Compile Data Set for Download or QSAR
Report error Found 19 Enz. Inhib. hit(s) with all data for entry = 50018632
TargetVoltage-dependent T-type calcium channel subunit alpha-1G(Human)
Institute of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50196467(3-(4-chlorobenzyl)-N-(3-(2-ethylpiperidin-1-yl)pro...)
Affinity DataIC50: 100nMAssay Description:Inhibition of alpha-1G T-type calcium channel expressed in HEK293 cells by electrophysiological methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVoltage-dependent T-type calcium channel subunit alpha-1G(Human)
Institute of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50148172(KYS-05042 | N-(4-(4-fluorophenylsulfonamido)benzyl...)
Affinity DataIC50: 200nMAssay Description:Inhibition of alpha-1G T-type calcium channel expressed in HEK293 cells by electrophysiological methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVoltage-dependent T-type calcium channel subunit alpha-1G(Human)
Institute of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50148180(KYS-05041 | N-(4-(4-methylphenylsulfonamido)benzyl...)
Affinity DataIC50: 250nMAssay Description:Inhibition of alpha-1G T-type calcium channel expressed in HEK293 cells by electrophysiological methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVoltage-dependent T-type calcium channel subunit alpha-1G(Human)
Institute of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50117922(CHEMBL45816 | Methoxy-acetic acid 2-(2-{[3-(1H-ben...)
Affinity DataIC50: 840nMAssay Description:Inhibition of alpha-1G T-type calcium channel expressed in HEK293 cells by electrophysiological methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVoltage-dependent T-type calcium channel subunit alpha-1G(Human)
Institute of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50148175(N-Benzyl-2-(3-phenyl-2-piperidin-1-yl-3,4-dihydro-...)
Affinity DataIC50: 900nMAssay Description:Inhibition of alpha-1G T-type calcium channel expressed in HEK293 cells by electrophysiological methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVoltage-dependent T-type calcium channel subunit alpha-1G(Human)
Institute of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50192101(2-(3-ethyl-2-(piperidin-1-yl)-3,4-dihydroquinazoli...)
Affinity DataIC50: 960nMAssay Description:Inhibition of alpha-1G T-type calcium channel expressed in HEK293 cells by electrophysiological methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVoltage-dependent T-type calcium channel subunit alpha-1G(Human)
Institute of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50197630(N-((3-(2-(trifluoromethyl)phenyl)isoxazol-5-yl)met...)
Affinity DataIC50: 1.02E+3nMAssay Description:Inhibition of alpha-1G T-type calcium channel expressed in HEK293 cells by electrophysiological methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVoltage-dependent T-type calcium channel subunit alpha-1G(Human)
Institute of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50197623(CHEMBL226876 | cid_6616154 | 3-(4-chlorobenzyl)-N-...)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of alpha-1G T-type calcium channel expressed in HEK293 cells by electrophysiological methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVoltage-dependent T-type calcium channel subunit alpha-1G(Human)
Institute of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50197622(3-(4-chlorobenzyl)-4-oxo-N-(3-(pyrrolidin-1-yl)pro...)
Affinity DataIC50: 1.16E+3nMAssay Description:Inhibition of alpha-1G T-type calcium channel expressed in HEK293 cells by electrophysiological methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVoltage-dependent T-type calcium channel subunit alpha-1G(Human)
Institute of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50197621(3-(4-chlorobenzyl)-N-(3-(azepan-1-yl)propyl)-4-oxo...)
Affinity DataIC50: 1.41E+3nMAssay Description:Inhibition of alpha-1G T-type calcium channel expressed in HEK293 cells by electrophysiological methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVoltage-dependent T-type calcium channel subunit alpha-1G(Human)
Institute of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50197624(2-(4-(2,4-dimethylphenyl)piperazin-1-yl)-N-((3-(2-...)
Affinity DataIC50: 1.53E+3nMAssay Description:Inhibition of alpha-1G T-type calcium channel expressed in HEK293 cells by electrophysiological methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVoltage-dependent T-type calcium channel subunit alpha-1G(Human)
Institute of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50197633(2-(4-(2,4-dimethylphenyl)piperazin-1-yl)-N-((3-(2-...)
Affinity DataIC50: 2.02E+3nMAssay Description:Inhibition of alpha-1G T-type calcium channel expressed in HEK293 cells by electrophysiological methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVoltage-dependent T-type calcium channel subunit alpha-1G(Human)
Institute of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50197632(N-((3-(2-methoxyphenyl)isoxazol-5-yl)methyl)-2-(4-...)
Affinity DataIC50: 2.04E+3nMAssay Description:Inhibition of alpha-1G T-type calcium channel expressed in HEK293 cells by electrophysiological methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVoltage-dependent T-type calcium channel subunit alpha-1G(Human)
Institute of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50197628(3-(4-chlorobenzyl)-4-oxo-N-(3-(piperidin-1-yl)prop...)
Affinity DataIC50: 2.08E+3nMAssay Description:Inhibition of alpha-1G T-type calcium channel expressed in HEK293 cells by electrophysiological methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVoltage-dependent T-type calcium channel subunit alpha-1G(Human)
Institute of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50197625(3-(4-chlorobenzyl)-N-(3-(4-ethylpiperazin-1-yl)pro...)
Affinity DataIC50: 2.53E+3nMAssay Description:Inhibition of alpha-1G T-type calcium channel expressed in HEK293 cells by electrophysiological methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVoltage-dependent T-type calcium channel subunit alpha-1G(Human)
Institute of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50197629(3-(4-chlorobenzyl)-N-(3-(benzyl(methyl)amino)propy...)
Affinity DataIC50: 4.69E+3nMAssay Description:Inhibition of alpha-1G T-type calcium channel expressed in HEK293 cells by electrophysiological methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVoltage-dependent T-type calcium channel subunit alpha-1G(Human)
Institute of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50197626(3-(4-chlorobenzyl)-N-(2-(butyl(methyl)amino)ethyl)...)
Affinity DataIC50: 1.14E+4nMAssay Description:Inhibition of alpha-1G T-type calcium channel expressed in HEK293 cells by electrophysiological methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVoltage-dependent T-type calcium channel subunit alpha-1G(Human)
Institute of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50197627(CHEMBL427449 | cid_3243445 | 3-(4-chlorobenzyl)-7-...)
Affinity DataIC50: 1.14E+4nMAssay Description:Inhibition of alpha-1G T-type calcium channel expressed in HEK293 cells by electrophysiological methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVoltage-dependent T-type calcium channel subunit alpha-1G(Human)
Institute of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50197631(3-(4-chlorobenzyl)-N-(2-(dimethylamino)ethyl)-4-ox...)
Affinity DataIC50: 5.35E+4nMAssay Description:Inhibition of alpha-1G T-type calcium channel expressed in HEK293 cells by electrophysiological methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed