Compile Data Set for Download or QSAR
Report error Found 20 Enz. Inhib. hit(s) with all data for entry = 50024708
TargetMuscarinic acetylcholine receptor M3(Human)
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50241913(nocardimicin B | GNF-PF-5618 | CHEMBL499519)
Affinity DataIC50: 630nMAssay Description:Displacement of [3H]NMS from human muscarinic M3 receptor expressed in insect Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M4(Human)
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50241913(nocardimicin B | GNF-PF-5618 | CHEMBL499519)
Affinity DataIC50: 1.04E+3nMAssay Description:Binding affinity to human muscarinic M4 receptor expressed in insect Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M3(Human)
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50241915(nocardimicin D | CHEMBL450986)
Affinity DataIC50: 1.10E+3nMAssay Description:Displacement of [3H]NMS from human muscarinic M3 receptor expressed in insect Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M5(Human)
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50241913(nocardimicin B | GNF-PF-5618 | CHEMBL499519)
Affinity DataIC50: 1.64E+3nMAssay Description:Binding affinity to human muscarinic M5 receptor expressed in insect Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Human)
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50241913(nocardimicin B | GNF-PF-5618 | CHEMBL499519)
Affinity DataIC50: 1.78E+3nMAssay Description:Binding affinity to human muscarinic M2 receptor expressed in insect Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50241913(nocardimicin B | GNF-PF-5618 | CHEMBL499519)
Affinity DataIC50: 2.03E+3nMAssay Description:Binding affinity to human muscarinic M1 receptor expressed in insect Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M3(Human)
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50241916(Noccardimicin E | CHEMBL510340)
Affinity DataIC50: 4.56E+3nMAssay Description:Displacement of [3H]NMS from human muscarinic M3 receptor expressed in insect Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M3(Human)
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50241914(nocardimicin C | CHEMBL507760)
Affinity DataIC50: 4.70E+3nMAssay Description:Displacement of [3H]NMS from human muscarinic M3 receptor expressed in insect Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M3(Human)
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50241912(Nocardimicin A | CHEMBL505197)
Affinity DataIC50: 5.89E+3nMAssay Description:Displacement of [3H]NMS from human muscarinic M3 receptor expressed in insect Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M3(Human)
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50241917(Nocardimicin F | CHEMBL508807)
Affinity DataIC50: 6.29E+3nMAssay Description:Displacement of [3H]NMS from human muscarinic M3 receptor expressed in insect Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M3(Human)
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50241913(nocardimicin B | GNF-PF-5618 | CHEMBL499519)
Affinity DataKi:  130nMAssay Description:Displacement of [3H]NMS from human muscarinic M3 receptor expressed in insect Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M4(Human)
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50241913(nocardimicin B | GNF-PF-5618 | CHEMBL499519)
Affinity DataKi:  140nMAssay Description:Binding affinity to human muscarinic M4 receptor expressed in insect Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M3(Human)
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50241915(nocardimicin D | CHEMBL450986)
Affinity DataKi:  230nMAssay Description:Displacement of [3H]NMS from human muscarinic M3 receptor expressed in insect Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50241913(nocardimicin B | GNF-PF-5618 | CHEMBL499519)
Affinity DataKi:  490nMAssay Description:Binding affinity to human muscarinic M1 receptor expressed in insect Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Human)
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50241913(nocardimicin B | GNF-PF-5618 | CHEMBL499519)
Affinity DataKi:  630nMAssay Description:Binding affinity to human muscarinic M2 receptor expressed in insect Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M3(Human)
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50241916(Noccardimicin E | CHEMBL510340)
Affinity DataKi:  970nMAssay Description:Displacement of [3H]NMS from human muscarinic M3 receptor expressed in insect Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M3(Human)
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50241914(nocardimicin C | CHEMBL507760)
Affinity DataKi:  1.00E+3nMAssay Description:Displacement of [3H]NMS from human muscarinic M3 receptor expressed in insect Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M5(Human)
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50241913(nocardimicin B | GNF-PF-5618 | CHEMBL499519)
Affinity DataKi:  1.18E+3nMAssay Description:Binding affinity to human muscarinic M5 receptor expressed in insect Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M3(Human)
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50241912(Nocardimicin A | CHEMBL505197)
Affinity DataKi:  1.25E+3nMAssay Description:Displacement of [3H]NMS from human muscarinic M3 receptor expressed in insect Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M3(Human)
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50241917(Nocardimicin F | CHEMBL508807)
Affinity DataKi:  1.33E+3nMAssay Description:Displacement of [3H]NMS from human muscarinic M3 receptor expressed in insect Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed