Compile Data Set for Download or QSAR
Report error Found 5 Enz. Inhib. hit(s) with all data for entry = 50017736
TargetPeroxisome proliferator-activated receptor gamma(Human)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50185944(N-(1-(4-fluorophenyl)-3-(thiophen-2-yl)-1H-pyrazol...)
Affinity DataEC50:  0.780nMAssay Description:Effect on Gal4/PPAR-gamma-LBD construct transactivation in Huh7 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50185943(3-FLUORO-N-[1-(4-FLUOROPHENYL)-3-(2-THIENYL)-1H-PY...)
Affinity DataEC50:  1.75E+3nMAssay Description:Effect on Gal4/PPAR-gamma-LBD construct transactivation in Huh7 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50185944(N-(1-(4-fluorophenyl)-3-(thiophen-2-yl)-1H-pyrazol...)
Affinity DataIC50: 23nMAssay Description:Displacement of [3H]rosiglitazone from PPARgamma by SPAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50185942((N-[1-(4-fluorophenyl)-3-(2-thienyl)-1H-pyrazol-5-...)
Affinity DataIC50: 175nMAssay Description:Displacement of [3H]rosiglitazone from PPARgamma by SPAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50185943(3-FLUORO-N-[1-(4-FLUOROPHENYL)-3-(2-THIENYL)-1H-PY...)
Affinity DataIC50: 512nMAssay Description:Displacement of [3H]rosiglitazone from PPARgamma by SPAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed