Compile Data Set for Download or QSAR
Report error Found 20 Enz. Inhib. hit(s) with all data for entry = 50017592
TargetIntegrase(Human immunodeficiency virus type 1)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50184349((Z)-4-[6-((Z)-3-carboxy-3-hydroxy-acryloyl)-1-(4-f...)
Affinity DataIC50: 12nMAssay Description:Inhibition of HIV1 integrase strand transfer activity in presence of MnCl2More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50184349((Z)-4-[6-((Z)-3-carboxy-3-hydroxy-acryloyl)-1-(4-f...)
Affinity DataIC50: 16nMAssay Description:Inhibition of HIV1 integrase strand transfer activity in presence of MgCl2 by plate-based electrochemiluminescent assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50184349((Z)-4-[6-((Z)-3-carboxy-3-hydroxy-acryloyl)-1-(4-f...)
Affinity DataIC50: 17nMAssay Description:Inhibition of HIV1 integrase strand transfer activity in presence of MgCl2 by gel-based assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50184349((Z)-4-[6-((Z)-3-carboxy-3-hydroxy-acryloyl)-1-(4-f...)
Affinity DataIC50: 200nMAssay Description:Inhibition of HIV1 integrase 3'-processing activity in presence of MnCl2More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50184346((Z)-4-[6-((Z)-3-ethoxycarbonyl-3-hydroxy-acryloyl)...)
Affinity DataIC50: 250nMAssay Description:Inhibition of HIV1 integrase strand transfer activity in presence of MnCl2More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50184346((Z)-4-[6-((Z)-3-ethoxycarbonyl-3-hydroxy-acryloyl)...)
Affinity DataIC50: 290nMAssay Description:Inhibition of HIV1 integrase strand transfer activity in presence of MgCl2 by gel-based assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50184346((Z)-4-[6-((Z)-3-ethoxycarbonyl-3-hydroxy-acryloyl)...)
Affinity DataIC50: 380nMAssay Description:Inhibition of HIV1 integrase strand transfer activity in presence of MgCl2 by plate-based electrochemiluminescent assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50184347((Z)-4-[6-((Z)-3-carboxy-3-hydroxy-acryloyl)-4-oxo-...)
Affinity DataIC50: 430nMAssay Description:Inhibition of HIV1 integrase strand transfer activity in presence of MnCl2More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50184349((Z)-4-[6-((Z)-3-carboxy-3-hydroxy-acryloyl)-1-(4-f...)
Affinity DataIC50: 440nMAssay Description:Inhibition of HIV1 integrase 3'-processing activity in presence of MgCl2More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50184347((Z)-4-[6-((Z)-3-carboxy-3-hydroxy-acryloyl)-4-oxo-...)
Affinity DataIC50: 2.90E+3nMAssay Description:Inhibition of HIV1 integrase strand transfer activity in presence of MgCl2 by gel-based assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50184347((Z)-4-[6-((Z)-3-carboxy-3-hydroxy-acryloyl)-4-oxo-...)
Affinity DataIC50: 4.10E+3nMAssay Description:Inhibition of HIV1 integrase 3'-processing activity in presence of MnCl2More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50184347((Z)-4-[6-((Z)-3-carboxy-3-hydroxy-acryloyl)-4-oxo-...)
Affinity DataIC50: 9.10E+3nMAssay Description:Inhibition of HIV1 integrase strand transfer activity in presence of MgCl2 by plate-based electrochemiluminescent assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50184346((Z)-4-[6-((Z)-3-ethoxycarbonyl-3-hydroxy-acryloyl)...)
Affinity DataIC50: 2.10E+4nMAssay Description:Inhibition of HIV1 integrase 3'-processing activity in presence of MgCl2More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50184347((Z)-4-[6-((Z)-3-carboxy-3-hydroxy-acryloyl)-4-oxo-...)
Affinity DataIC50: 2.20E+4nMAssay Description:Inhibition of HIV1 integrase 3'-processing activity in presence of MgCl2More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50184348((Z)-4-[6-((Z)-3-ethoxycarbonyl-3-hydroxy-acryloyl)...)
Affinity DataIC50: 2.80E+4nMAssay Description:Inhibition of HIV1 integrase 3'-processing activity in presence of MgCl2More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50184348((Z)-4-[6-((Z)-3-ethoxycarbonyl-3-hydroxy-acryloyl)...)
Affinity DataIC50: 3.90E+4nMAssay Description:Inhibition of HIV1 integrase strand transfer activity in presence of MgCl2 by gel-based assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50184346((Z)-4-[6-((Z)-3-ethoxycarbonyl-3-hydroxy-acryloyl)...)
Affinity DataIC50: 4.00E+4nMAssay Description:Inhibition of HIV1 integrase 3'-processing activity in presence of MnCl2More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50184348((Z)-4-[6-((Z)-3-ethoxycarbonyl-3-hydroxy-acryloyl)...)
Affinity DataIC50: 7.70E+4nMAssay Description:Inhibition of HIV1 integrase strand transfer activity in presence of MgCl2 by plate-based electrochemiluminescent assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50184348((Z)-4-[6-((Z)-3-ethoxycarbonyl-3-hydroxy-acryloyl)...)
Affinity DataIC50: 8.00E+4nMAssay Description:Inhibition of HIV1 integrase strand transfer activity in presence of MnCl2More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50184348((Z)-4-[6-((Z)-3-ethoxycarbonyl-3-hydroxy-acryloyl)...)
Affinity DataIC50: 3.33E+5nMAssay Description:Inhibition of HIV1 integrase 3'-processing activity in presence of MnCl2More data for this Ligand-Target Pair
In DepthDetails Article
PubMed