Compile Data Set for Download or QSAR
Report error Found 10 Enz. Inhib. hit(s) with all data for entry = 50016689
TargetMu-type opioid receptor(Guinea pig)
University of Cagliari

Curated by ChEMBL
LigandPNGBDBM50172014(H-Dmt-D-Arg(NO2)-Phe-Lys(Z)-NH2 | CHEMBL371856)
Affinity DataIC50: 0.509nMAssay Description:Agonist activity against mu opioid receptor of guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
University of Cagliari

Curated by ChEMBL
LigandPNGBDBM50010483(CHEMBL2181202)
Affinity DataIC50: 1.40nMAssay Description:Agonist activity against mu opioid receptor of guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDelta-type opioid receptor(Mouse)
University of Cagliari

Curated by ChEMBL
LigandPNGBDBM50172014(H-Dmt-D-Arg(NO2)-Phe-Lys(Z)-NH2 | CHEMBL371856)
Affinity DataIC50: 1.70nMAssay Description:Agonistic activity against delta opioid receptor of mouse vas deferens assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDelta-type opioid receptor(Mouse)
University of Cagliari

Curated by ChEMBL
LigandPNGBDBM50010483(CHEMBL2181202)
Affinity DataIC50: 23nMAssay Description:Agonistic activity against delta opioid receptor of mouse vas deferens assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
University of Cagliari

Curated by ChEMBL
LigandPNGBDBM50172013(H-Dmt-D-Arg(NO2)-Phe-Lys(Z)-OH | CHEMBL370701)
Affinity DataIC50: 63nMAssay Description:Agonist activity against mu opioid receptor of guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDelta-type opioid receptor(Mouse)
University of Cagliari

Curated by ChEMBL
LigandPNGBDBM50172013(H-Dmt-D-Arg(NO2)-Phe-Lys(Z)-OH | CHEMBL370701)
Affinity DataIC50: 682nMAssay Description:Agonistic activity against delta opioid receptor of mouse vas deferens assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
University of Cagliari

Curated by ChEMBL
LigandPNGBDBM50172017({(S)-5-[(S)-2-({2-[2-Amino-3-(4-hydroxy-2,6-dimeth...)
Affinity DataIC50: 1.89E+3nMAssay Description:Agonist activity against mu opioid receptor of guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDelta-type opioid receptor(Mouse)
University of Cagliari

Curated by ChEMBL
LigandPNGBDBM50172017({(S)-5-[(S)-2-({2-[2-Amino-3-(4-hydroxy-2,6-dimeth...)
Affinity DataIC50: 1.00E+4nMAssay Description:Agonistic activity against delta opioid receptor of mouse vas deferens assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDelta-type opioid receptor(Mouse)
University of Cagliari

Curated by ChEMBL
LigandPNGBDBM50172015((S)-2-[(S)-2-({2-[2-Amino-3-(4-hydroxy-2,6-dimethy...)
Affinity DataIC50: 1.00E+4nMAssay Description:Agonistic activity against delta opioid receptor of mouse vas deferens assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
University of Cagliari

Curated by ChEMBL
LigandPNGBDBM50172015((S)-2-[(S)-2-({2-[2-Amino-3-(4-hydroxy-2,6-dimethy...)
Affinity DataIC50: 1.00E+4nMAssay Description:Agonist activity against mu opioid receptor of guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed