Compile Data Set for Download or QSAR
Report error Found 7 Enz. Inhib. hit(s) with all data for entry = 50041443
TargetVitamin D3 receptor(Human)
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50262540((3S,5S)-5-((R)-2-((1R,3aS,7aR)-4-(2-((3S,5R)-3,5-d...)
Affinity DataIC50: 207nMAssay Description:Antagonist activity assessed by differentiation of 1,25-D3-induced HL60 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetVitamin D3 receptor(Human)
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50262542((3S,5S)-5-((R)-2-((1R,3aS,7aR)-4-(2-((3S,5R)-3,5-d...)
Affinity DataIC50: 390nMAssay Description:Antagonist activity assessed by differentiation of 1,25-D3-induced HL60 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetVitamin D3 receptor(Human)
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50410853(CHEMBL203485)
Affinity DataIC50: 660nMAssay Description:Antagonist activity assessed by differentiation of 1,25-D3-induced HL60 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetVitamin D3 receptor(Human)
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50262539((3S,5S)-1-benzyl-5-((R)-2-((1R,3aS,7aR)-4-(2-((3S,...)
Affinity DataIC50: 700nMAssay Description:Antagonist activity assessed by differentiation of 1,25-D3-induced HL60 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetVitamin D3 receptor(Human)
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50410854(CHEMBL383450)
Affinity DataIC50: 1.00E+3nMAssay Description:Antagonist activity assessed by differentiation of 1,25-D3-induced HL60 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetVitamin D3 receptor(Human)
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50313152((3R,5S)-5-((R)-2-((1R,3aS,7aR,E)-4-((Z)-2-((3S,5R)...)
Affinity DataIC50: 2.00E+3nMAssay Description:Antagonist activity assessed by differentiation of 1,25-D3-induced HL60 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetVitamin D3 receptor(Human)
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50262541((3S,5S)-5-((R)-2-((1R,3aS,7aR)-4-(2-((3S,5R)-3,5-d...)
Affinity DataIC50: 2.20E+3nMAssay Description:Antagonist activity assessed by differentiation of 1,25-D3-induced HL60 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed