Compile Data Set for Download or QSAR
Report error Found 26 Enz. Inhib. hit(s) with all data for entry = 50000565
TargetMu-type opioid receptor(Rat)
Clinical Research Institute of Montreal

Curated by ChEMBL
LigandPNGBDBM50007327(CHEMBL107580 | 13-[2-Amino-3-(4-hydroxy-phenyl)-pr...)
Affinity DataKi:  0.981nMAssay Description:Displacement of [3H]DAGO from rat brain membrane opioid receptor muMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Clinical Research Institute of Montreal

Curated by ChEMBL
LigandPNGBDBM50007332(CHEMBL321335 | 13-[2-Amino-3-(4-hydroxy-phenyl)-pr...)
Affinity DataKi:  1.70nMAssay Description:Displacement of [3H]DAGO from rat brain membrane opioid receptor muMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Clinical Research Institute of Montreal

Curated by ChEMBL
LigandPNGBDBM50007330(CHEMBL323024 | 13-[2-Amino-3-(4-hydroxy-phenyl)-pr...)
Affinity DataKi:  1.90nMAssay Description:Displacement of [3H]DAGO from rat brain membrane opioid receptor muMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Clinical Research Institute of Montreal

Curated by ChEMBL
LigandPNGBDBM50007329(2-[2-(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propionyl...)
Affinity DataKi:  2.5nMAssay Description:Displacement of [3H]DSLET from rat brain membrane opioid receptor deltaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Clinical Research Institute of Montreal

Curated by ChEMBL
LigandPNGBDBM50007331(CHEMBL263021 | 13-[2-Amino-3-(4-hydroxy-phenyl)-pr...)
Affinity DataKi:  2.60nMAssay Description:Displacement of [3H]DAGO from rat brain membrane opioid receptor muMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Clinical Research Institute of Montreal

Curated by ChEMBL
LigandPNGBDBM50007327(CHEMBL107580 | 13-[2-Amino-3-(4-hydroxy-phenyl)-pr...)
Affinity DataKi:  3.20nMAssay Description:Displacement of [3H]DSLET from rat brain membrane opioid receptor deltaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Clinical Research Institute of Montreal

Curated by ChEMBL
LigandPNGBDBM50007324(CHEMBL106849 | H-Tyr-c[D-Orn-Aic-Glu]-NH2)
Affinity DataKi:  4.20nMAssay Description:Displacement of [3H]DAGO from rat brain membrane opioid receptor muMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Clinical Research Institute of Montreal

Curated by ChEMBL
LigandPNGBDBM50007325(CHEMBL325810 | 13-[2-Amino-3-(4-hydroxy-phenyl)-pr...)
Affinity DataKi:  7.20nMAssay Description:Displacement of [3H]DAGO from rat brain membrane opioid receptor muMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Clinical Research Institute of Montreal

Curated by ChEMBL
LigandPNGBDBM50007326(CHEMBL3037875 | H-Tyr-c[D-Orn-(D or L)Atc-Glu]-NH2)
Affinity DataKi:  8.26nMAssay Description:Displacement of [3H]DSLET from rat brain membrane opioid receptor deltaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Clinical Research Institute of Montreal

Curated by ChEMBL
LigandPNGBDBM50007326(CHEMBL3037875 | H-Tyr-c[D-Orn-(D or L)Atc-Glu]-NH2)
Affinity DataKi:  8.30nMAssay Description:Displacement of [3H]DAGO from rat brain membrane opioid receptor muMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Clinical Research Institute of Montreal

Curated by ChEMBL
LigandPNGBDBM50007330(CHEMBL323024 | 13-[2-Amino-3-(4-hydroxy-phenyl)-pr...)
Affinity DataKi:  9.20nMAssay Description:Displacement of [3H]DSLET from rat brain membrane opioid receptor deltaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Clinical Research Institute of Montreal

Curated by ChEMBL
LigandPNGBDBM50007329(2-[2-(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propionyl...)
Affinity DataKi:  9.40nMAssay Description:Displacement of [3H]DAGO from rat brain membrane opioid receptor muMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Clinical Research Institute of Montreal

Curated by ChEMBL
LigandPNGBDBM50007332(CHEMBL321335 | 13-[2-Amino-3-(4-hydroxy-phenyl)-pr...)
Affinity DataKi:  15nMAssay Description:Displacement of [3H]DSLET from rat brain membrane opioid receptor deltaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Clinical Research Institute of Montreal

Curated by ChEMBL
LigandPNGBDBM50453021(CHEMBL3084310)
Affinity DataKi:  26nMAssay Description:Displacement of [3H]DAGO from rat brain membrane opioid receptor muMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Clinical Research Institute of Montreal

Curated by ChEMBL
LigandPNGBDBM50007331(CHEMBL263021 | 13-[2-Amino-3-(4-hydroxy-phenyl)-pr...)
Affinity DataKi:  51nMAssay Description:Displacement of [3H]DSLET from rat brain membrane opioid receptor deltaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Clinical Research Institute of Montreal

Curated by ChEMBL
LigandPNGBDBM50007325(CHEMBL325810 | 13-[2-Amino-3-(4-hydroxy-phenyl)-pr...)
Affinity DataKi:  55nMAssay Description:Displacement of [3H]DSLET from rat brain membrane opioid receptor deltaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Clinical Research Institute of Montreal

Curated by ChEMBL
LigandPNGBDBM50007324(CHEMBL106849 | H-Tyr-c[D-Orn-Aic-Glu]-NH2)
Affinity DataKi:  209nMAssay Description:Displacement of [3H]DSLET from rat brain membrane opioid receptor deltaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Clinical Research Institute of Montreal

Curated by ChEMBL
LigandPNGBDBM50007334(CHEMBL105453 | 13-[2-Amino-3-(4-hydroxy-phenyl)-pr...)
Affinity DataKi:  258nMAssay Description:Displacement of [3H]DAGO from rat brain membrane opioid receptor muMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Clinical Research Institute of Montreal

Curated by ChEMBL
LigandPNGBDBM50007328(CHEMBL104838 | 13-[2-Amino-3-(4-hydroxy-phenyl)-pr...)
Affinity DataKi:  1.00E+3nMAssay Description:Displacement of [3H]DAGO from rat brain membrane opioid receptor muMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Clinical Research Institute of Montreal

Curated by ChEMBL
LigandPNGBDBM50007323(CHEMBL105568 | 13-[2-Amino-3-(4-hydroxy-phenyl)-pr...)
Affinity DataKi:  1.66E+3nMAssay Description:Displacement of [3H]DAGO from rat brain membrane opioid receptor muMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Clinical Research Institute of Montreal

Curated by ChEMBL
LigandPNGBDBM50007333(CHEMBL107906 | 7-[2-Amino-3-(4-hydroxy-phenyl)-pro...)
Affinity DataKi:  2.41E+3nMAssay Description:Displacement of [3H]DAGO from rat brain membrane opioid receptor muMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Clinical Research Institute of Montreal

Curated by ChEMBL
LigandPNGBDBM50007334(CHEMBL105453 | 13-[2-Amino-3-(4-hydroxy-phenyl)-pr...)
Affinity DataKi:  2.60E+3nMAssay Description:Displacement of [3H]DSLET from rat brain membrane opioid receptor deltaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Clinical Research Institute of Montreal

Curated by ChEMBL
LigandPNGBDBM50453021(CHEMBL3084310)
Affinity DataKi:  3.51E+3nMAssay Description:Displacement of [3H]DSLET from rat brain membrane opioid receptor deltaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Clinical Research Institute of Montreal

Curated by ChEMBL
LigandPNGBDBM50007328(CHEMBL104838 | 13-[2-Amino-3-(4-hydroxy-phenyl)-pr...)
Affinity DataKi:  1.28E+4nMAssay Description:Displacement of [3H]DSLET from rat brain membrane opioid receptor deltaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Clinical Research Institute of Montreal

Curated by ChEMBL
LigandPNGBDBM50007323(CHEMBL105568 | 13-[2-Amino-3-(4-hydroxy-phenyl)-pr...)
Affinity DataKi:  1.40E+4nMAssay Description:Displacement of [3H]DSLET from rat brain membrane opioid receptor deltaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Clinical Research Institute of Montreal

Curated by ChEMBL
LigandPNGBDBM50007333(CHEMBL107906 | 7-[2-Amino-3-(4-hydroxy-phenyl)-pro...)
Affinity DataKi:  5.01E+4nMAssay Description:Displacement of [3H]DSLET from rat brain membrane opioid receptor deltaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed