Compile Data Set for Download or QSAR
Report error Found 5 Enz. Inhib. hit(s) with all data for entry = 50042252
TargetBeta-1 adrenergic receptor(Rat)
University of Melbourne

Curated by ChEMBL
LigandPNGBDBM50422862(125I-CYP | CHEMBL210309)
Affinity DataKd:  0.316nMAssay Description:Antagonist activity at rat beta-1 adrenergic receptor Y356A mutant expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Rat)
University of Melbourne

Curated by ChEMBL
LigandPNGBDBM50422862(125I-CYP | CHEMBL210309)
Affinity DataKd:  0.0631nMAssay Description:Antagonist activity at rat beta-1 adrenergic receptor S190A mutant expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Rat)
University of Melbourne

Curated by ChEMBL
LigandPNGBDBM50422862(125I-CYP | CHEMBL210309)
Affinity DataKd:  0.0631nMAssay Description:Antagonist activity at rat wild type beta-1 adrenergic receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Rat)
University of Melbourne

Curated by ChEMBL
LigandPNGBDBM50422862(125I-CYP | CHEMBL210309)
Affinity DataKd:  0.0794nMAssay Description:Antagonist activity at rat beta-1 adrenergic receptor Y356F mutant expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Rat)
University of Melbourne

Curated by ChEMBL
LigandPNGBDBM50422862(125I-CYP | CHEMBL210309)
Affinity DataKd:  0.0631nMAssay Description:Antagonist activity at rat beta-1 adrenergic receptor W134A mutant expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed