Compile Data Set for Download or QSAR
Report error Found 13 Enz. Inhib. hit(s) with all data for entry = 50017871
TargetIntegrase(Human immunodeficiency virus type 1)
Gilead Sciences

Curated by ChEMBL
LigandPNGBDBM50187761(7-(4-fluorobenzyl)-9-hydroxy-5-(morpholine-4-carbo...)
Affinity DataIC50: 36nMAssay Description:Inhibition of strand transfer activity of HIV integraseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Gilead Sciences

Curated by ChEMBL
LigandPNGBDBM23403(CHEMBL209440 | 7-[(4-fluorophenyl)methyl]-9-hydrox...)
Affinity DataIC50: 50nMAssay Description:Inhibition of strand transfer activity of HIV integraseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Gilead Sciences

Curated by ChEMBL
LigandPNGBDBM23402(5-(1,1-dioxo-1,2-thiazinan-2-yl)-N-[(4-fluoropheny...)
Affinity DataIC50: 50nMAssay Description:Inhibition of strand transfer activity of HIV integraseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Gilead Sciences

Curated by ChEMBL
LigandPNGBDBM50187760(7-(4-fluorobenzyl)-9-hydroxy-6,7-dihydropyrrolo[3,...)
Affinity DataIC50: 70nMAssay Description:Inhibition of strand transfer activity of HIV integraseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Gilead Sciences

Curated by ChEMBL
LigandPNGBDBM50187764(7-(4-fluorobenzyl)-9-hydroxy-5-methoxy-7H-pyrrolo[...)
Affinity DataIC50: 80nMAssay Description:Inhibition of strand transfer activity of HIV integraseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Gilead Sciences

Curated by ChEMBL
LigandPNGBDBM50187759(7-(4-fluorobenzyl)-9-hydroxy-8-oxo-N-(pyridin-2-yl...)
Affinity DataIC50: 190nMAssay Description:Inhibition of strand transfer activity of HIV integraseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Gilead Sciences

Curated by ChEMBL
LigandPNGBDBM50187765(7-(4-fluorobenzyl)-5-(2,6-difluorophenyl)-9-hydrox...)
Affinity DataIC50: 335nMAssay Description:Inhibition of strand transfer activity of HIV integraseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Gilead Sciences

Curated by ChEMBL
LigandPNGBDBM50187767(ethyl 2-(7-(4-fluorobenzyl)-9-hydroxy-8-oxo-7,8-di...)
Affinity DataIC50: 350nMAssay Description:Inhibition of strand transfer activity of HIV integraseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Gilead Sciences

Curated by ChEMBL
LigandPNGBDBM50187763(7-(4-fluorobenzyl)-9-hydroxy-8-oxo-7,8-dihydro-6H-...)
Affinity DataIC50: 760nMAssay Description:Inhibition of strand transfer activity of HIV integraseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Gilead Sciences

Curated by ChEMBL
LigandPNGBDBM50187758(7-(4-fluorobenzyl)-5-(4-ethoxyphenyl)-9-hydroxy-6,...)
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of strand transfer activity of HIV integraseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Gilead Sciences

Curated by ChEMBL
LigandPNGBDBM50187768(N-(4-fluorobenzyl)-8-hydroxyquinoline-7-carboxamid...)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of strand transfer activity of HIV integraseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Gilead Sciences

Curated by ChEMBL
LigandPNGBDBM50187762(ethyl 3-(7-(4-fluorobenzyl)-9-hydroxy-8-oxo-7,8-di...)
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of strand transfer activity of HIV integraseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Gilead Sciences

Curated by ChEMBL
LigandPNGBDBM50187766(7-(4-fluorobenzyl)-9-hydroxy-6,8-dioxo-7,8-dihydro...)
Affinity DataIC50: 2.40E+3nMAssay Description:Inhibition of strand transfer activity of HIV integraseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed