Compile Data Set for Download or QSAR
Report error Found 46 Enz. Inhib. hit(s) with all data for entry = 50016744
TargetVascular endothelial growth factor receptor 2(Human)
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50173019(4-[4-(4-tert-Butyl-phenylamino)-phthalazin-1-yl]-b...)
Affinity DataIC50: 78nMAssay Description:Inhibition of Vascular endothelial growth factor receptor 2 kinase phosphorylation of pGAT-biotin peptideMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50173031(4-(4-(4-bromophenylamino)phthalazin-1-yl)benzamide...)
Affinity DataIC50: 100nMAssay Description:Inhibition of Vascular endothelial growth factor receptor 2 kinase phosphorylation of pGAT-biotin peptideMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50173045(4-(4-(4-tert-butylphenylamino)phthalazin-1-yl)-N-m...)
Affinity DataIC50: 130nMAssay Description:Inhibition of Vascular endothelial growth factor receptor 2 kinase phosphorylation of pGAT-biotin peptideMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50173049(4-{4-[4-(Chloro-difluoro-methoxy)-phenylamino]-pht...)
Affinity DataIC50: 190nMAssay Description:Inhibition of Vascular endothelial growth factor receptor 2 kinase phosphorylation of pGAT-biotin peptideMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50173007(4-[4-(4-Chloro-phenylamino)-phthalazin-1-yl]-benzo...)
Affinity DataIC50: 360nMAssay Description:Inhibition of Vascular endothelial growth factor receptor 2 kinase phosphorylation of pGAT-biotin peptideMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50173022(3-[4-(4-tert-Butyl-phenylamino)-phthalazin-1-yl]-b...)
Affinity DataIC50: 400nMAssay Description:Inhibition of Vascular endothelial growth factor receptor 2 kinase phosphorylation of pGAT-biotin peptideMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50173034(4-(4-(3-tert-butylphenylamino)phthalazin-1-yl)benz...)
Affinity DataIC50: 470nMAssay Description:Inhibition of Vascular endothelial growth factor receptor 2 kinase phosphorylation of pGAT-biotin peptideMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50173021(4-{4-[4-(Chloro-difluoro-methoxy)-phenylamino]-pht...)
Affinity DataIC50: 630nMAssay Description:Inhibition of Vascular endothelial growth factor receptor 2 kinase phosphorylation of pGAT-biotin peptideMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50173051(4-(4-(3,4-dichlorophenylamino)phthalazin-1-yl)benz...)
Affinity DataIC50: 840nMAssay Description:Inhibition of Vascular endothelial growth factor receptor 2 kinase phosphorylation of pGAT-biotin peptideMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50173024(4-(4-(4-(chlorodifluoromethoxy)phenylamino)phthala...)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of Vascular endothelial growth factor receptor 2 kinase phosphorylation of pGAT-biotin peptideMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50173041(3,5-dimethoxy-N-(1-(naphthalen-2-ylmethyl)piperidi...)
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of Vascular endothelial growth factor receptor 2 kinase phosphorylation of pGAT-biotin peptideMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50173011(4-(4-(4-chlorophenylamino)phthalazin-1-yl)benzamid...)
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of Vascular endothelial growth factor receptor 2 kinase phosphorylation of pGAT-biotin peptideMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50173029(4-(4-m-Tolylamino-phthalazin-1-yl)-benzamide | 4-(...)
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of Vascular endothelial growth factor receptor 2 kinase phosphorylation of pGAT-biotin peptideMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50173012(4-[4-(3-Chloro-phenylamino)-phthalazin-1-yl]-benza...)
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of Vascular endothelial growth factor receptor 2 kinase phosphorylation of pGAT-biotin peptideMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50173017(4-(4-(p-tolylamino)phthalazin-1-yl)benzamide | 4-(...)
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of Vascular endothelial growth factor receptor 2 kinase phosphorylation of pGAT-biotin peptideMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50173043(4-[4-(4-Methoxy-phenylamino)-phthalazin-1-yl]-benz...)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of Vascular endothelial growth factor receptor 2 kinase phosphorylation of pGAT-biotin peptideMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50173025(methyl 4-(4-(4-carbamoylphenyl)phthalazin-1-ylamin...)
Affinity DataIC50: 2.70E+3nMAssay Description:Inhibition of Vascular endothelial growth factor receptor 2 kinase phosphorylation of pGAT-biotin peptideMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50173013(4-[4-(4-Chloro-phenylamino)-phthalazin-1-yl]-N-met...)
Affinity DataIC50: 3.10E+3nMAssay Description:Inhibition of Vascular endothelial growth factor receptor 2 kinase phosphorylation of pGAT-biotin peptideMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50173047(3-{4-[4-(Chloro-difluoro-methoxy)-phenylamino]-pht...)
Affinity DataIC50: 4.10E+3nMAssay Description:Inhibition of Vascular endothelial growth factor receptor 2 kinase phosphorylation of pGAT-biotin peptideMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50173020((4-{4-[4-(Chloro-difluoro-methoxy)-phenylamino]-ph...)
Affinity DataIC50: 4.90E+3nMAssay Description:Inhibition of Vascular endothelial growth factor receptor 2 kinase phosphorylation of pGAT-biotin peptideMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50173040(4-[4-(2,4-Dimethyl-phenylamino)-phthalazin-1-yl]-b...)
Affinity DataIC50: 6.90E+3nMAssay Description:Inhibition of Vascular endothelial growth factor receptor 2 kinase phosphorylation of pGAT-biotin peptideMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50173030(4-[4-(4-Sulfamoyl-phenylamino)-phthalazin-1-yl]-be...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of Vascular endothelial growth factor receptor 2 kinase phosphorylation of pGAT-biotin peptideMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50173044([4-(Chloro-difluoro-methoxy)-phenyl]-[4-(4-chloro-...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of Vascular endothelial growth factor receptor 2 kinase phosphorylation of pGAT-biotin peptideMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50173036(4-[4-(4-Pyridin-1-yl-phenylamino)-phthalazin-1-yl]...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of Vascular endothelial growth factor receptor 2 kinase phosphorylation of pGAT-biotin peptideMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50173046([4-(4-Ethoxy-phenyl)-phthalazin-1-yl]-(4-methoxy-p...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of Vascular endothelial growth factor receptor 2 kinase phosphorylation of pGAT-biotin peptideMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50173038((3,4-Dichloro-phenyl)-(4-p-tolyl-phthalazin-1-yl)-...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of Vascular endothelial growth factor receptor 2 kinase phosphorylation of pGAT-biotin peptideMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50173042(4-[4-(4-carbamoylanilino)-1-phthalazinyl]benzamide...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of Vascular endothelial growth factor receptor 2 kinase phosphorylation of pGAT-biotin peptideMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50173048(5-{4-[4-(Chloro-difluoro-methoxy)-phenylamino]-pht...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of Vascular endothelial growth factor receptor 2 kinase phosphorylation of pGAT-biotin peptideMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50173050(4-(4-(4-(trifluoromethoxy)phenylthio)phthalazin-1-...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of Vascular endothelial growth factor receptor 2 kinase phosphorylation of pGAT-biotin peptideMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50173052(5-{4-[4-(Chloro-difluoro-methoxy)-phenylamino]-pht...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of Vascular endothelial growth factor receptor 2 kinase phosphorylation of pGAT-biotin peptideMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50173039((4-Chloro-phenyl)-(4-p-tolyl-phthalazin-1-yl)-amin...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of Vascular endothelial growth factor receptor 2 kinase phosphorylation of pGAT-biotin peptideMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50173037([4-(Chloro-difluoro-methoxy)-phenyl]-(4-phenyl-pht...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of Vascular endothelial growth factor receptor 2 kinase phosphorylation of pGAT-biotin peptideMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50173035((4-Chloro-phenyl)-[4-(4-ethoxy-phenyl)-phthalazin-...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of Vascular endothelial growth factor receptor 2 kinase phosphorylation of pGAT-biotin peptideMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50173033((3,4-Dichloro-phenyl)-[4-(4-methoxy-phenyl)-phthal...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of Vascular endothelial growth factor receptor 2 kinase phosphorylation of pGAT-biotin peptideMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50173027(N,N-Dimethyl-4-(4-p-tolylamino-phthalazin-1-yl)-be...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of Vascular endothelial growth factor receptor 2 kinase phosphorylation of pGAT-biotin peptideMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50173028(4-[4-(4-Benzyloxy-phenylamino)-phthalazin-1-yl]-be...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of Vascular endothelial growth factor receptor 2 kinase phosphorylation of pGAT-biotin peptideMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50173032(4-[4-(4-Morpholin-4-yl-phenylamino)-phthalazin-1-y...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of Vascular endothelial growth factor receptor 2 kinase phosphorylation of pGAT-biotin peptideMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50173026([4-(4-Ethoxy-phenyl)-phthalazin-1-yl]-p-tolyl-amin...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of Vascular endothelial growth factor receptor 2 kinase phosphorylation of pGAT-biotin peptideMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50173023((4-Methoxy-phenyl)-(4-phenyl-phthalazin-1-yl)-amin...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of Vascular endothelial growth factor receptor 2 kinase phosphorylation of pGAT-biotin peptideMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50173018([4-(Chloro-difluoro-methoxy)-phenyl]-[4-(4-methoxy...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of Vascular endothelial growth factor receptor 2 kinase phosphorylation of pGAT-biotin peptideMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50173015(N-tert-butyl-4-(4-(4-(chlorodifluoromethoxy)phenyl...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of Vascular endothelial growth factor receptor 2 kinase phosphorylation of pGAT-biotin peptideMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50173016(4-(4-(phenylamino)phthalazin-1-yl)benzamide | 4-(4...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of Vascular endothelial growth factor receptor 2 kinase phosphorylation of pGAT-biotin peptideMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50173014([4-(Chloro-difluoro-methoxy)-phenyl]-(4-p-tolyl-ph...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of Vascular endothelial growth factor receptor 2 kinase phosphorylation of pGAT-biotin peptideMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50173010((4-Chloro-phenyl)-[4-(4-methoxy-phenyl)-phthalazin...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of Vascular endothelial growth factor receptor 2 kinase phosphorylation of pGAT-biotin peptideMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50173008(4-[4-(4-Trifluoromethoxy-phenoxy)-phthalazin-1-yl]...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of Vascular endothelial growth factor receptor 2 kinase phosphorylation of pGAT-biotin peptideMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50173009(4-(4-(4-(chlorodifluoromethoxy)phenylamino)phthala...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of Vascular endothelial growth factor receptor 2 kinase phosphorylation of pGAT-biotin peptideMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed