Compile Data Set for Download or QSAR
Report error Found 32 Enz. Inhib. hit(s) with all data for entry = 50017107
TargetMelanocortin receptor 4(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50177564(N-((R)-3-(4-chlorophenyl)-1-(4-(2-(diethylamino)-1...)
Affinity DataKi:  5.80nMAssay Description:Displacement of [125I]NDP-alpha-MSH from cloned human MC4R expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMelanocortin receptor 4(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50177560(N-((R)-3-(4-chlorophenyl)-1-(4-(1-(2-chlorophenyl)...)
Affinity DataKi:  6.40nMAssay Description:Displacement of [125I]NDP-alpha-MSH from cloned human MC4R expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMelanocortin receptor 4(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50177560(N-((R)-3-(4-chlorophenyl)-1-(4-(1-(2-chlorophenyl)...)
Affinity DataKi:  6.40nMAssay Description:Displacement of [125I]NDP-alpha-MSH from cloned human MC4R expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMelanocortin receptor 4(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50177563(N-((R)-3-(4-chlorophenyl)-1-(4-(2-(diethylamino)-1...)
Affinity DataKi:  7.30nMAssay Description:Displacement of [125I]NDP-alpha-MSH from cloned human MC4R expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMelanocortin receptor 4(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50177557(N-((R)-3-(4-chlorophenyl)-1-(4-(2-(diethylamino)-1...)
Affinity DataKi:  10nMAssay Description:Displacement of [125I]NDP-alpha-MSH from cloned human MC4R expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMelanocortin receptor 4(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50177565(N-((R)-3-(4-chlorophenyl)-1-(4-(2-(diethylamino)-1...)
Affinity DataKi:  17nMAssay Description:Displacement of [125I]NDP-alpha-MSH from cloned human MC4R expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMelanocortin receptor 4(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50177561((R)-N-((R)-3-(4-chlorophenyl)-1-(4-(2-(diethylamin...)
Affinity DataKi:  41nMAssay Description:Displacement of [125I]NDP-alpha-MSH from cloned human MC4R expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMelanocortin receptor 4(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50177558(N-((R)-3-(4-chlorophenyl)-1-(4-(2-(diethylamino)-1...)
Affinity DataKi:  74nMAssay Description:Displacement of [125I]NDP-alpha-MSH from cloned human MC4R expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMelanocortin receptor 4(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50177562(N-((R)-3-(4-chlorophenyl)-1-(4-(2-(diethylamino)-1...)
Affinity DataKi:  96nMAssay Description:Displacement of [125I]NDP-alpha-MSH from cloned human MC4R expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMelanocortin receptor 4(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50177559(N-((R)-3-(4-chlorophenyl)-1-(4-(1-(2-chlorophenyl)...)
Affinity DataKi:  107nMAssay Description:Displacement of [125I]NDP-alpha-MSH from cloned human MC4R expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMelanocortin receptor 4(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50177559(N-((R)-3-(4-chlorophenyl)-1-(4-(1-(2-chlorophenyl)...)
Affinity DataKi:  107nMAssay Description:Displacement of [125I]NDP-alpha-MSH from cloned human MC4R expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMelanocortin receptor 5(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50177564(N-((R)-3-(4-chlorophenyl)-1-(4-(2-(diethylamino)-1...)
Affinity DataKi:  420nMAssay Description:Displacement of [125I]NDP-alpha-MSH from cloned human MC5R expressed in HEK293 cellMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMelanocortin receptor 5(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50177557(N-((R)-3-(4-chlorophenyl)-1-(4-(2-(diethylamino)-1...)
Affinity DataKi:  910nMAssay Description:Displacement of [125I]NDP-alpha-MSH from cloned human MC5R expressed in HEK293 cellMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMelanocortin receptor 5(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50177562(N-((R)-3-(4-chlorophenyl)-1-(4-(2-(diethylamino)-1...)
Affinity DataKi:  920nMAssay Description:Displacement of [125I]NDP-alpha-MSH from cloned human MC5R expressed in HEK293 cellMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMelanocortin receptor 5(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50177561((R)-N-((R)-3-(4-chlorophenyl)-1-(4-(2-(diethylamin...)
Affinity DataKi:  950nMAssay Description:Displacement of [125I]NDP-alpha-MSH from cloned human MC5R expressed in HEK293 cellMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMelanocortin receptor 5(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50177563(N-((R)-3-(4-chlorophenyl)-1-(4-(2-(diethylamino)-1...)
Affinity DataKi:  1.20E+3nMAssay Description:Displacement of [125I]NDP-alpha-MSH from cloned human MC5R expressed in HEK293 cellMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMelanocortin receptor 3(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50177562(N-((R)-3-(4-chlorophenyl)-1-(4-(2-(diethylamino)-1...)
Affinity DataKi:  1.40E+3nMAssay Description:Displacement of [125I]NDP-alpha-MSH from cloned human MC3R expressed in HEK293 cellMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMelanocortin receptor 5(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50177558(N-((R)-3-(4-chlorophenyl)-1-(4-(2-(diethylamino)-1...)
Affinity DataKi:  1.40E+3nMAssay Description:Displacement of [125I]NDP-alpha-MSH from cloned human MC5R expressed in HEK293 cellMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMelanocortin receptor 3(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50177564(N-((R)-3-(4-chlorophenyl)-1-(4-(2-(diethylamino)-1...)
Affinity DataKi:  1.90E+3nMAssay Description:Displacement of [125I]NDP-alpha-MSH from cloned human MC3R expressed in HEK293 cellMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMelanocortin receptor 5(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50177565(N-((R)-3-(4-chlorophenyl)-1-(4-(2-(diethylamino)-1...)
Affinity DataKi:  2.00E+3nMAssay Description:Displacement of [125I]NDP-alpha-MSH from cloned human MC5R expressed in HEK293 cellMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50177557(N-((R)-3-(4-chlorophenyl)-1-(4-(2-(diethylamino)-1...)
Affinity DataKi:  3.00E+3nMAssay Description:Displacement of [125I]NDP-alpha-MSH from cloned human MC1R expressed in HEK293 cellMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMelanocortin receptor 3(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50177563(N-((R)-3-(4-chlorophenyl)-1-(4-(2-(diethylamino)-1...)
Affinity DataKi:  3.40E+3nMAssay Description:Displacement of [125I]NDP-alpha-MSH from cloned human MC3R expressed in HEK293 cellMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMelanocortin receptor 3(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50177557(N-((R)-3-(4-chlorophenyl)-1-(4-(2-(diethylamino)-1...)
Affinity DataKi:  4.20E+3nMAssay Description:Displacement of [125I]NDP-alpha-MSH from cloned human MC3R expressed in HEK293 cellMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMelanocortin receptor 3(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50177565(N-((R)-3-(4-chlorophenyl)-1-(4-(2-(diethylamino)-1...)
Affinity DataKi:  4.60E+3nMAssay Description:Displacement of [125I]NDP-alpha-MSH from cloned human MC3R expressed in HEK293 cellMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50177561((R)-N-((R)-3-(4-chlorophenyl)-1-(4-(2-(diethylamin...)
Affinity DataKi:  5.80E+3nMAssay Description:Displacement of [125I]NDP-alpha-MSH from cloned human MC1R expressed in HEK293 cellMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50177563(N-((R)-3-(4-chlorophenyl)-1-(4-(2-(diethylamino)-1...)
Affinity DataKi:  6.00E+3nMAssay Description:Displacement of [125I]NDP-alpha-MSH from cloned human MC1R expressed in HEK293 cellMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50177562(N-((R)-3-(4-chlorophenyl)-1-(4-(2-(diethylamino)-1...)
Affinity DataKi:  7.00E+3nMAssay Description:Displacement of [125I]NDP-alpha-MSH from cloned human MC1R expressed in HEK293 cellMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMelanocortin receptor 3(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50177561((R)-N-((R)-3-(4-chlorophenyl)-1-(4-(2-(diethylamin...)
Affinity DataKi:  7.00E+3nMAssay Description:Displacement of [125I]NDP-alpha-MSH from cloned human MC3R expressed in HEK293 cellMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50177564(N-((R)-3-(4-chlorophenyl)-1-(4-(2-(diethylamino)-1...)
Affinity DataKi:  7.00E+3nMAssay Description:Displacement of [125I]NDP-alpha-MSH from cloned human MC1R expressed in HEK293 cellMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50177565(N-((R)-3-(4-chlorophenyl)-1-(4-(2-(diethylamino)-1...)
Affinity DataKi:  8.60E+3nMAssay Description:Displacement of [125I]NDP-alpha-MSH from cloned human MC1R expressed in HEK293 cellMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMelanocortin receptor 3(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50177558(N-((R)-3-(4-chlorophenyl)-1-(4-(2-(diethylamino)-1...)
Affinity DataKi:  1.60E+4nMAssay Description:Displacement of [125I]NDP-alpha-MSH from cloned human MC3R expressed in HEK293 cellMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50177558(N-((R)-3-(4-chlorophenyl)-1-(4-(2-(diethylamino)-1...)
Affinity DataKi:  2.00E+4nMAssay Description:Displacement of [125I]NDP-alpha-MSH from cloned human MC1R expressed in HEK293 cellMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed