Compile Data Set for Download or QSAR
Report error Found 13 Enz. Inhib. hit(s) with all data for entry = 50016155
Target72 kDa type IV collagenase(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50161327({(S)-4-[(Biphenyl-4-sulfonyl)-isopropoxy-amino]-4-...)
Affinity DataIC50: 0.410nMAssay Description:Inhibition of Matrix metalloprotease-2 in MMPi assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMatrix metalloproteinase-14(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50161327({(S)-4-[(Biphenyl-4-sulfonyl)-isopropoxy-amino]-4-...)
Affinity DataIC50: 7.70nMAssay Description:Inhibition of Matrix metalloprotease-14 in MMPi assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMatrix metalloproteinase-9(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50165670(N-(3-{(R)-3-[(Biphenyl-4-sulfonyl)-isopropoxy-amin...)
Affinity DataIC50: 8.30nMAssay Description:Inhibition of Matrix metalloprotease-9 in MMPi assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50165670(N-(3-{(R)-3-[(Biphenyl-4-sulfonyl)-isopropoxy-amin...)
Affinity DataIC50: 9.80nMAssay Description:Inhibition of Matrix metalloprotease-2 in MMPi assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMatrix metalloproteinase-9(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50161327({(S)-4-[(Biphenyl-4-sulfonyl)-isopropoxy-amino]-4-...)
Affinity DataIC50: 16nMAssay Description:Inhibition of Matrix metalloprotease-9 in MMPi assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50165671(N-{(R)-3-[(Biphenyl-4-sulfonyl)-isopropoxy-amino]-...)
Affinity DataIC50: 197nMAssay Description:Inhibition of Matrix metalloprotease-2 in MMPi assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetInterstitial collagenase(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50165670(N-(3-{(R)-3-[(Biphenyl-4-sulfonyl)-isopropoxy-amin...)
Affinity DataIC50: 397nMAssay Description:Inhibition of Matrix metalloprotease-1 in MMPi assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMatrix metalloproteinase-9(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50165671(N-{(R)-3-[(Biphenyl-4-sulfonyl)-isopropoxy-amino]-...)
Affinity DataIC50: 983nMAssay Description:Inhibition of Matrix metalloprotease-9 in MMPi assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMatrix metalloproteinase-14(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50165671(N-{(R)-3-[(Biphenyl-4-sulfonyl)-isopropoxy-amino]-...)
Affinity DataIC50: 1.49E+3nMAssay Description:Inhibition of Matrix metalloprotease-14 in MMPi assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50165672((R)-2-[(Biphenyl-4-sulfonyl)-isopropoxy-amino]-4-(...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of Matrix metalloprotease-2 in MMPi assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetInterstitial collagenase(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50165671(N-{(R)-3-[(Biphenyl-4-sulfonyl)-isopropoxy-amino]-...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of Matrix metalloprotease-1 in MMPi assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMatrix metalloproteinase-9(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50165672((R)-2-[(Biphenyl-4-sulfonyl)-isopropoxy-amino]-4-(...)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of Matrix metalloprotease-9 in MMPi assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetInterstitial collagenase(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50161327({(S)-4-[(Biphenyl-4-sulfonyl)-isopropoxy-amino]-4-...)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of Matrix metalloprotease-1 in MMPi assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed