Compile Data Set for Download or QSAR
Report error Found 22 Enz. Inhib. hit(s) with all data for entry = 50042256
TargetMelanin-concentrating hormone receptor 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50241083(6-(4-chlorophenyl)-3-(3-methoxy-4-(2-(pyrrolidin-1...)
Affinity DataIC50: 0.5nMAssay Description:Antagonist activity against human MCHR1 expressed in CHO cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50422940(CHEMBL213008)
Affinity DataIC50: 1nMAssay Description:Antagonist activity against human MCHR1 expressed in CHO cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50422936(CHEMBL212657)
Affinity DataIC50: 1.30nMAssay Description:Antagonist activity against human MCHR1 expressed in CHO cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50422927(CHEMBL441368)
Affinity DataIC50: 1.60nMAssay Description:Antagonist activity against human MCHR1 expressed in CHO cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50422930(CHEMBL214276)
Affinity DataIC50: 2nMAssay Description:Antagonist activity against human MCHR1 expressed in CHO cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50422924(CHEMBL214416)
Affinity DataIC50: 2.5nMAssay Description:Antagonist activity against human MCHR1 expressed in CHO cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50422926(CHEMBL215565)
Affinity DataIC50: 3.20nMAssay Description:Antagonist activity against human MCHR1 expressed in CHO cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50422939(CHEMBL439146)
Affinity DataIC50: 5nMAssay Description:Antagonist activity against human MCHR1 expressed in CHO cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50422932(CHEMBL212958)
Affinity DataIC50: 5nMAssay Description:Antagonist activity against human MCHR1 expressed in CHO cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50422922(CHEMBL384113)
Affinity DataIC50: 6.30nMAssay Description:Antagonist activity against human MCHR1 expressed in CHO cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50422933(CHEMBL212137)
Affinity DataIC50: 6.30nMAssay Description:Antagonist activity against human MCHR1 expressed in CHO cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50422938(CHEMBL215862)
Affinity DataIC50: 13nMAssay Description:Antagonist activity against human MCHR1 expressed in CHO cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50422921(CHEMBL214429)
Affinity DataIC50: 20nMAssay Description:Antagonist activity against human MCHR1 expressed in CHO cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50422929(CHEMBL212883)
Affinity DataIC50: 25nMAssay Description:Antagonist activity against human MCHR1 expressed in CHO cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50422935(CHEMBL215334)
Affinity DataIC50: 25nMAssay Description:Antagonist activity against human MCHR1 expressed in CHO cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50422923(CHEMBL387195)
Affinity DataIC50: 100nMAssay Description:Antagonist activity against human MCHR1 expressed in CHO cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50422928(CHEMBL214427)
Affinity DataIC50: 126nMAssay Description:Antagonist activity against human MCHR1 expressed in CHO cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50422941(CHEMBL213154)
Affinity DataIC50: 200nMAssay Description:Antagonist activity against human MCHR1 expressed in CHO cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50422931(CHEMBL266415)
Affinity DataIC50: 1.26E+3nMAssay Description:Antagonist activity against human MCHR1 expressed in CHO cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50422925(CHEMBL212963)
Affinity DataIC50: 1.59E+3nMAssay Description:Antagonist activity against human MCHR1 expressed in CHO cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50422937(CHEMBL377758)
Affinity DataIC50: 3.16E+3nMAssay Description:Antagonist activity against human MCHR1 expressed in CHO cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50422934(CHEMBL424723)
Affinity DataIC50: 3.98E+3nMAssay Description:Antagonist activity against human MCHR1 expressed in CHO cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed