Compile Data Set for Download or QSAR
Report error Found 23 Enz. Inhib. hit(s) with all data for entry = 50017608
TargetDimer of Tryptase beta-2(Human)
Mochida Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50184499(N-(2-(3-(4-(aminomethyl)phenyl)propylamino)ethyl)-...)
Affinity DataIC50: 5nMAssay Description:Inhibition of human beta tryptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDimer of Tryptase beta-2(Human)
Mochida Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM16127(CHEMBL542712 | AIDS007118 | 2,2 -methanediylbis(1H...)
Affinity DataIC50: 51nMAssay Description:Inhibition of human beta tryptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDimer of Tryptase beta-2(Human)
Mochida Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50184504(N-(2-(3-(4-(aminomethyl)phenyl)propylamino)ethyl)n...)
Affinity DataIC50: 73nMAssay Description:Inhibition of human beta tryptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDimer of Tryptase beta-2(Human)
Mochida Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50184505(N-(2-((3-(4-(aminomethyl)phenyl)propyl)(methyl)ami...)
Affinity DataIC50: 120nMAssay Description:Inhibition of human beta tryptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDimer of Tryptase beta-2(Human)
Mochida Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50184508(N-(2-(3-(4-(aminomethyl)phenyl)propylamino)ethyl)b...)
Affinity DataIC50: 130nMAssay Description:Inhibition of human beta tryptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDimer of Tryptase beta-2(Human)
Mochida Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50184512(N-(2-(3-(4-(aminomethyl)phenyl)propylamino)ethyl)-...)
Affinity DataIC50: 190nMAssay Description:Inhibition of human beta tryptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDimer of Tryptase beta-2(Human)
Mochida Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50184513(N-(2-(3-(4-(aminomethyl)phenyl)propylamino)ethyl)-...)
Affinity DataIC50: 200nMAssay Description:Inhibition of human beta tryptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDimer of Tryptase beta-2(Human)
Mochida Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50184514(N-(2-(3-(4-(aminomethyl)phenyl)propylamino)ethyl)b...)
Affinity DataIC50: 210nMAssay Description:Inhibition of human beta tryptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDimer of Tryptase beta-2(Human)
Mochida Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50184500(N-(2-(3-(4-(aminomethyl)phenyl)propylamino)ethyl)-...)
Affinity DataIC50: 270nMAssay Description:Inhibition of human beta tryptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDimer of Tryptase beta-2(Human)
Mochida Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50184507(N-(2-(3-(4-(aminomethyl)phenyl)propylamino)ethyl)b...)
Affinity DataIC50: 760nMAssay Description:Inhibition of human beta tryptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDimer of Tryptase beta-2(Human)
Mochida Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50184506(N-(2-(4-(aminomethyl)phenethylamino)ethyl)naphthal...)
Affinity DataIC50: 810nMAssay Description:Inhibition of human beta tryptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDimer of Tryptase beta-2(Human)
Mochida Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50184501(N-(3-(4-(aminomethyl)phenyl)propyl)-2-(naphthalene...)
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of human beta tryptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDimer of Tryptase beta-2(Human)
Mochida Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50184503(N-(2-((1-(4-(aminomethyl)phenyl)piperidin-4-yl)met...)
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of human beta tryptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Mochida Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM16127(CHEMBL542712 | AIDS007118 | 2,2 -methanediylbis(1H...)
Affinity DataIC50: 4.50E+3nMAssay Description:Inhibition of F10aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDimer of Tryptase beta-2(Human)
Mochida Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50184509(1-(4-(aminomethyl)phenyl)-N-((1-(naphthalen-2-ylsu...)
Affinity DataIC50: 5.10E+3nMAssay Description:Inhibition of human beta tryptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDimer of Tryptase beta-2(Human)
Mochida Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50184511((4-(4-((4-(naphthalen-2-ylsulfonyl)piperazin-1-yl)...)
Affinity DataIC50: 5.60E+3nMAssay Description:Inhibition of human beta tryptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDimer of Tryptase beta-2(Human)
Mochida Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50184510(N-(2-(3-(4-(aminomethyl)phenyl)propoxy)ethyl)napht...)
Affinity DataIC50: 5.70E+3nMAssay Description:Inhibition of human beta tryptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDimer of Tryptase beta-2(Human)
Mochida Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50184502(N-(1-(4-(aminomethyl)phenyl)piperidin-4-yl)-1-(nap...)
Affinity DataIC50: 2.11E+4nMAssay Description:Inhibition of human beta tryptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlasminogen(Human)
Mochida Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM16127(CHEMBL542712 | AIDS007118 | 2,2 -methanediylbis(1H...)
Affinity DataIC50: 2.60E+4nMAssay Description:Inhibition of plasminMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProthrombin(Human)
Mochida Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM16127(CHEMBL542712 | AIDS007118 | 2,2 -methanediylbis(1H...)
Affinity DataIC50: 3.10E+4nMAssay Description:Inhibition of thrombinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlasminogen(Human)
Mochida Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50184499(N-(2-(3-(4-(aminomethyl)phenyl)propylamino)ethyl)-...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of plasminMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Mochida Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50184499(N-(2-(3-(4-(aminomethyl)phenyl)propylamino)ethyl)-...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of F10aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProthrombin(Human)
Mochida Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50184499(N-(2-(3-(4-(aminomethyl)phenyl)propylamino)ethyl)-...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of thrombinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed