Compile Data Set for Download or QSAR
Report error Found 39 Enz. Inhib. hit(s) with all data for entry = 50017687
TargetCytosolic phospholipase A2(Human)
University of MüNster

Curated by ChEMBL
LigandPNGBDBM50185354(3-methylhydrogen 1-[3-(4-decyloxyphenoxy)-2-oxopro...)
Affinity DataIC50: 0.900nMAssay Description:Inhibition of cPLA2-alpha activity assessed by TPA-induced arachidonic acid release in human plateletMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCytosolic phospholipase A2(Human)
University of MüNster

Curated by ChEMBL
LigandPNGBDBM50185348(3-methylhydrogen 1-[3-(4-octylphenoxy)-2-oxopropyl...)
Affinity DataIC50: 1.10nMAssay Description:Inhibition of cPLA2-alpha activity assessed by TPA-induced arachidonic acid release in human plateletMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCytosolic phospholipase A2(Human)
University of MüNster

Curated by ChEMBL
LigandPNGBDBM50185354(3-methylhydrogen 1-[3-(4-decyloxyphenoxy)-2-oxopro...)
Affinity DataIC50: 4.30nMAssay Description:Inhibition of human isolated cPLA2-alpha by vesicle assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCytosolic phospholipase A2(Human)
University of MüNster

Curated by ChEMBL
LigandPNGBDBM50185348(3-methylhydrogen 1-[3-(4-octylphenoxy)-2-oxopropyl...)
Affinity DataIC50: 4.90nMAssay Description:Inhibition of human isolated cPLA2-alpha by vesicle assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCytosolic phospholipase A2(Human)
University of MüNster

Curated by ChEMBL
LigandPNGBDBM50185351(3-acetyl-1-[3-(4-octylphenoxy)-2-oxopropyl]indole-...)
Affinity DataIC50: 6.40nMAssay Description:Inhibition of cPLA2-alpha activity assessed by TPA-induced arachidonic acid release in human plateletMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCytosolic phospholipase A2(Human)
University of MüNster

Curated by ChEMBL
LigandPNGBDBM50185350(1-[3-(4-decyloxyphenoxy)-2-oxopropyl]indole-5-carb...)
Affinity DataIC50: 7.80nMAssay Description:Inhibition of cPLA2-alpha activity assessed by TPA-induced arachidonic acid release in human plateletMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCytosolic phospholipase A2(Human)
University of MüNster

Curated by ChEMBL
LigandPNGBDBM50185349(3-formyl-1-[3-(4-octylphenoxy)-2-oxopropyl]indole-...)
Affinity DataIC50: 9.70nMAssay Description:Inhibition of cPLA2-alpha activity assessed by TPA-induced arachidonic acid release in human plateletMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCytosolic phospholipase A2(Human)
University of MüNster

Curated by ChEMBL
LigandPNGBDBM50185345(3-cyano-1-(3-(4-octylphenoxy)-2-oxopropyl)-1H-indo...)
Affinity DataIC50: 11nMAssay Description:Inhibition of cPLA2-alpha activity assessed by TPA-induced arachidonic acid release in human plateletMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCytosolic phospholipase A2(Human)
University of MüNster

Curated by ChEMBL
LigandPNGBDBM50110846(4-[3-(4-Decyloxy-phenoxy)-2-oxo-propoxy]-benzoic a...)
Affinity DataIC50: 11nMAssay Description:Inhibition of human isolated cPLA2-alpha by vesicle assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCytosolic phospholipase A2(Human)
University of MüNster

Curated by ChEMBL
LigandPNGBDBM50185345(3-cyano-1-(3-(4-octylphenoxy)-2-oxopropyl)-1H-indo...)
Affinity DataIC50: 15nMAssay Description:Inhibition of human isolated cPLA2-alpha by vesicle assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCytosolic phospholipase A2(Human)
University of MüNster

Curated by ChEMBL
LigandPNGBDBM50185351(3-acetyl-1-[3-(4-octylphenoxy)-2-oxopropyl]indole-...)
Affinity DataIC50: 16nMAssay Description:Inhibition of human isolated cPLA2-alpha by vesicle assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCytosolic phospholipase A2(Human)
University of MüNster

Curated by ChEMBL
LigandPNGBDBM50185349(3-formyl-1-[3-(4-octylphenoxy)-2-oxopropyl]indole-...)
Affinity DataIC50: 16nMAssay Description:Inhibition of human isolated cPLA2-alpha by vesicle assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCytosolic phospholipase A2(Human)
University of MüNster

Curated by ChEMBL
LigandPNGBDBM50185356(1-(3-(4-octylphenoxy)-2-oxopropyl)-1H-indole-5-car...)
Affinity DataIC50: 18nMAssay Description:Inhibition of cPLA2-alpha activity assessed by TPA-induced arachidonic acid release in human plateletMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCytosolic phospholipase A2(Human)
University of MüNster

Curated by ChEMBL
LigandPNGBDBM50185350(1-[3-(4-decyloxyphenoxy)-2-oxopropyl]indole-5-carb...)
Affinity DataIC50: 20nMAssay Description:Inhibition of human isolated cPLA2-alpha by vesicle assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCytosolic phospholipase A2(Human)
University of MüNster

Curated by ChEMBL
LigandPNGBDBM50185356(1-(3-(4-octylphenoxy)-2-oxopropyl)-1H-indole-5-car...)
Affinity DataIC50: 35nMAssay Description:Inhibition of human isolated cPLA2-alpha by vesicle assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCytosolic phospholipase A2(Human)
University of MüNster

Curated by ChEMBL
LigandPNGBDBM50185347(3-chloro-1-[3-(4-octylphenoxy)-2-oxopropyl]indole-...)
Affinity DataIC50: 110nMAssay Description:Inhibition of human isolated cPLA2-alpha by vesicle assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCytosolic phospholipase A2(Human)
University of MüNster

Curated by ChEMBL
LigandPNGBDBM50185347(3-chloro-1-[3-(4-octylphenoxy)-2-oxopropyl]indole-...)
Affinity DataIC50: 120nMAssay Description:Inhibition of cPLA2-alpha activity assessed by TPA-induced arachidonic acid release in human plateletMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCytosolic phospholipase A2(Human)
University of MüNster

Curated by ChEMBL
LigandPNGBDBM50185355(1-[3-(4-octylphenoxy)-2-oxopropyl]indole-5-carboxa...)
Affinity DataIC50: 120nMAssay Description:Inhibition of human isolated cPLA2-alpha by vesicle assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCytosolic phospholipase A2(Human)
University of MüNster

Curated by ChEMBL
LigandPNGBDBM50185350(1-[3-(4-decyloxyphenoxy)-2-oxopropyl]indole-5-carb...)
Affinity DataIC50: 210nMAssay Description:Inhibition of cPLA2alpha activity assessed by A23187-induced arachidonic acid release in human plateletMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCytosolic phospholipase A2(Human)
University of MüNster

Curated by ChEMBL
LigandPNGBDBM50185353(3-tert-butyl-1-(3-(4-octylphenoxy)-2-oxopropyl)-1H...)
Affinity DataIC50: 230nMAssay Description:Inhibition of cPLA2-alpha activity assessed by TPA-induced arachidonic acid release in human plateletMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCytosolic phospholipase A2(Human)
University of MüNster

Curated by ChEMBL
LigandPNGBDBM50110846(4-[3-(4-Decyloxy-phenoxy)-2-oxo-propoxy]-benzoic a...)
Affinity DataIC50: 250nMAssay Description:Inhibition of cPLA2alpha activity assessed by A23187-induced arachidonic acid release in human plateletMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCytosolic phospholipase A2(Human)
University of MüNster

Curated by ChEMBL
LigandPNGBDBM50185353(3-tert-butyl-1-(3-(4-octylphenoxy)-2-oxopropyl)-1H...)
Affinity DataIC50: 340nMAssay Description:Inhibition of human isolated cPLA2-alpha by vesicle assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCytosolic phospholipase A2(Human)
University of MüNster

Curated by ChEMBL
LigandPNGBDBM50185345(3-cyano-1-(3-(4-octylphenoxy)-2-oxopropyl)-1H-indo...)
Affinity DataIC50: 370nMAssay Description:Inhibition of cPLA2alpha activity assessed by A23187-induced arachidonic acid release in human plateletMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCytosolic phospholipase A2(Human)
University of MüNster

Curated by ChEMBL
LigandPNGBDBM50185349(3-formyl-1-[3-(4-octylphenoxy)-2-oxopropyl]indole-...)
Affinity DataIC50: 380nMAssay Description:Inhibition of cPLA2alpha activity assessed by A23187-induced arachidonic acid release in human plateletMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCytosolic phospholipase A2(Human)
University of MüNster

Curated by ChEMBL
LigandPNGBDBM50185356(1-(3-(4-octylphenoxy)-2-oxopropyl)-1H-indole-5-car...)
Affinity DataIC50: 410nMAssay Description:Inhibition of cPLA2alpha activity assessed by A23187-induced arachidonic acid release in human plateletMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCytosolic phospholipase A2(Human)
University of MüNster

Curated by ChEMBL
LigandPNGBDBM50185352(1-(3-(4-octylphenoxy)-2-oxopropyl)-1H-indole-3,5-d...)
Affinity DataIC50: 560nMAssay Description:Inhibition of cPLA2-alpha activity assessed by TPA-induced arachidonic acid release in human plateletMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCytosolic phospholipase A2(Human)
University of MüNster

Curated by ChEMBL
LigandPNGBDBM50185354(3-methylhydrogen 1-[3-(4-decyloxyphenoxy)-2-oxopro...)
Affinity DataIC50: 570nMAssay Description:Inhibition of cPLA2alpha activity assessed by A23187-induced arachidonic acid release in human plateletMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCytosolic phospholipase A2(Human)
University of MüNster

Curated by ChEMBL
LigandPNGBDBM50185355(1-[3-(4-octylphenoxy)-2-oxopropyl]indole-5-carboxa...)
Affinity DataIC50: 770nMAssay Description:Inhibition of cPLA2alpha activity assessed by A23187-induced arachidonic acid release in human plateletMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCytosolic phospholipase A2(Human)
University of MüNster

Curated by ChEMBL
LigandPNGBDBM50185352(1-(3-(4-octylphenoxy)-2-oxopropyl)-1H-indole-3,5-d...)
Affinity DataIC50: 890nMAssay Description:Inhibition of human isolated cPLA2-alpha by vesicle assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCytosolic phospholipase A2(Human)
University of MüNster

Curated by ChEMBL
LigandPNGBDBM50185351(3-acetyl-1-[3-(4-octylphenoxy)-2-oxopropyl]indole-...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of cPLA2alpha activity assessed by A23187-induced arachidonic acid release in human plateletMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCytosolic phospholipase A2(Human)
University of MüNster

Curated by ChEMBL
LigandPNGBDBM50185346(1-[3-(4-octylphenoxy)-2-oxopropyl]indole-6-carboxy...)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of human isolated cPLA2-alpha by vesicle assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCytosolic phospholipase A2(Human)
University of MüNster

Curated by ChEMBL
LigandPNGBDBM50185348(3-methylhydrogen 1-[3-(4-octylphenoxy)-2-oxopropyl...)
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of cPLA2alpha activity assessed by A23187-induced arachidonic acid release in human plateletMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCytosolic phospholipase A2(Human)
University of MüNster

Curated by ChEMBL
LigandPNGBDBM50185347(3-chloro-1-[3-(4-octylphenoxy)-2-oxopropyl]indole-...)
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of cPLA2alpha activity assessed by A23187-induced arachidonic acid release in human plateletMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCytosolic phospholipase A2(Human)
University of MüNster

Curated by ChEMBL
LigandPNGBDBM50185353(3-tert-butyl-1-(3-(4-octylphenoxy)-2-oxopropyl)-1H...)
Affinity DataIC50: 3.30E+3nMAssay Description:Inhibition of cPLA2alpha activity assessed by A23187-induced arachidonic acid release in human plateletMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCytosolic phospholipase A2(Human)
University of MüNster

Curated by ChEMBL
LigandPNGBDBM50185357(1-(3-(4-octylphenoxy)-2-oxopropyl)-1H-indole-5-car...)
Affinity DataIC50: 4.30E+3nMAssay Description:Inhibition of human isolated cPLA2-alpha by vesicle assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCytosolic phospholipase A2(Human)
University of MüNster

Curated by ChEMBL
LigandPNGBDBM50185346(1-[3-(4-octylphenoxy)-2-oxopropyl]indole-6-carboxy...)
Affinity DataIC50: 4.70E+3nMAssay Description:Inhibition of cPLA2alpha activity assessed by A23187-induced arachidonic acid release in human plateletMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCytosolic phospholipase A2(Human)
University of MüNster

Curated by ChEMBL
LigandPNGBDBM50185357(1-(3-(4-octylphenoxy)-2-oxopropyl)-1H-indole-5-car...)
Affinity DataIC50: 4.90E+3nMAssay Description:Inhibition of cPLA2alpha activity assessed by A23187-induced arachidonic acid release in human plateletMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCytosolic phospholipase A2(Human)
University of MüNster

Curated by ChEMBL
LigandPNGBDBM50185352(1-(3-(4-octylphenoxy)-2-oxopropyl)-1H-indole-3,5-d...)
Affinity DataIC50: 6.50E+3nMAssay Description:Inhibition of cPLA2alpha activity assessed by A23187-induced arachidonic acid release in human plateletMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCytosolic phospholipase A2(Human)
University of MüNster

Curated by ChEMBL
LigandPNGBDBM50185358(1-[3-(4-octylphenoxy)-2-oxopropyl]indole-2-carboxy...)
Affinity DataIC50: 8.00E+3nMAssay Description:Inhibition of cPLA2alpha activity assessed by A23187-induced arachidonic acid release in human plateletMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed