaptosomeMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
University of Sassari

Curated by ChEMBL
LigandPNGBDBM50084717(CHEMBL120901 | 3-Naphthalen-2-yl-8-oxa-bicyclo[3.2...)
Affinity DataKi:  111nMAssay Description:Inhibition of [3H]dopamine uptake at DAT in Sprague-Dawley rat striatum synaptosomeMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed