Compile Data Set for Download or QSAR
Report error Found 35 Enz. Inhib. hit(s) with all data for entry = 50017259
LigandPNGBDBM50179795(PVKRRL-(3-Cl)F-NH2 | CHEMBL382690)
Affinity DataIC50: 0.600nMAssay Description:Inhibition of CDK2/CyclinAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50179784(N-((S)-1-((S)-1-(trans-2-(3-chlorophenyl)cyclohexy...)
Affinity DataIC50: 6nMAssay Description:Inhibition of CDK2/CyclinAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50179797(PAKRRLFG | CHEMBL206400)
Affinity DataIC50: 10nMAssay Description:Inhibition of CDK2/CyclinAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50179803(PVKRRLFA | CHEMBL440581)
Affinity DataIC50: 10nMAssay Description:Inhibition of CDK2/CyclinAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50179798(PVKRRLFG | CHEMBL206617)
Affinity DataIC50: 12nMAssay Description:Inhibition of CDK2/CyclinAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50179789(PVKRRLF | CHEMBL381309)
Affinity DataIC50: 14nMAssay Description:Inhibition of CDK2/CyclinAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50179801(AVKRRLFG | CHEMBL381957)
Affinity DataIC50: 16nMAssay Description:Inhibition of CDK2/CyclinAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50179814(N-((S)-1-((S)-1-(trans-2-(3-chlorophenyl)cyclohexy...)
Affinity DataIC50: 21nMAssay Description:Inhibition of CDK2/CyclinAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50179782(PVKRRLF-NH2 | CHEMBL382815)
Affinity DataIC50: 28nMAssay Description:Inhibition of CDK2/CyclinAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50179806(N-((S)-1-((S)-1-(trans-2-(3-chlorophenyl)cyclohexy...)
Affinity DataIC50: 31nMAssay Description:Inhibition of CDK2/CyclinAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50179802(trans-N-((S)-4-methyl-1-oxo-1-(trans-2-phenylcyclo...)
Affinity DataIC50: 40nMAssay Description:Inhibition of CDK2/CyclinAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50179787(N-((S)-1-((S)-1-(trans-2-(3-chlorophenyl)cyclohexy...)
Affinity DataIC50: 47nMAssay Description:Inhibition of CDK2/CyclinAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50179812(N-((S)-1-((S)-1-(trans-2-(3-chlorophenyl)cyclohexy...)
Affinity DataIC50: 58nMAssay Description:Inhibition of CDK2/CyclinAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50179790(PVARRLFG | CHEMBL381396)
Affinity DataIC50: 62nMAssay Description:Inhibition of CDK2/CyclinAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50179796(VKRRLFG | CHEMBL381307)
Affinity DataIC50: 120nMAssay Description:Inhibition of CDK2/CyclinAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50179792(PVKRALFG | CHEMBL206769)
Affinity DataIC50: 130nMAssay Description:Inhibition of CDK2/CyclinAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50179808((S)-2-[(S)-5-guanidino-2-(5-guanidino-pentanoylami...)
Affinity DataIC50: 200nMAssay Description:Inhibition of CDK2/CyclinAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50179805(N-((S)-1-((S)-1-(trans-2-(3-chlorophenyl)cyclohexy...)
Affinity DataIC50: 251nMAssay Description:Inhibition of CDK2/CyclinAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50179780(N-((S)-1-((S)-1-((S)-1-amino-3-(3-chlorophenyl)-1-...)
Affinity DataIC50: 700nMAssay Description:Inhibition of CDK2/CyclinAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50179804(KRRLFG | CHEMBL382403)
Affinity DataIC50: 770nMAssay Description:Inhibition of CDK2/CyclinAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50179811(N-((S)-1-((S)-1-(trans-2-(3-chlorophenyl)cyclohexy...)
Affinity DataIC50: 790nMAssay Description:Inhibition of CDK2/CyclinAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50179785(RRLFG | CHEMBL206763)
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of CDK2/CyclinAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50179807(PVKARLFG | CHEMBL199789)
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of CDK2/CyclinAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50179793(N-((S)-1-((S)-1-((S)-1-amino-3-(3-chlorophenyl)-1-...)
Affinity DataIC50: 2.70E+3nMAssay Description:Inhibition of CDK2/CyclinAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50179783((S)-2-{(S)-5-Guanidino-2-[2-(4-guanidino-phenyl)-a...)
Affinity DataIC50: 2.70E+3nMAssay Description:Inhibition of CDK2/CyclinAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50179786((desNH2)-RRL-(3Cl)F-NH2 | CHEMBL206668)
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of CDK2/CyclinAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50179800((S)-N-((S)-1-(trans-2-(3-chlorophenyl)cyclohexylam...)
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of CDK2/CyclinAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50179810(N-((S)-1-((S)-1-((S)-1-amino-3-(3-chlorophenyl)-1-...)
Affinity DataIC50: 3.30E+3nMAssay Description:Inhibition of CDK2/CyclinAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50179781((S)-2-[(S)-5-Guanidino-2-(5-guanidino-pentanoylami...)
Affinity DataIC50: 4.00E+3nMAssay Description:Inhibition of CDK2/CyclinAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50179813(N-((S)-1-((S)-1-((S)-1-amino-3-(3-chlorophenyl)-1-...)
Affinity DataIC50: 6.90E+3nMAssay Description:Inhibition of CDK2/CyclinAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50179809(PVKRRLAG | CHEMBL203024)
Affinity DataIC50: 8.20E+3nMAssay Description:Inhibition of CDK2/CyclinAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50179791((S)-2-[(S)-5-guanidino-2-(5-guanidino-pentanoylami...)
Affinity DataIC50: 9.00E+3nMAssay Description:Inhibition of CDK2/CyclinAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50179799(1-((1S,5S,9S)-4-(((S)-1-((S)-1-((S)-1-amino-3-(3-c...)
Affinity DataIC50: 1.90E+4nMAssay Description:Inhibition of CDK2/CyclinAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50179788(PVKRRAFG | CHEMBL383664)
Affinity DataIC50: 2.20E+4nMAssay Description:Inhibition of CDK2/CyclinAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50179794(N-((R)-1-((S)-1-(trans-2-(3-chlorophenyl)cyclohexy...)
Affinity DataIC50: 3.10E+4nMAssay Description:Inhibition of CDK2/CyclinAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed