Compile Data Set for Download or QSAR
Report error Found 13 Enz. Inhib. hit(s) with all data for entry = 50018061
Target5-hydroxytryptamine receptor 2A(Rat)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50190613((+/-)-(2,3-dihydro-4,5,6-trimethoxy-1H-inden-1-yl)...)
Affinity DataEC50:  6.10E+3nMAssay Description:Activity at rat 5HT2A receptor assessed as 5-HT-stimulated IP3 accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Rat)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50059891(3,4,5-trimethoxyphenylethylamine | 3,4,5-trimethox...)
Affinity DataEC50:  1.13E+4nMAssay Description:Activity at rat 5HT2A receptor assessed as 5-HT-stimulated IP3 accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Rat)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50190614((S)-(-)-(4,5,6-trimethoxyindan-1-yl)methanamine | ...)
Affinity DataEC50: >5.00E+4nMAssay Description:Activity at rat 5HT2A receptor assessed as 5-HT-stimulated IP3 accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Rat)
Purdue University

Curated by ChEMBL
LigandPNGBDBM21342((4R,7R)-N,N-diethyl-6-methyl-6,11-diazatetracyclo[...)
Affinity DataEC50:  9.80nMAssay Description:Activity at rat 5HT2A receptor assessed as 5-HT-stimulated IP3 accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMedPDB3D3D Structure (crystal)
Target5-hydroxytryptamine receptor 2A(Rat)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50190615((R)-(+)-(4,5,6-trimethoxyindan-1-yl)methanamine | ...)
Affinity DataEC50:  3.20E+3nMAssay Description:Activity at rat 5HT2A receptor assessed as 5-HT-stimulated IP3 accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Rat)
Purdue University

Curated by ChEMBL
LigandPNGBDBM21342((4R,7R)-N,N-diethyl-6-methyl-6,11-diazatetracyclo[...)
Affinity DataKi:  3.5nMAssay Description:Displacement of [125I]DOI from rat 5HT2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMedPDB3D3D Structure (crystal)
Target5-hydroxytryptamine receptor 2C(Rat)
Purdue University

Curated by ChEMBL
LigandPNGBDBM21342((4R,7R)-N,N-diethyl-6-methyl-6,11-diazatetracyclo[...)
Affinity DataKi:  5.5nMAssay Description:Displacement of [125I]DOI from rat 5HT2C receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Rat)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50190613((+/-)-(2,3-dihydro-4,5,6-trimethoxy-1H-inden-1-yl)...)
Affinity DataKi:  60nMAssay Description:Displacement of [125I]DOI from rat 5HT2C receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Rat)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50190615((R)-(+)-(4,5,6-trimethoxyindan-1-yl)methanamine | ...)
Affinity DataKi:  69nMAssay Description:Displacement of [125I]DOI from rat 5HT2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Rat)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50190613((+/-)-(2,3-dihydro-4,5,6-trimethoxy-1H-inden-1-yl)...)
Affinity DataKi:  130nMAssay Description:Displacement of [125I]DOI from rat 5HT2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Rat)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50059891(3,4,5-trimethoxyphenylethylamine | 3,4,5-trimethox...)
Affinity DataKi:  360nMAssay Description:Displacement of [125I]DOI from rat 5HT2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Rat)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50059891(3,4,5-trimethoxyphenylethylamine | 3,4,5-trimethox...)
Affinity DataKi:  380nMAssay Description:Displacement of [125I]DOI from rat 5HT2C receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Rat)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50190614((S)-(-)-(4,5,6-trimethoxyindan-1-yl)methanamine | ...)
Affinity DataKi:  1.12E+3nMAssay Description:Displacement of [125I]DOI from rat 5HT2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed