Compile Data Set for Download or QSAR
Report error Found 55 Enz. Inhib. hit(s) with all data for entry = 1915
LigandPNGBDBM15105(3-[(2S)-2-amino-3-({5-[(E)-2-phenylethenyl]pyridin...)
Affinity DataAssay Description:The kinase assay uses His-Akt1 and a biotinylated peptide as substrate. The biotinylated peptides were immobilized on streptavidin-coated FLASH plat...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM15107(3-[(2S)-2-amino-3-({4-[(E)-2-(pyridin-4-yl)ethenyl...)
Affinity DataAssay Description:The kinase assay uses His-Akt1 and a biotinylated peptide as substrate. The biotinylated peptides were immobilized on streptavidin-coated FLASH plat...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM15106(3-[(2S)-2-amino-3-{3-[(E)-2-(pyridin-4-yl)ethenyl]...)
Affinity DataAssay Description:The kinase assay uses His-Akt1 and a biotinylated peptide as substrate. The biotinylated peptides were immobilized on streptavidin-coated FLASH plat...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM15073((2R)-2-amino-3-({5-[(E)-2-(pyridin-4-yl)ethenyl]py...)
Affinity DatapH: 7.5 T: 2°CAssay Description:The kinase assay uses His-Akt1 and a biotinylated peptide as substrate. The biotinylated peptides were immobilized on streptavidin-coated FLASH plat...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM15099((2S)-2-amino-3-(1H-imidazol-5-yl)-N-{5-[(E)-2-(pyr...)
Affinity DataAssay Description:The kinase assay uses His-Akt1 and a biotinylated peptide as substrate. The biotinylated peptides were immobilized on streptavidin-coated FLASH plat...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM15080((2R)-2-amino-N-(naphthalen-2-yl)-3-({5-[(E)-2-(pyr...)
Affinity DatapH: 7.5 T: 2°CAssay Description:The kinase assay uses His-Akt1 and a biotinylated peptide as substrate. The biotinylated peptides were immobilized on streptavidin-coated FLASH plat...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM15109(3-[(2S)-2-amino-3-phenylpropoxy]-4-[(E)-2-(pyridin...)
Affinity DataAssay Description:The kinase assay uses His-Akt1 and a biotinylated peptide as substrate. The biotinylated peptides were immobilized on streptavidin-coated FLASH plat...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM15097(N-[(2S)-2-amino-3-(1H-indol-3-yl)propyl]-5-[(E)-2-...)
Affinity DataIC50: 9.70nMAssay Description:The kinase assay uses His-Akt1 and a biotinylated peptide as substrate. The biotinylated peptides were immobilized on streptavidin-coated FLASH plat...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM15022(3-[(2S)-2-amino-3-({5-[(E)-2-(pyridin-4-yl)ethenyl...)
Affinity DataIC50: 14nMAssay Description:The kinase assay uses His-Akt1 and a biotinylated peptide as substrate. The biotinylated peptides were immobilized on streptavidin-coated FLASH plat...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM15095(N-[(2S)-2-amino-3-(1H-indol-3-yl)propyl]-6-chloro-...)
Affinity DataIC50: 19nMAssay Description:The kinase assay uses His-Akt1 and a biotinylated peptide as substrate. The biotinylated peptides were immobilized on streptavidin-coated FLASH plat...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM15088(3-[(2S)-2-amino-3-({6-chloro-5-[(E)-2-(pyridin-4-y...)
Affinity DataIC50: 23nMAssay Description:The kinase assay uses His-Akt1 and a biotinylated peptide as substrate. The biotinylated peptides were immobilized on streptavidin-coated FLASH plat...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM15022(3-[(2S)-2-amino-3-({5-[(E)-2-(pyridin-4-yl)ethenyl...)
Affinity DataIC50: 38nMAssay Description:The kinase assay uses purified recombinant enzyme and a biotinylated peptide as substrate. The biotinylated peptides were immobilized on streptavidi...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM15118(4-[(E)-2-{5-[(2S)-2-amino-3-(1H-indol-3-yl)propoxy...)
Affinity DataIC50: 69nMAssay Description:The kinase assay uses His-Akt1 and a biotinylated peptide as substrate. The biotinylated peptides were immobilized on streptavidin-coated FLASH plat...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM15096(N-[(2S)-2-amino-3-(2,3-dihydro-1H-indol-3-yl)propy...)
Affinity DataIC50: 79nMAssay Description:The kinase assay uses His-Akt1 and a biotinylated peptide as substrate. The biotinylated peptides were immobilized on streptavidin-coated FLASH plat...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM15115(4-[(E)-2-{5-[(2S)-2-amino-3-(1H-indol-3-yl)propoxy...)
Affinity DataIC50: 121nMAssay Description:The kinase assay uses His-Akt1 and a biotinylated peptide as substrate. The biotinylated peptides were immobilized on streptavidin-coated FLASH plat...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM15085(3-[(2S)-2-amino-3-(1-benzothiophen-3-yl)propoxy]-5...)
Affinity DataIC50: 142nMAssay Description:The kinase assay uses His-Akt1 and a biotinylated peptide as substrate. The biotinylated peptides were immobilized on streptavidin-coated FLASH plat...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM15084(3-[(2S)-2-amino-3-(naphthalen-2-yl)propoxy]-5-[(E)...)
Affinity DataIC50: 146nMpH: 7.5 T: 2°CAssay Description:The kinase assay uses His-Akt1 and a biotinylated peptide as substrate. The biotinylated peptides were immobilized on streptavidin-coated FLASH plat...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM15119(4-[(E)-2-{5-[(2S)-2-amino-3-(1H-indol-3-yl)propoxy...)
Affinity DataIC50: 147nMAssay Description:The kinase assay uses His-Akt1 and a biotinylated peptide as substrate. The biotinylated peptides were immobilized on streptavidin-coated FLASH plat...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM15117(4-[(E)-2-{5-[(2S)-2-amino-3-(1H-indol-3-yl)propoxy...)
Affinity DataIC50: 163nMAssay Description:The kinase assay uses His-Akt1 and a biotinylated peptide as substrate. The biotinylated peptides were immobilized on streptavidin-coated FLASH plat...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM15116(4-[(E)-2-{5-[(2S)-2-amino-3-(1H-indol-3-yl)propoxy...)
Affinity DataIC50: 176nMAssay Description:The kinase assay uses His-Akt1 and a biotinylated peptide as substrate. The biotinylated peptides were immobilized on streptavidin-coated FLASH plat...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM15094((2R)-4-{6-chloro-5-[(E)-2-(pyridin-4-yl)ethenyl]py...)
Affinity DataIC50: 198nMAssay Description:The kinase assay uses His-Akt1 and a biotinylated peptide as substrate. The biotinylated peptides were immobilized on streptavidin-coated FLASH plat...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRAC-beta serine/threonine-protein kinase(Human)
Abbott Laboratories

LigandPNGBDBM15022(3-[(2S)-2-amino-3-({5-[(E)-2-(pyridin-4-yl)ethenyl...)
Affinity DataIC50: 257nMAssay Description:The kinase assay uses His-Akt1 and a biotinylated peptide as substrate. The biotinylated peptides were immobilized on streptavidin-coated FLASH plat...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM15089(3-[(2S)-2-amino-3-({2-chloro-5-[(E)-2-(pyridin-4-y...)
Affinity DataIC50: 273nMAssay Description:The kinase assay uses His-Akt1 and a biotinylated peptide as substrate. The biotinylated peptides were immobilized on streptavidin-coated FLASH plat...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM15098((2S)-2-amino-3-(1H-indol-3-yl)-N-{5-[(E)-2-(pyridi...)
Affinity DataIC50: 278nMAssay Description:The kinase assay uses His-Akt1 and a biotinylated peptide as substrate. The biotinylated peptides were immobilized on streptavidin-coated FLASH plat...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM15103(2-phenyl-2-{5-[(E)-2-(pyridin-4-yl)ethenyl]pyridin...)
Affinity DataIC50: 284nMAssay Description:The kinase assay uses His-Akt1 and a biotinylated peptide as substrate. The biotinylated peptides were immobilized on streptavidin-coated FLASH plat...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM15082(3-[(2S)-2-amino-3-({5-[(E)-2-(pyridin-4-yl)ethenyl...)
Affinity DataIC50: 320nMpH: 7.5 T: 2°CAssay Description:The kinase assay uses His-Akt1 and a biotinylated peptide as substrate. The biotinylated peptides were immobilized on streptavidin-coated FLASH plat...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM15083(3-[(2S)-2-amino-3-(naphthalen-1-yl)propoxy]-5-[(E)...)
Affinity DataIC50: 324nMpH: 7.5 T: 2°CAssay Description:The kinase assay uses His-Akt1 and a biotinylated peptide as substrate. The biotinylated peptides were immobilized on streptavidin-coated FLASH plat...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRAC-gamma serine/threonine-protein kinase(Human)
Abbott Laboratories

LigandPNGBDBM15022(3-[(2S)-2-amino-3-({5-[(E)-2-(pyridin-4-yl)ethenyl...)
Affinity DataIC50: 354nMAssay Description:The kinase assay uses His-Akt1 and a biotinylated peptide as substrate. The biotinylated peptides were immobilized on streptavidin-coated FLASH plat...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM15087(3-[(2R)-2-amino-3-({5-[(E)-2-(pyridin-4-yl)ethenyl...)
Affinity DataIC50: 360nMAssay Description:The kinase assay uses His-Akt1 and a biotinylated peptide as substrate. The biotinylated peptides were immobilized on streptavidin-coated FLASH plat...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM15090(3-[(2S)-2-amino-3-({5-[(E)-2-(pyridin-4-yl)ethenyl...)
Affinity DataIC50: 500nMAssay Description:The kinase assay uses His-Akt1 and a biotinylated peptide as substrate. The biotinylated peptides were immobilized on streptavidin-coated FLASH plat...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM15101((2S)-2-amino-3-(naphthalen-1-yl)-N-{5-[(E)-2-(pyri...)
Affinity DataIC50: 668nMAssay Description:The kinase assay uses His-Akt1 and a biotinylated peptide as substrate. The biotinylated peptides were immobilized on streptavidin-coated FLASH plat...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM15021(trans-bispyridinylethylene analog 2g | 3-[(2S)-2-a...)
Affinity DataIC50: 690nMpH: 7.5 T: 2°CAssay Description:The kinase assay uses His-Akt1 and a biotinylated peptide as substrate. The biotinylated peptides were immobilized on streptavidin-coated FLASH plat...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM15104(2-(1-methyl-1H-indol-3-yl)-2-{5-[(E)-2-(pyridin-4-...)
Affinity DataIC50: 760nMAssay Description:The kinase assay uses His-Akt1 and a biotinylated peptide as substrate. The biotinylated peptides were immobilized on streptavidin-coated FLASH plat...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM15081(3-[(2S)-2-amino-3-({5-[(E)-2-(pyridin-4-yl)ethenyl...)
Affinity DataIC50: 875nMpH: 7.5 T: 2°CAssay Description:The kinase assay uses His-Akt1 and a biotinylated peptide as substrate. The biotinylated peptides were immobilized on streptavidin-coated FLASH plat...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM15091([(2S)-1-(1H-indol-3-yl)-3-({5-[(E)-2-(pyridin-4-yl...)
Affinity DataIC50: 1.10E+3nMAssay Description:The kinase assay uses His-Akt1 and a biotinylated peptide as substrate. The biotinylated peptides were immobilized on streptavidin-coated FLASH plat...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM15111(3-[(2S)-2-amino-3-({5-[(E)-2-(2-methoxypyridin-4-y...)
Affinity DataIC50: 2.67E+3nMAssay Description:The kinase assay uses His-Akt1 and a biotinylated peptide as substrate. The biotinylated peptides were immobilized on streptavidin-coated FLASH plat...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM15114(3-[(2S)-2-amino-3-({5-[(E)-2-[2-(benzylsulfanyl)py...)
Affinity DataIC50: 3.11E+3nMAssay Description:The kinase assay uses His-Akt1 and a biotinylated peptide as substrate. The biotinylated peptides were immobilized on streptavidin-coated FLASH plat...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM15100((2S)-2-amino-3-phenyl-N-{5-[(E)-2-(pyridin-4-yl)et...)
Affinity DataIC50: 3.20E+3nMAssay Description:The kinase assay uses His-Akt1 and a biotinylated peptide as substrate. The biotinylated peptides were immobilized on streptavidin-coated FLASH plat...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM15120(1-{4-[(E)-2-{5-[(2S)-2-amino-3-(1H-indol-3-yl)prop...)
Affinity DataIC50: 3.34E+3nMAssay Description:The kinase assay uses His-Akt1 and a biotinylated peptide as substrate. The biotinylated peptides were immobilized on streptavidin-coated FLASH plat...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM15079((2S)-1-(benzyloxy)-3-({5-[(E)-2-(pyridin-4-yl)ethe...)
Affinity DataIC50: 4.04E+3nMpH: 7.5 T: 2°CAssay Description:The kinase assay uses His-Akt1 and a biotinylated peptide as substrate. The biotinylated peptides were immobilized on streptavidin-coated FLASH plat...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM15070(3-(2-aminoethoxy)-5-[(E)-2-(pyridin-4-yl)ethenyl]p...)
Affinity DataIC50: 5.08E+3nMpH: 7.5 T: 2°CAssay Description:The kinase assay uses His-Akt1 and a biotinylated peptide as substrate. The biotinylated peptides were immobilized on streptavidin-coated FLASH plat...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM15069(CHEMBL419932 | 5-[(2S)-2-aminopropoxy]-2-chloro-3-...)
Affinity DataIC50: 5.29E+3nMpH: 7.5 T: 2°CAssay Description:The kinase assay uses His-Akt1 and a biotinylated peptide as substrate. The biotinylated peptides were immobilized on streptavidin-coated FLASH plat...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM15113(3-[(2S)-2-amino-3-({5-[(E)-2-[2-(phenylsulfanyl)py...)
Affinity DataIC50: 6.35E+3nMAssay Description:The kinase assay uses His-Akt1 and a biotinylated peptide as substrate. The biotinylated peptides were immobilized on streptavidin-coated FLASH plat...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM15112(3-[(2S)-2-amino-3-({5-[(E)-2-(2-phenoxypyridin-4-y...)
Affinity DataIC50: 6.45E+3nMAssay Description:The kinase assay uses His-Akt1 and a biotinylated peptide as substrate. The biotinylated peptides were immobilized on streptavidin-coated FLASH plat...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM15077(3-[(2S)-2-amino-3,3-diphenylpropoxy]-5-[(E)-2-(pyr...)
Affinity DataIC50: 6.76E+3nMpH: 7.5 T: 2°CAssay Description:The kinase assay uses His-Akt1 and a biotinylated peptide as substrate. The biotinylated peptides were immobilized on streptavidin-coated FLASH plat...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM15078(3-[(2S)-2-amino-4-phenylbutoxy]-5-[(E)-2-(pyridin-...)
Affinity DataIC50: 8.02E+3nMpH: 7.5 T: 2°CAssay Description:The kinase assay uses His-Akt1 and a biotinylated peptide as substrate. The biotinylated peptides were immobilized on streptavidin-coated FLASH plat...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM15074(3-[(2S)-azetidin-2-ylmethoxy]-5-[(E)-2-(pyridin-4-...)
Affinity DataIC50: 1.09E+4nMpH: 7.5 T: 2°CAssay Description:The kinase assay uses His-Akt1 and a biotinylated peptide as substrate. The biotinylated peptides were immobilized on streptavidin-coated FLASH plat...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM15071(3-(3-aminopropoxy)-5-[(E)-2-(pyridin-4-yl)ethenyl]...)
Affinity DataIC50: 1.47E+4nMpH: 7.5 T: 2°CAssay Description:The kinase assay uses His-Akt1 and a biotinylated peptide as substrate. The biotinylated peptides were immobilized on streptavidin-coated FLASH plat...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM15072(3-[(2S)-2-amino-3-methylbutoxy]-5-[(E)-2-(pyridin-...)
Affinity DataIC50: 1.93E+4nMpH: 7.5 T: 2°CAssay Description:The kinase assay uses His-Akt1 and a biotinylated peptide as substrate. The biotinylated peptides were immobilized on streptavidin-coated FLASH plat...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM15108(3-[(2S)-2-amino-3-({6-[(E)-2-(pyridin-4-yl)ethenyl...)
Affinity DataIC50: 2.33E+4nMAssay Description:The kinase assay uses His-Akt1 and a biotinylated peptide as substrate. The biotinylated peptides were immobilized on streptavidin-coated FLASH plat...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Displayed 1 to 50 (of 55 total ) | Next | Last >>
Jump to: