Report error Found 62 Enz. Inhib. hit(s) with all data for entry = 50037630
Affinity DataEC50: 2.55E+4nMAssay Description:Antiproliferative activity mediated by sigma 1 receptor in rat C6 glioma cells by MTT assayMore data for this Ligand-Target Pair
Affinity DataEC50: 4.02E+4nMAssay Description:Antiproliferative activity mediated by sigma 1 receptor in rat C6 glioma cells by MTT assayMore data for this Ligand-Target Pair
Affinity DataEC50: 1.50E+4nMAssay Description:Antiproliferative activity mediated by sigma 1 receptor in rat C6 glioma cells by MTT assayMore data for this Ligand-Target Pair
Affinity DataEC50: 1.94E+4nMAssay Description:Antiproliferative activity mediated by sigma 1 receptor in rat C6 glioma cells by MTT assayMore data for this Ligand-Target Pair
Affinity DataEC50: 1.07E+4nMAssay Description:Antiproliferative activity mediated by sigma 1 receptor in rat C6 glioma cells by MTT assayMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
University of Bari Aldo Moro
Curated by ChEMBL
University of Bari Aldo Moro
Curated by ChEMBL
Affinity DataKi: 0.0300nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membranesMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
University of Bari Aldo Moro
Curated by ChEMBL
University of Bari Aldo Moro
Curated by ChEMBL
Affinity DataKi: 0.240nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membranesMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
University of Bari Aldo Moro
Curated by ChEMBL
University of Bari Aldo Moro
Curated by ChEMBL
Affinity DataKi: 0.300nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membranesMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
University of Bari Aldo Moro
Curated by ChEMBL
University of Bari Aldo Moro
Curated by ChEMBL
Affinity DataKi: 0.350nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membranesMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
University of Bari Aldo Moro
Curated by ChEMBL
University of Bari Aldo Moro
Curated by ChEMBL
Affinity DataKi: 0.360nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membranesMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
University of Bari Aldo Moro
Curated by ChEMBL
University of Bari Aldo Moro
Curated by ChEMBL
Affinity DataKi: 0.420nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membranesMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
University of Bari Aldo Moro
Curated by ChEMBL
University of Bari Aldo Moro
Curated by ChEMBL
Affinity DataKi: 0.5nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membranesMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
University of Bari Aldo Moro
Curated by ChEMBL
University of Bari Aldo Moro
Curated by ChEMBL
Affinity DataKi: 0.660nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membranesMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
University of Bari Aldo Moro
Curated by ChEMBL
University of Bari Aldo Moro
Curated by ChEMBL
Affinity DataKi: 1.01nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membranesMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
University of Bari Aldo Moro
Curated by ChEMBL
University of Bari Aldo Moro
Curated by ChEMBL
Affinity DataKi: 1.03nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membranesMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
University of Bari Aldo Moro
Curated by ChEMBL
University of Bari Aldo Moro
Curated by ChEMBL
Affinity DataKi: 1.14nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membranesMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
University of Bari Aldo Moro
Curated by ChEMBL
University of Bari Aldo Moro
Curated by ChEMBL
Affinity DataKi: 1.18nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membranesMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
University of Bari Aldo Moro
Curated by ChEMBL
University of Bari Aldo Moro
Curated by ChEMBL
Affinity DataKi: 1.20nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membranesMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
University of Bari Aldo Moro
Curated by ChEMBL
University of Bari Aldo Moro
Curated by ChEMBL
Affinity DataKi: 1.35nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membranesMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
University of Bari Aldo Moro
Curated by ChEMBL
University of Bari Aldo Moro
Curated by ChEMBL
Affinity DataKi: 1.43nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membranesMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
University of Bari Aldo Moro
Curated by ChEMBL
University of Bari Aldo Moro
Curated by ChEMBL
Affinity DataKi: 1.47nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membranesMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
University of Bari Aldo Moro
Curated by ChEMBL
University of Bari Aldo Moro
Curated by ChEMBL
Affinity DataKi: 1.5nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membranesMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
University of Bari Aldo Moro
Curated by ChEMBL
University of Bari Aldo Moro
Curated by ChEMBL
Affinity DataKi: 1.78nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membranesMore data for this Ligand-Target Pair
Target3-beta-hydroxysteroid-Delta(8),Delta(7)-isomerase(Guinea pig)
University of Bari Aldo Moro
Curated by ChEMBL
University of Bari Aldo Moro
Curated by ChEMBL
Affinity DataKi: 1.82nMAssay Description:Displacement of [3H](+/-)-emopamil from delta8-delta7 sterol isomerase (SI) site in guinea pig liver membranesMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
University of Bari Aldo Moro
Curated by ChEMBL
University of Bari Aldo Moro
Curated by ChEMBL
Affinity DataKi: 1.83nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membranesMore data for this Ligand-Target Pair
Target3-beta-hydroxysteroid-Delta(8),Delta(7)-isomerase(Guinea pig)
University of Bari Aldo Moro
Curated by ChEMBL
University of Bari Aldo Moro
Curated by ChEMBL
Affinity DataKi: 1.89nMAssay Description:Displacement of [3H](+/-)-emopamil from delta8-delta7 sterol isomerase (SI) site in guinea pig liver membranesMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
University of Bari Aldo Moro
Curated by ChEMBL
University of Bari Aldo Moro
Curated by ChEMBL
Affinity DataKi: 2.25nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membranesMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
University of Bari Aldo Moro
Curated by ChEMBL
University of Bari Aldo Moro
Curated by ChEMBL
Affinity DataKi: 2.80nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membranesMore data for this Ligand-Target Pair
Target3-beta-hydroxysteroid-Delta(8),Delta(7)-isomerase(Guinea pig)
University of Bari Aldo Moro
Curated by ChEMBL
University of Bari Aldo Moro
Curated by ChEMBL
Affinity DataKi: 2.81nMAssay Description:Displacement of [3H](+/-)-emopamil from delta8-delta7 sterol isomerase (SI) site in guinea pig liver membranesMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
University of Bari Aldo Moro
Curated by ChEMBL
University of Bari Aldo Moro
Curated by ChEMBL
Affinity DataKi: 3.32nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membranesMore data for this Ligand-Target Pair
Target3-beta-hydroxysteroid-Delta(8),Delta(7)-isomerase(Guinea pig)
University of Bari Aldo Moro
Curated by ChEMBL
University of Bari Aldo Moro
Curated by ChEMBL
Affinity DataKi: 3.41nMAssay Description:Displacement of [3H](+/-)-emopamil from delta8-delta7 sterol isomerase (SI) site in guinea pig liver membranesMore data for this Ligand-Target Pair
Target3-beta-hydroxysteroid-Delta(8),Delta(7)-isomerase(Guinea pig)
University of Bari Aldo Moro
Curated by ChEMBL
University of Bari Aldo Moro
Curated by ChEMBL
Affinity DataKi: 3.57nMAssay Description:Displacement of [3H](+/-)-emopamil from delta8-delta7 sterol isomerase (SI) site in guinea pig liver membranesMore data for this Ligand-Target Pair
Target3-beta-hydroxysteroid-Delta(8),Delta(7)-isomerase(Guinea pig)
University of Bari Aldo Moro
Curated by ChEMBL
University of Bari Aldo Moro
Curated by ChEMBL
Affinity DataKi: 4.11nMAssay Description:Displacement of [3H](+/-)-emopamil from delta8-delta7 sterol isomerase (SI) site in guinea pig liver membranesMore data for this Ligand-Target Pair
Target3-beta-hydroxysteroid-Delta(8),Delta(7)-isomerase(Guinea pig)
University of Bari Aldo Moro
Curated by ChEMBL
University of Bari Aldo Moro
Curated by ChEMBL
Affinity DataKi: 4.70nMAssay Description:Displacement of [3H](+/-)-emopamil from delta8-delta7 sterol isomerase (SI) site in guinea pig liver membranesMore data for this Ligand-Target Pair
Target3-beta-hydroxysteroid-Delta(8),Delta(7)-isomerase(Guinea pig)
University of Bari Aldo Moro
Curated by ChEMBL
University of Bari Aldo Moro
Curated by ChEMBL
Affinity DataKi: 5.34nMAssay Description:Displacement of [3H](+/-)-emopamil from delta8-delta7 sterol isomerase (SI) site in guinea pig liver membranesMore data for this Ligand-Target Pair
Target3-beta-hydroxysteroid-Delta(8),Delta(7)-isomerase(Guinea pig)
University of Bari Aldo Moro
Curated by ChEMBL
University of Bari Aldo Moro
Curated by ChEMBL
Affinity DataKi: 5.39nMAssay Description:Displacement of [3H](+/-)-emopamil from delta8-delta7 sterol isomerase (SI) site in guinea pig liver membranesMore data for this Ligand-Target Pair
Target3-beta-hydroxysteroid-Delta(8),Delta(7)-isomerase(Guinea pig)
University of Bari Aldo Moro
Curated by ChEMBL
University of Bari Aldo Moro
Curated by ChEMBL
Affinity DataKi: 5.55nMAssay Description:Displacement of [3H](+/-)-emopamil from delta8-delta7 sterol isomerase (SI) site in guinea pig liver membranesMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
University of Bari Aldo Moro
Curated by ChEMBL
University of Bari Aldo Moro
Curated by ChEMBL
Affinity DataKi: 6.16nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membranesMore data for this Ligand-Target Pair
Target3-beta-hydroxysteroid-Delta(8),Delta(7)-isomerase(Guinea pig)
University of Bari Aldo Moro
Curated by ChEMBL
University of Bari Aldo Moro
Curated by ChEMBL
Affinity DataKi: 6.44nMAssay Description:Displacement of [3H](+/-)-emopamil from delta8-delta7 sterol isomerase (SI) site in guinea pig liver membranesMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
University of Bari Aldo Moro
Curated by ChEMBL
University of Bari Aldo Moro
Curated by ChEMBL
Affinity DataKi: 7.05nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membranesMore data for this Ligand-Target Pair
Target3-beta-hydroxysteroid-Delta(8),Delta(7)-isomerase(Guinea pig)
University of Bari Aldo Moro
Curated by ChEMBL
University of Bari Aldo Moro
Curated by ChEMBL
Affinity DataKi: 7.20nMAssay Description:Displacement of [3H](+/-)-emopamil from delta8-delta7 sterol isomerase (SI) site in guinea pig liver membranesMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
University of Bari Aldo Moro
Curated by ChEMBL
University of Bari Aldo Moro
Curated by ChEMBL
Affinity DataKi: 7.80nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membranesMore data for this Ligand-Target Pair
Target3-beta-hydroxysteroid-Delta(8),Delta(7)-isomerase(Guinea pig)
University of Bari Aldo Moro
Curated by ChEMBL
University of Bari Aldo Moro
Curated by ChEMBL
Affinity DataKi: 8.04nMAssay Description:Displacement of [3H](+/-)-emopamil from delta8-delta7 sterol isomerase (SI) site in guinea pig liver membranesMore data for this Ligand-Target Pair
Target3-beta-hydroxysteroid-Delta(8),Delta(7)-isomerase(Guinea pig)
University of Bari Aldo Moro
Curated by ChEMBL
University of Bari Aldo Moro
Curated by ChEMBL
Affinity DataKi: 8.71nMAssay Description:Displacement of [3H](+/-)-emopamil from delta8-delta7 sterol isomerase (SI) site in guinea pig liver membranesMore data for this Ligand-Target Pair
Target3-beta-hydroxysteroid-Delta(8),Delta(7)-isomerase(Guinea pig)
University of Bari Aldo Moro
Curated by ChEMBL
University of Bari Aldo Moro
Curated by ChEMBL
Affinity DataKi: 8.97nMAssay Description:Displacement of [3H](+/-)-emopamil from delta8-delta7 sterol isomerase (SI) site in guinea pig liver membranesMore data for this Ligand-Target Pair
Target3-beta-hydroxysteroid-Delta(8),Delta(7)-isomerase(Guinea pig)
University of Bari Aldo Moro
Curated by ChEMBL
University of Bari Aldo Moro
Curated by ChEMBL
Affinity DataKi: 9.04nMAssay Description:Displacement of [3H](+/-)-emopamil from delta8-delta7 sterol isomerase (SI) site in guinea pig liver membranesMore data for this Ligand-Target Pair
Target3-beta-hydroxysteroid-Delta(8),Delta(7)-isomerase(Guinea pig)
University of Bari Aldo Moro
Curated by ChEMBL
University of Bari Aldo Moro
Curated by ChEMBL
Affinity DataKi: 11.1nMAssay Description:Displacement of [3H](+/-)-emopamil from delta8-delta7 sterol isomerase (SI) site in guinea pig liver membranesMore data for this Ligand-Target Pair
Target3-beta-hydroxysteroid-Delta(8),Delta(7)-isomerase(Guinea pig)
University of Bari Aldo Moro
Curated by ChEMBL
University of Bari Aldo Moro
Curated by ChEMBL
Affinity DataKi: 11.7nMAssay Description:Displacement of [3H](+/-)-emopamil from delta8-delta7 sterol isomerase (SI) site in guinea pig liver membranesMore data for this Ligand-Target Pair
Target3-beta-hydroxysteroid-Delta(8),Delta(7)-isomerase(Guinea pig)
University of Bari Aldo Moro
Curated by ChEMBL
University of Bari Aldo Moro
Curated by ChEMBL
Affinity DataKi: 14.6nMAssay Description:Displacement of [3H](+/-)-emopamil from delta8-delta7 sterol isomerase (SI) site in guinea pig liver membranesMore data for this Ligand-Target Pair
Target3-beta-hydroxysteroid-Delta(8),Delta(7)-isomerase(Guinea pig)
University of Bari Aldo Moro
Curated by ChEMBL
University of Bari Aldo Moro
Curated by ChEMBL
Affinity DataKi: 14.6nMAssay Description:Displacement of [3H](+/-)-emopamil from delta8-delta7 sterol isomerase (SI) site in guinea pig liver membranesMore data for this Ligand-Target Pair
