Compile Data Set for Download or QSAR
Report error Found 24 Enz. Inhib. hit(s) with all data for entry = 50003754
TargetCannabinoid receptor 1(Rat)
University of Kuopio

Curated by ChEMBL
LigandPNGBDBM22988(Arachidonoyl ethanolamide | Arachidonoylethanolami...)
Affinity DataEC50:  1.58E+4nMAssay Description:Displacement of [35S]GTP-gamma-S from rat cerebellar CB1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
University of Kuopio

Curated by ChEMBL
LigandPNGBDBM50072760(3-hydroxy-N-icosa-5,8,11,14-tetraenyl)propanamide ...)
Affinity DataEC50:  7.94E+3nMAssay Description:Displacement of [35S]GTP-gamma-S from rat cerebellar CB1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
University of Kuopio

Curated by ChEMBL
LigandPNGBDBM50072775(ChEMBL_75020 | 5-(1,1-Dimethyl-heptyl)-2-[(1R,2R,5...)
Affinity DataEC50:  100nMAssay Description:Displacement of [35S]GTP-gamma-S from rat cerebellar CB1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetCannabinoid receptor 1(Rat)
University of Kuopio

Curated by ChEMBL
LigandPNGBDBM50006255(CHEMBL418353)
Affinity DataEC50:  398nMAssay Description:Displacement of [35S]GTP-gamma-S from rat cerebellar CB1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
University of Kuopio

Curated by ChEMBL
LigandPNGBDBM50475555(CHEMBL199668)
Affinity DataEC50:  5.01E+4nMAssay Description:Displacement of [35S]GTP-gamma-S from rat cerebellar CB1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
University of Kuopio

Curated by ChEMBL
LigandPNGBDBM50475554(CHEMBL200113)
Affinity DataEC50:  3.98E+4nMAssay Description:Displacement of [35S]GTP-gamma-S from rat cerebellar CB1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
University of Kuopio

Curated by ChEMBL
LigandPNGBDBM50061117(6,6,9-Trimethyl-3-pentyl-6H-benzo[c]chromen-1-ol(C...)
Affinity DataEC50:  316nMAssay Description:Displacement of [35S]GTP-gamma-S from rat cerebellar CB1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
University of Kuopio

Curated by ChEMBL
LigandPNGBDBM50072769(N-(2-chloroethyl)icosa-5,8,11,14-tetraenamide | (5...)
Affinity DataEC50:  316nMAssay Description:Displacement of [35S]GTP-gamma-S from rat cerebellar CB1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
University of Kuopio

Curated by ChEMBL
LigandPNGBDBM50475553(CHEMBL371953)
Affinity DataEC50:  5.01E+4nMAssay Description:Displacement of [35S]GTP-gamma-S from rat cerebellar CB1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
University of Kuopio

Curated by ChEMBL
LigandPNGBDBM50067499((6aR,10aR)-3-(1,1-dimethyl-heptyl)-9-hydroxymethyl...)
Affinity DataEC50:  5nMAssay Description:Displacement of [35S]GTP-gamma-S from rat cerebellar CB1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetCannabinoid receptor 1(Rat)
University of Kuopio

Curated by ChEMBL
LigandPNGBDBM50404269(CHEMBL320549)
Affinity DataEC50:  3.98E+4nMAssay Description:Displacement of [35S]GTP-gamma-S from rat cerebellar CB1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
University of Kuopio

Curated by ChEMBL
LigandPNGBDBM50475552(CHEMBL201758)
Affinity DataEC50:  1.26E+3nMAssay Description:Displacement of [35S]GTP-gamma-S from rat cerebellar CB1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
University of Kuopio

Curated by ChEMBL
LigandPNGBDBM50475547(CHEMBL201260)
Affinity DataEC50:  3.16E+3nMAssay Description:Displacement of [35S]GTP-gamma-S from rat cerebellar CB1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
University of Kuopio

Curated by ChEMBL
LigandPNGBDBM50404270(CHEMBL113473)
Affinity DataEC50:  2.51E+4nMAssay Description:Displacement of [35S]GTP-gamma-S from rat cerebellar CB1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
University of Kuopio

Curated by ChEMBL
LigandPNGBDBM50067740(6-((6aR,10aR)-1-Hydroxy-6,6,9-trimethyl-6a,7,10,10...)
Affinity DataEC50:  10nMAssay Description:Displacement of [35S]GTP-gamma-S from rat cerebellar CB1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
University of Kuopio

Curated by ChEMBL
LigandPNGBDBM50067734(6,6,9-Trimethyl-3-pentyl-6a,7,10,10a-tetrahydro-6H...)
Affinity DataEC50:  631nMAssay Description:Displacement of [35S]GTP-gamma-S from rat cerebellar CB1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
University of Kuopio

Curated by ChEMBL
LigandPNGBDBM50059523(Arachidonyltrifluoromethane | (6Z,9Z,12Z,15Z)-1,1,...)
Affinity DataEC50:  2.51E+4nMAssay Description:Displacement of [35S]GTP-gamma-S from rat cerebellar CB1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
University of Kuopio

Curated by ChEMBL
LigandPNGBDBM50213599((6aR,10aR)-3-(6-bromo-2-methylhexan-2-yl)-6,6,9-tr...)
Affinity DataEC50:  10nMAssay Description:Displacement of [35S]GTP-gamma-S from rat cerebellar CB1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
University of Kuopio

Curated by ChEMBL
LigandPNGBDBM50475551(CHEMBL380923)
Affinity DataEC50:  2.00E+3nMAssay Description:Displacement of [35S]GTP-gamma-S from rat cerebellar CB1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
University of Kuopio

Curated by ChEMBL
LigandPNGBDBM50475550(CHEMBL199911)
Affinity DataEC50:  3.16E+3nMAssay Description:Displacement of [35S]GTP-gamma-S from rat cerebellar CB1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
University of Kuopio

Curated by ChEMBL
LigandPNGBDBM60994((10R,10aR)-6,6,9-Trimethyl-3-pentyl-6a,7,8,10a-tet...)
Affinity DataEC50:  200nMAssay Description:Displacement of [35S]GTP-gamma-S from rat cerebellar CB1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
University of Kuopio

Curated by ChEMBL
LigandPNGBDBM50475549(CHEMBL203474)
Affinity DataEC50:  1.58E+4nMAssay Description:Displacement of [35S]GTP-gamma-S from rat cerebellar CB1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
University of Kuopio

Curated by ChEMBL
LigandPNGBDBM50475548(CHEMBL381893)
Affinity DataEC50:  5.01E+4nMAssay Description:Displacement of [35S]GTP-gamma-S from rat cerebellar CB1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
University of Kuopio

Curated by ChEMBL
LigandPNGBDBM50180036(CHEMBL371214 | (6aR,10aR)-3-(1,1-dimethylbutyl)-6a...)
Affinity DataEC50:  2.00E+3nMAssay Description:Displacement of [35S]GTP-gamma-S from rat cerebellar CB1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed