Compile Data Set for Download or QSAR
Report error Found 13 Enz. Inhib. hit(s) with all data for entry = 50019635
TargetCytosolic phospholipase A2(Human)
University of MüNster

Curated by ChEMBL
LigandPNGBDBM50185348(3-methylhydrogen 1-[3-(4-octylphenoxy)-2-oxopropyl...)
Affinity DataIC50: 5nMAssay Description:Inhibition of human platelet cPLA2-alpha assessed as arachidonic acid release by vesicle assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCytosolic phospholipase A2(Human)
University of MüNster

Curated by ChEMBL
LigandPNGBDBM50110846(4-[3-(4-Decyloxy-phenoxy)-2-oxo-propoxy]-benzoic a...)
Affinity DataIC50: 11nMAssay Description:Inhibition of human platelet cPLA2-alpha assessed as arachidonic acid release by vesicle assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCytosolic phospholipase A2(Human)
University of MüNster

Curated by ChEMBL
LigandPNGBDBM50185356(1-(3-(4-octylphenoxy)-2-oxopropyl)-1H-indole-5-car...)
Affinity DataIC50: 35nMAssay Description:Inhibition of human platelet cPLA2-alpha assessed as arachidonic acid release by vesicle assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCytosolic phospholipase A2(Human)
University of MüNster

Curated by ChEMBL
LigandPNGBDBM50185355(1-[3-(4-octylphenoxy)-2-oxopropyl]indole-5-carboxa...)
Affinity DataIC50: 120nMAssay Description:Inhibition of human platelet cPLA2-alpha assessed as arachidonic acid release by vesicle assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCytosolic phospholipase A2(Human)
University of MüNster

Curated by ChEMBL
LigandPNGBDBM50206343(N-methyl-1-[3-(4-octylphenoxy)-2-oxopropyl]indole-...)
Affinity DataIC50: 310nMAssay Description:Inhibition of human platelet cPLA2-alpha assessed as arachidonic acid release by vesicle assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCytosolic phospholipase A2(Human)
University of MüNster

Curated by ChEMBL
LigandPNGBDBM50206338(N-methyl-1-[3-(4-octylphenoxy)-2-oxopropyl]indole-...)
Affinity DataIC50: 370nMAssay Description:Inhibition of human platelet cPLA2-alpha assessed as arachidonic acid release by vesicle assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCytosolic phospholipase A2(Human)
University of MüNster

Curated by ChEMBL
LigandPNGBDBM50206342(1-[3-(4-octylphenoxy)-2-oxopropyl]indole-5-sulfona...)
Affinity DataIC50: 390nMAssay Description:Inhibition of human platelet cPLA2-alpha assessed as arachidonic acid release by vesicle assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCytosolic phospholipase A2(Human)
University of MüNster

Curated by ChEMBL
LigandPNGBDBM50206339(1-[5-(morpholine-4-carbonyl)indol-1-yl]-3-(4-octyl...)
Affinity DataIC50: 500nMAssay Description:Inhibition of human platelet cPLA2-alpha assessed as arachidonic acid release by vesicle assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCytosolic phospholipase A2(Human)
University of MüNster

Curated by ChEMBL
LigandPNGBDBM50206340(N,N-dimethyl-1-[3-(4-octylphenoxy)-2-oxopropyl]ind...)
Affinity DataIC50: 500nMAssay Description:Inhibition of human platelet cPLA2-alpha assessed as arachidonic acid release by vesicle assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCytosolic phospholipase A2(Human)
University of MüNster

Curated by ChEMBL
LigandPNGBDBM50206336(N,N-dimethyl-1-[3-(4-octylphenoxy)-2-oxopropyl]ind...)
Affinity DataIC50: 840nMAssay Description:Inhibition of human platelet cPLA2-alpha assessed as arachidonic acid release by vesicle assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCytosolic phospholipase A2(Human)
University of MüNster

Curated by ChEMBL
LigandPNGBDBM50206337(1-(4-octylphenoxy)-3-[5-(1H-tetrazol-5-yl)indol-1-...)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of human platelet cPLA2-alpha assessed as arachidonic acid release by vesicle assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCytosolic phospholipase A2(Human)
University of MüNster

Curated by ChEMBL
LigandPNGBDBM50059523(Arachidonyltrifluoromethane | (6Z,9Z,12Z,15Z)-1,1,...)
Affinity DataIC50: 2.30E+3nMAssay Description:Inhibition of human platelet cPLA2-alpha assessed as arachidonic acid release by vesicle assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCytosolic phospholipase A2(Human)
University of MüNster

Curated by ChEMBL
LigandPNGBDBM50206341(3-{1-[3-(4-octylphenoxy)-2-oxopropyl]indol-5-yl}-4...)
Affinity DataIC50: 3.50E+3nMAssay Description:Inhibition of human platelet cPLA2-alpha assessed as arachidonic acid release by vesicle assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed