Compile Data Set for Download or QSAR
Report error Found 113 Enz. Inhib. hit(s) with all data for entry = 50018370
LigandPNGBDBM50194955(2-((6-(2-(2-(3-chlorophenyl)-5-methyloxazol-4-yl)e...)
Affinity DataEC50:  1nMAssay Description:Agonist activity at human PPAR gamma in a HepG2 cells by PPAR-GAL4 transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50194957(2-((6-(2-(2-(3-methoxyphenyl)-5-methyloxazol-4-yl)...)
Affinity DataEC50:  2nMAssay Description:Agonist activity at human PPAR gamma in a HepG2 cells by PPAR-GAL4 transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50194950(2-((6-(2-(2-(4-methoxyphenyl)-5-methyloxazol-4-yl)...)
Affinity DataEC50:  5nMAssay Description:Agonist activity at human PPAR gamma in a HepG2 cells by PPAR-GAL4 transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50194961(2-((6-(2-(5-methyl-2-m-tolyloxazol-4-yl)ethoxy)pyr...)
Affinity DataEC50:  5nMAssay Description:Agonist activity at human PPAR gamma in a HepG2 cells by PPAR-GAL4 transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50194953(2-ethoxy-3-(6-(2-(5-methyl-2-phenyloxazol-4-yl)eth...)
Affinity DataEC50:  6nMAssay Description:Agonist activity at human PPAR gamma in a HepG2 cells by PPAR-GAL4 transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50194970(2-((6-(2-(5-methyl-2-(4-(trifluoromethyl)phenyl)ox...)
Affinity DataEC50:  6nMAssay Description:Agonist activity at human PPAR gamma in a HepG2 cells by PPAR-GAL4 transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50194976((S)-2-((6-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)...)
Affinity DataKi:  6nMAssay Description:Displacement of radiolabeled darglitazone from human PPAR gamma by SPA binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50194957(2-((6-(2-(2-(3-methoxyphenyl)-5-methyloxazol-4-yl)...)
Affinity DataKi:  7nMAssay Description:Displacement of radiolabeled darglitazone from human PPAR gamma by SPA binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50194971(2-((6-(2-(5-methyl-2-(3-(trifluoromethyl)phenyl)ox...)
Affinity DataEC50:  8nMAssay Description:Agonist activity at human PPAR alpha in a HepG2 cells by PPAR-GAL4 transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50194969(2-((6-(2-(2-(4-chlorophenyl)-5-methyloxazol-4-yl)e...)
Affinity DataEC50:  10nMAssay Description:Agonist activity at human PPAR alpha in a HepG2 cells by PPAR-GAL4 transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50194955(2-((6-(2-(2-(3-chlorophenyl)-5-methyloxazol-4-yl)e...)
Affinity DataKi:  11nMAssay Description:Displacement of radiolabeled darglitazone from human PPAR gamma by SPA binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50194970(2-((6-(2-(5-methyl-2-(4-(trifluoromethyl)phenyl)ox...)
Affinity DataEC50:  11nMAssay Description:Agonist activity at human PPAR alpha in a HepG2 cells by PPAR-GAL4 transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50194967(2-((6-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)pyri...)
Affinity DataEC50:  12nMAssay Description:Agonist activity at human PPAR gamma in a HepG2 cells by PPAR-GAL4 transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50194968(3-(6-(4-(3-chlorophenoxy)-2-methylphenethoxy)pyrid...)
Affinity DataEC50:  13nMAssay Description:Displacement of radiolabeled GW-2331 from human PPAR alpha by SPA binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50194963(2-methoxy-3-(6-(2-(5-methyl-2-phenyloxazol-4-yl)et...)
Affinity DataEC50:  13nMAssay Description:Agonist activity at human PPAR gamma in a HepG2 cells by PPAR-GAL4 transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50194969(2-((6-(2-(2-(4-chlorophenyl)-5-methyloxazol-4-yl)e...)
Affinity DataEC50:  14nMAssay Description:Displacement of radiolabeled GW-2331 from human PPAR alpha by SPA binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50194976((S)-2-((6-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)...)
Affinity DataEC50:  14nMAssay Description:Agonist activity at human PPAR gamma in a HepG2 cells by PPAR-GAL4 transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50194968(3-(6-(4-(3-chlorophenoxy)-2-methylphenethoxy)pyrid...)
Affinity DataKi:  15nMAssay Description:Displacement of radiolabeled darglitazone from human PPAR gamma by SPA binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50194971(2-((6-(2-(5-methyl-2-(3-(trifluoromethyl)phenyl)ox...)
Affinity DataKi:  15nMAssay Description:Displacement of radiolabeled darglitazone from human PPAR gamma by SPA binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50194961(2-((6-(2-(5-methyl-2-m-tolyloxazol-4-yl)ethoxy)pyr...)
Affinity DataKi:  16nMAssay Description:Displacement of radiolabeled darglitazone from human PPAR gamma by SPA binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50194950(2-((6-(2-(2-(4-methoxyphenyl)-5-methyloxazol-4-yl)...)
Affinity DataKi:  17nMAssay Description:Displacement of radiolabeled darglitazone from human PPAR gamma by SPA binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50194970(2-((6-(2-(5-methyl-2-(4-(trifluoromethyl)phenyl)ox...)
Affinity DataEC50:  21nMAssay Description:Displacement of radiolabeled GW-2331 from human PPAR alpha by SPA binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50194974(2-((6-(2-(5-methyl-2-p-tolyloxazol-4-yl)ethoxy)pyr...)
Affinity DataEC50:  22nMAssay Description:Agonist activity at human PPAR gamma in a HepG2 cells by PPAR-GAL4 transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50194974(2-((6-(2-(5-methyl-2-p-tolyloxazol-4-yl)ethoxy)pyr...)
Affinity DataEC50:  23nMAssay Description:Agonist activity at human PPAR alpha in a HepG2 cells by PPAR-GAL4 transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50194974(2-((6-(2-(5-methyl-2-p-tolyloxazol-4-yl)ethoxy)pyr...)
Affinity DataKi:  23nMAssay Description:Displacement of radiolabeled darglitazone from human PPAR gamma by SPA binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50194973(2-((6-(2-(2-(4-cyanophenyl)-5-methyloxazol-4-yl)et...)
Affinity DataEC50:  28nMAssay Description:Agonist activity at human PPAR gamma in a HepG2 cells by PPAR-GAL4 transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50194973(2-((6-(2-(2-(4-cyanophenyl)-5-methyloxazol-4-yl)et...)
Affinity DataEC50:  31nMAssay Description:Agonist activity at human PPAR alpha in a HepG2 cells by PPAR-GAL4 transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50194974(2-((6-(2-(5-methyl-2-p-tolyloxazol-4-yl)ethoxy)pyr...)
Affinity DataEC50:  31nMAssay Description:Displacement of radiolabeled GW-2331 from human PPAR alpha by SPA binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50194976((S)-2-((6-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)...)
Affinity DataEC50:  32nMAssay Description:Displacement of radiolabeled GW-2331 from human PPAR alpha by SPA binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50194953(2-ethoxy-3-(6-(2-(5-methyl-2-phenyloxazol-4-yl)eth...)
Affinity DataEC50:  33nMAssay Description:Agonist activity at human PPAR alpha in a HepG2 cells by PPAR-GAL4 transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50194967(2-((6-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)pyri...)
Affinity DataKi:  38nMAssay Description:Displacement of radiolabeled darglitazone from human PPAR gamma by SPA binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50194969(2-((6-(2-(2-(4-chlorophenyl)-5-methyloxazol-4-yl)e...)
Affinity DataEC50:  42nMAssay Description:Agonist activity at human PPAR gamma in a HepG2 cells by PPAR-GAL4 transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50194953(2-ethoxy-3-(6-(2-(5-methyl-2-phenyloxazol-4-yl)eth...)
Affinity DataEC50:  43nMAssay Description:Displacement of radiolabeled GW-2331 from human PPAR alpha by SPA binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50194955(2-((6-(2-(2-(3-chlorophenyl)-5-methyloxazol-4-yl)e...)
Affinity DataEC50:  46nMAssay Description:Agonist activity at human PPAR alpha in a HepG2 cells by PPAR-GAL4 transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50194967(2-((6-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)pyri...)
Affinity DataEC50:  48nMAssay Description:Agonist activity at human PPAR alpha in a HepG2 cells by PPAR-GAL4 transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50194968(3-(6-(4-(3-chlorophenoxy)-2-methylphenethoxy)pyrid...)
Affinity DataEC50:  50nMAssay Description:Agonist activity at human PPAR gamma in a HepG2 cells by PPAR-GAL4 transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50194969(2-((6-(2-(2-(4-chlorophenyl)-5-methyloxazol-4-yl)e...)
Affinity DataKi:  52nMAssay Description:Displacement of radiolabeled darglitazone from human PPAR gamma by SPA binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50194963(2-methoxy-3-(6-(2-(5-methyl-2-phenyloxazol-4-yl)et...)
Affinity DataKi:  63nMAssay Description:Displacement of radiolabeled darglitazone from human PPAR gamma by SPA binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50194950(2-((6-(2-(2-(4-methoxyphenyl)-5-methyloxazol-4-yl)...)
Affinity DataEC50:  65nMAssay Description:Displacement of radiolabeled GW-2331 from human PPAR alpha by SPA binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50194954(2-((6-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)pyri...)
Affinity DataEC50:  65nMAssay Description:Agonist activity at human PPAR gamma in a HepG2 cells by PPAR-GAL4 transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50194967(2-((6-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)pyri...)
Affinity DataEC50:  78nMAssay Description:Displacement of radiolabeled GW-2331 from human PPAR alpha by SPA binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50194952(2-((6-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)pyri...)
Affinity DataEC50:  78nMAssay Description:Displacement of radiolabeled GW-2331 from human PPAR alpha by SPA binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50194952(2-((6-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)pyri...)
Affinity DataKi:  81nMAssay Description:Displacement of radiolabeled darglitazone from human PPAR gamma by SPA binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50194963(2-methoxy-3-(6-(2-(5-methyl-2-phenyloxazol-4-yl)et...)
Affinity DataEC50:  83nMAssay Description:Agonist activity at human PPAR alpha in a HepG2 cells by PPAR-GAL4 transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50194957(2-((6-(2-(2-(3-methoxyphenyl)-5-methyloxazol-4-yl)...)
Affinity DataEC50:  90nMAssay Description:Agonist activity at human PPAR alpha in a HepG2 cells by PPAR-GAL4 transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50194970(2-((6-(2-(5-methyl-2-(4-(trifluoromethyl)phenyl)ox...)
Affinity DataKi:  94nMAssay Description:Displacement of radiolabeled darglitazone from human PPAR gamma by SPA binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50194955(2-((6-(2-(2-(3-chlorophenyl)-5-methyloxazol-4-yl)e...)
Affinity DataEC50:  99nMAssay Description:Displacement of radiolabeled GW-2331 from human PPAR alpha by SPA binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50194971(2-((6-(2-(5-methyl-2-(3-(trifluoromethyl)phenyl)ox...)
Affinity DataEC50:  100nMAssay Description:Displacement of radiolabeled GW-2331 from human PPAR alpha by SPA binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50194965((S)-2-methoxy-2-methyl-3-(6-(2-(5-methyl-2-phenylo...)
Affinity DataEC50:  110nMAssay Description:Agonist activity at human PPAR gamma in a HepG2 cells by PPAR-GAL4 transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50194965((S)-2-methoxy-2-methyl-3-(6-(2-(5-methyl-2-phenylo...)
Affinity DataEC50:  111nMAssay Description:Agonist activity at human PPAR alpha in a HepG2 cells by PPAR-GAL4 transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
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