Compile Data Set for Download or QSAR
Report error Found 8 Enz. Inhib. hit(s) with all data for entry = 50037832
TargetVitamin D3 receptor(Bovine)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50205233((20S,22R)-22-methyl-1-alpha-25-dihydroxy-vitamin D...)
Affinity DataEC50:  0.0180nMAssay Description:Displacement of [3H]1,25-(OH)2D3 from vitamin D receptor in bovine thymusMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetVitamin D3 receptor(Bovine)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50205234((20S,22R)-22-methyl-1-alpha-25-dihydroxy-vitamin D...)
Affinity DataEC50:  0.0310nMAssay Description:Displacement of [3H]1,25-(OH)2D3 from vitamin D receptor in bovine thymusMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetVitamin D3 receptor(Bovine)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50200182((1S,3R,5Z,7E)-9,10-secocholesta-5,7,10(19)-triene-...)
Affinity DataEC50:  0.0710nMAssay Description:Displacement of [3H]1,25-(OH)2D3 from vitamin D receptor in bovine thymusMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetVitamin D3 receptor(Human)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50200182((1S,3R,5Z,7E)-9,10-secocholesta-5,7,10(19)-triene-...)
Affinity DataEC50:  0.5nMAssay Description:Induction of transactivation of human VDR responsive gene in COS7 cells by rat osteopontin luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetVitamin D3 receptor(Human)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50205234((20S,22R)-22-methyl-1-alpha-25-dihydroxy-vitamin D...)
Affinity DataEC50:  0.00300nMAssay Description:Induction of transactivation of human VDR responsive gene in COS7 cells by rat osteopontin luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetVitamin D3 receptor(Human)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50205233((20S,22R)-22-methyl-1-alpha-25-dihydroxy-vitamin D...)
Affinity DataEC50:  0.00200nMAssay Description:Induction of transactivation of human VDR responsive gene in COS7 cells by rat osteopontin luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetVitamin D3 receptor(Human)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50205235((20S,22R)-22-methyl-1-alpha-25-dihydroxy-vitamin D...)
Affinity DataEC50:  0.200nMAssay Description:Induction of transactivation of human VDR responsive gene in COS7 cells by rat osteopontin luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetVitamin D3 receptor(Bovine)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50205235((20S,22R)-22-methyl-1-alpha-25-dihydroxy-vitamin D...)
Affinity DataEC50:  0.890nMAssay Description:Displacement of [3H]1,25-(OH)2D3 from vitamin D receptor in bovine thymusMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed