Compile Data Set for Download or QSAR
Report error Found 36 Enz. Inhib. hit(s) with all data for entry = 50017896
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Human)
De Montfort University

Curated by ChEMBL
LigandPNGBDBM50188069(12-oxo-10,12-dihydro-10-aza-4b-azonia-indeno[2,1-b...)
Affinity DataIC50: 410nMAssay Description:Inhibition of Cdk4/Cyclin D1More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Human)
De Montfort University

Curated by ChEMBL
LigandPNGBDBM50188071(biphenyl-4-carboxylic acid [2-(1H-indol-3-yl)-ethy...)
Affinity DataIC50: 6.20E+3nMAssay Description:Inhibition of Cdk4/Cyclin D1More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Human)
De Montfort University

Curated by ChEMBL
LigandPNGBDBM50188075(N-(2-(1H-indol-3-yl)ethyl)-4-bromo-N-methylbenzami...)
Affinity DataIC50: 3.70E+4nMAssay Description:Inhibition of Cdk4/Cyclin D1More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Human)
De Montfort University

Curated by ChEMBL
LigandPNGBDBM50188066(N-(2-(1H-indol-3-yl)ethyl)-4-chloro-N-methylbenzam...)
Affinity DataIC50: 3.80E+4nMAssay Description:Inhibition of Cdk4/Cyclin D1More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Human)
De Montfort University

Curated by ChEMBL
LigandPNGBDBM50188073(N-(2-(1H-indol-3-yl)ethyl)-2-chloro-N-methylbenzam...)
Affinity DataIC50: 4.60E+4nMAssay Description:Inhibition of Cdk4/Cyclin D1More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Human)
De Montfort University

Curated by ChEMBL
LigandPNGBDBM50188064(N-(2-(1H-indol-3-yl)ethyl)-4-tert-butyl-N-methylbe...)
Affinity DataIC50: 4.90E+4nMAssay Description:Inhibition of Cdk4/Cyclin D1More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Human)
De Montfort University

Curated by ChEMBL
LigandPNGBDBM50188068(N-(2-(1H-indol-3-yl)ethyl)-4-fluoro-N-methylbenzam...)
Affinity DataIC50: 5.90E+4nMAssay Description:Inhibition of Cdk4/Cyclin D1More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Human)
De Montfort University

Curated by ChEMBL
LigandPNGBDBM50188078(N-(2-(1H-indol-3-yl)ethyl)-N,4-dimethylbenzamide |...)
Affinity DataIC50: 6.30E+4nMAssay Description:Inhibition of Cdk4/Cyclin D1More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Human)
De Montfort University

Curated by ChEMBL
LigandPNGBDBM50188072(N-(2-(1H-indol-3-yl)ethyl)-3-bromo-N-methylbenzami...)
Affinity DataIC50: 7.40E+4nMAssay Description:Inhibition of Cdk4/Cyclin D1More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Human)
De Montfort University

Curated by ChEMBL
LigandPNGBDBM50188067(N-(2-(1H-indol-3-yl)ethyl)-N,3-dimethylbenzamide |...)
Affinity DataIC50: 7.80E+4nMAssay Description:Inhibition of Cdk4/Cyclin D1More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Human)
De Montfort University

Curated by ChEMBL
LigandPNGBDBM50188079(N-(2-(1H-indol-3-yl)ethyl)-2-methoxy-N-methylbenza...)
Affinity DataIC50: 7.90E+4nMAssay Description:Inhibition of Cdk4/Cyclin D1More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Human)
De Montfort University

Curated by ChEMBL
LigandPNGBDBM50188081(N-(2-(1H-indol-3-yl)ethyl)-3-methoxy-N-methylbenza...)
Affinity DataIC50: 8.10E+4nMAssay Description:Inhibition of Cdk4/Cyclin D1More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Human)
De Montfort University

Curated by ChEMBL
LigandPNGBDBM50188070(N-(2-(1H-indol-3-yl)ethyl)-3-fluoro-N-methylbenzam...)
Affinity DataIC50: 8.80E+4nMAssay Description:Inhibition of Cdk4/Cyclin D1More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Human)
De Montfort University

Curated by ChEMBL
LigandPNGBDBM50188074(N-(2-(1H-indol-3-yl)ethyl)-N-methylbenzamide | CHE...)
Affinity DataIC50: 8.80E+4nMAssay Description:Inhibition of Cdk4/Cyclin D1More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Human)
De Montfort University

Curated by ChEMBL
LigandPNGBDBM50188077(N-(2-(1H-indol-3-yl)ethyl)-2-bromo-N-methylbenzami...)
Affinity DataIC50: 9.50E+4nMAssay Description:Inhibition of Cdk4/Cyclin D1More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Human)
De Montfort University

Curated by ChEMBL
LigandPNGBDBM50188065(N-(2-(1H-indol-3-yl)ethyl)-2-fluoro-N-methylbenzam...)
Affinity DataIC50: 1.03E+5nMAssay Description:Inhibition of Cdk4/Cyclin D1More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Human)
De Montfort University

Curated by ChEMBL
LigandPNGBDBM50188076(N-(2-(1H-indol-3-yl)ethyl)-3-chloro-N-methylbenzam...)
Affinity DataIC50: 1.09E+5nMAssay Description:Inhibition of Cdk4/Cyclin D1More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Human)
De Montfort University

Curated by ChEMBL
LigandPNGBDBM50188080(N-(2-(1H-indol-3-yl)ethyl)-N,2-dimethylbenzamide |...)
Affinity DataIC50: 1.13E+5nMAssay Description:Inhibition of Cdk4/Cyclin D1More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCyclin-A1/Cyclin-A2/Cyclin-dependent kinase 2(Human)
De Montfort University

Curated by ChEMBL
LigandPNGBDBM50188069(12-oxo-10,12-dihydro-10-aza-4b-azonia-indeno[2,1-b...)
Affinity DataIC50: 2.50E+5nMAssay Description:Inhibition of Cdk2/Cyclin AMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCyclin-A1/Cyclin-A2/Cyclin-dependent kinase 2(Human)
De Montfort University

Curated by ChEMBL
LigandPNGBDBM50188071(biphenyl-4-carboxylic acid [2-(1H-indol-3-yl)-ethy...)
Affinity DataIC50: 5.21E+5nMAssay Description:Inhibition of Cdk2/Cyclin AMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCyclin-A1/Cyclin-A2/Cyclin-dependent kinase 2(Human)
De Montfort University

Curated by ChEMBL
LigandPNGBDBM50188075(N-(2-(1H-indol-3-yl)ethyl)-4-bromo-N-methylbenzami...)
Affinity DataIC50: 5.80E+5nMAssay Description:Inhibition of Cdk2/Cyclin AMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCyclin-A1/Cyclin-A2/Cyclin-dependent kinase 2(Human)
De Montfort University

Curated by ChEMBL
LigandPNGBDBM50188077(N-(2-(1H-indol-3-yl)ethyl)-2-bromo-N-methylbenzami...)
Affinity DataIC50: 5.84E+5nMAssay Description:Inhibition of Cdk2/Cyclin AMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCyclin-A1/Cyclin-A2/Cyclin-dependent kinase 2(Human)
De Montfort University

Curated by ChEMBL
LigandPNGBDBM50188072(N-(2-(1H-indol-3-yl)ethyl)-3-bromo-N-methylbenzami...)
Affinity DataIC50: 6.35E+5nMAssay Description:Inhibition of Cdk2/Cyclin AMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCyclin-A1/Cyclin-A2/Cyclin-dependent kinase 2(Human)
De Montfort University

Curated by ChEMBL
LigandPNGBDBM50188064(N-(2-(1H-indol-3-yl)ethyl)-4-tert-butyl-N-methylbe...)
Affinity DataIC50: 6.58E+5nMAssay Description:Inhibition of Cdk2/Cyclin AMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCyclin-A1/Cyclin-A2/Cyclin-dependent kinase 2(Human)
De Montfort University

Curated by ChEMBL
LigandPNGBDBM50188066(N-(2-(1H-indol-3-yl)ethyl)-4-chloro-N-methylbenzam...)
Affinity DataIC50: 7.31E+5nMAssay Description:Inhibition of Cdk2/Cyclin AMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCyclin-A1/Cyclin-A2/Cyclin-dependent kinase 2(Human)
De Montfort University

Curated by ChEMBL
LigandPNGBDBM50188070(N-(2-(1H-indol-3-yl)ethyl)-3-fluoro-N-methylbenzam...)
Affinity DataIC50: 7.65E+5nMAssay Description:Inhibition of Cdk2/Cyclin AMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCyclin-A1/Cyclin-A2/Cyclin-dependent kinase 2(Human)
De Montfort University

Curated by ChEMBL
LigandPNGBDBM50188073(N-(2-(1H-indol-3-yl)ethyl)-2-chloro-N-methylbenzam...)
Affinity DataIC50: 7.84E+5nMAssay Description:Inhibition of Cdk2/Cyclin AMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCyclin-A1/Cyclin-A2/Cyclin-dependent kinase 2(Human)
De Montfort University

Curated by ChEMBL
LigandPNGBDBM50188078(N-(2-(1H-indol-3-yl)ethyl)-N,4-dimethylbenzamide |...)
Affinity DataIC50: 7.90E+5nMAssay Description:Inhibition of Cdk2/Cyclin AMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCyclin-A1/Cyclin-A2/Cyclin-dependent kinase 2(Human)
De Montfort University

Curated by ChEMBL
LigandPNGBDBM50188067(N-(2-(1H-indol-3-yl)ethyl)-N,3-dimethylbenzamide |...)
Affinity DataIC50: 8.30E+5nMAssay Description:Inhibition of Cdk2/Cyclin AMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCyclin-A1/Cyclin-A2/Cyclin-dependent kinase 2(Human)
De Montfort University

Curated by ChEMBL
LigandPNGBDBM50188079(N-(2-(1H-indol-3-yl)ethyl)-2-methoxy-N-methylbenza...)
Affinity DataIC50: 8.49E+5nMAssay Description:Inhibition of Cdk2/Cyclin AMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCyclin-A1/Cyclin-A2/Cyclin-dependent kinase 2(Human)
De Montfort University

Curated by ChEMBL
LigandPNGBDBM50188068(N-(2-(1H-indol-3-yl)ethyl)-4-fluoro-N-methylbenzam...)
Affinity DataIC50: 8.50E+5nMAssay Description:Inhibition of Cdk2/Cyclin AMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCyclin-A1/Cyclin-A2/Cyclin-dependent kinase 2(Human)
De Montfort University

Curated by ChEMBL
LigandPNGBDBM50188081(N-(2-(1H-indol-3-yl)ethyl)-3-methoxy-N-methylbenza...)
Affinity DataIC50: 9.38E+5nMAssay Description:Inhibition of Cdk2/Cyclin AMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCyclin-A1/Cyclin-A2/Cyclin-dependent kinase 2(Human)
De Montfort University

Curated by ChEMBL
LigandPNGBDBM50188080(N-(2-(1H-indol-3-yl)ethyl)-N,2-dimethylbenzamide |...)
Affinity DataIC50: 1.13E+6nMAssay Description:Inhibition of Cdk2/Cyclin AMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCyclin-A1/Cyclin-A2/Cyclin-dependent kinase 2(Human)
De Montfort University

Curated by ChEMBL
LigandPNGBDBM50188074(N-(2-(1H-indol-3-yl)ethyl)-N-methylbenzamide | CHE...)
Affinity DataIC50: 1.52E+6nMAssay Description:Inhibition of Cdk2/Cyclin AMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCyclin-A1/Cyclin-A2/Cyclin-dependent kinase 2(Human)
De Montfort University

Curated by ChEMBL
LigandPNGBDBM50188076(N-(2-(1H-indol-3-yl)ethyl)-3-chloro-N-methylbenzam...)
Affinity DataIC50: 1.12E+6nMAssay Description:Inhibition of Cdk2/Cyclin AMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCyclin-A1/Cyclin-A2/Cyclin-dependent kinase 2(Human)
De Montfort University

Curated by ChEMBL
LigandPNGBDBM50188065(N-(2-(1H-indol-3-yl)ethyl)-2-fluoro-N-methylbenzam...)
Affinity DataIC50: 1.23E+6nMAssay Description:Inhibition of Cdk2/Cyclin AMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed