Compile Data Set for Download or QSAR
Report error Found 22 Enz. Inhib. hit(s) with all data for entry = 50037405
TargetKappa-type opioid receptor(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50169772((3S,4aR,6S,8R,8aR,10aR)-3-Furan-3-yl-6-methoxymeth...)
Affinity DataEC50:  0.600nMAssay Description:Activation of human k-opioid receptor as increased [35S]GTPcS binding More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2012
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50169775((3S,4aR,6S,8R,8aR,10aR)-3-Furan-3-yl-6-hydroxy-4a,...)
Affinity DataEC50:  193nMAssay Description:Activation of human k-opioid receptor as increased [35S]GTPcS binding More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2012
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50169777((3S,4aR,6S,8R,8aR,10aR)-6-Acetoxy-3-furan-3-yl-4a,...)
Affinity DataEC50:  4.5nMAssay Description:Activation of human k-opioid receptor as increased [35S]GTPcS binding More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2012
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50169775((3S,4aR,6S,8R,8aR,10aR)-3-Furan-3-yl-6-hydroxy-4a,...)
Affinity DataEC50:  193nMAssay Description:Activation of human k-opioid receptor as increased [35S]GTPcS binding More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2012
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50000296(CHEMBL441765 | CHEMBL482811 | U-50488H | US1149237...)
Affinity DataEC50:  4.5nMAssay Description:Activation of human k-opioid receptor as increased [35S]GTPcS binding More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2012
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50169775((3S,4aR,6S,8R,8aR,10aR)-3-Furan-3-yl-6-hydroxy-4a,...)
Affinity DataEC50:  193nMAssay Description:Activation of human k-opioid receptor as increased [35S]GTPcS binding More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2012
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50169777((3S,4aR,6S,8R,8aR,10aR)-6-Acetoxy-3-furan-3-yl-4a,...)
Affinity DataEC50:  4.5nMAssay Description:Activation of human k-opioid receptor as increased [35S]GTPcS binding More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2012
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50169772((3S,4aR,6S,8R,8aR,10aR)-3-Furan-3-yl-6-methoxymeth...)
Affinity DataEC50:  0.600nMAssay Description:Activation of human k-opioid receptor as increased [35S]GTPcS binding More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2012
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50169772((3S,4aR,6S,8R,8aR,10aR)-3-Furan-3-yl-6-methoxymeth...)
Affinity DataKi:  0.400nMAssay Description:Agonistic activity against human k-opioid receptor using [3H]diprenorphineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2012
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50169772((3S,4aR,6S,8R,8aR,10aR)-3-Furan-3-yl-6-methoxymeth...)
Affinity DataKi:  0.400nMAssay Description:Agonistic activity against human k-opioid receptor using [3H]diprenorphineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2012
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50169777((3S,4aR,6S,8R,8aR,10aR)-6-Acetoxy-3-furan-3-yl-4a,...)
Affinity DataKi:  1.30nMAssay Description:Agonistic activity against human k-opioid receptor using [3H]diprenorphineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2012
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50169777((3S,4aR,6S,8R,8aR,10aR)-6-Acetoxy-3-furan-3-yl-4a,...)
Affinity DataKi:  1.30nMAssay Description:Agonistic activity against human k-opioid receptor using [3H]diprenorphineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2012
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50000296(CHEMBL441765 | CHEMBL482811 | U-50488H | US1149237...)
Affinity DataKi:  1.40nMAssay Description:Agonistic activity against human k-opioid receptor using [3H]diprenorphineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2012
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50169775((3S,4aR,6S,8R,8aR,10aR)-3-Furan-3-yl-6-hydroxy-4a,...)
Affinity DataKi:  43nMAssay Description:Agonistic activity against human k-opioid receptor using [3H]diprenorphineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2012
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50169775((3S,4aR,6S,8R,8aR,10aR)-3-Furan-3-yl-6-hydroxy-4a,...)
Affinity DataKi:  43nMAssay Description:Agonistic activity against human k-opioid receptor using [3H]diprenorphineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2012
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50169775((3S,4aR,6S,8R,8aR,10aR)-3-Furan-3-yl-6-hydroxy-4a,...)
Affinity DataKi:  43nMAssay Description:Agonistic activity against human k-opioid receptor using [3H]diprenorphineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2012
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50169778((3S,4aR,6S,8R,8aR,10aR)-6-(3-Fluoro-benzoyloxy)-3-...)
Affinity DataKi: >1.00E+3nMAssay Description:Agonistic activity against human k-opioid receptor using [3H]diprenorphineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2012
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50169776((3S,4aS,8aR,10aR)-3-Furan-3-yl-4a,8a-dimethyl-1,6-...)
Affinity DataKi: >1.00E+3nMAssay Description:Agonistic activity against human k-opioid receptor using [3H]diprenorphineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2012
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50169779((3S,4aR,6S,8R,8aR,10aR)-3-Furan-3-yl-4a,8a-dimethy...)
Affinity DataKi: >1.00E+3nMAssay Description:Agonistic activity against human k-opioid receptor using [3H]diprenorphineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2012
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50169779((3S,4aR,6S,8R,8aR,10aR)-3-Furan-3-yl-4a,8a-dimethy...)
Affinity DataKi: >1.00E+3nMAssay Description:Agonistic activity against human k-opioid receptor using [3H]diprenorphineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2012
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50169780((3S,4aR,6S,8R,8aR,10aR)-6-Cyclopropanecarbonyloxy-...)
Affinity DataKi: >1.00E+3nMAssay Description:Agonistic activity against human k-opioid receptor using [3H]diprenorphineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2012
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50169773((3S,4aR,6S,8R,8aR,10aR)-3-Furan-3-yl-4a,8a-dimethy...)
Affinity DataKi: >1.00E+3nMAssay Description:Agonistic activity against human k-opioid receptor using [3H]diprenorphineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2012
Entry Details Article
PubMed