Compile Data Set for Download or QSAR
Report error Found 20 Enz. Inhib. hit(s) with all data for entry = 50015786
TargetHistamine H1 receptor(Guinea pig)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50160938(4-Chloro-2-{2-[4-(1-furan-3-ylmethyl-1H-indol-3-yl...)
Affinity DataIC50: 70nMAssay Description:Inhibitory concentration against histamine-H1 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50160937(2-(2-{4-[1-(2-Ethoxy-ethyl)-1H-indol-3-yl]-piperid...)
Affinity DataIC50: 86nMAssay Description:Inhibitory concentration against histamine-H1 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50160930(2-{2-[4-(1-Butyl-1H-indol-3-yl)-piperidin-1-yl]-et...)
Affinity DataIC50: 120nMAssay Description:Inhibitory concentration against histamine-H1 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50160942(4-Chloro-2-(2-{4-[1-(5-chloro-thiophen-2-ylmethyl)...)
Affinity DataIC50: 135nMAssay Description:Inhibitory concentration against histamine-H1 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50160939(2-{2-[4-(1-Furan-3-ylmethyl-1H-indol-3-yl)-piperid...)
Affinity DataIC50: 170nMAssay Description:Inhibitory concentration against histamine-H1 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50156893(2-(2-{4-[1-(2-ethoxyethyl)-1H-indol-3-yl]piperidin...)
Affinity DataIC50: 185nMAssay Description:Inhibitory concentration against histamine-H1 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50156867(2-(2-{4-[1-(2-ethoxyethyl)-1H-indol-3-yl]piperidin...)
Affinity DataIC50: 190nMAssay Description:Inhibitory concentration against histamine-H1 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50160935(5-[4-(1-Furan-3-ylmethyl-1H-indol-3-yl)-piperidin-...)
Affinity DataIC50: 205nMAssay Description:Inhibitory concentration against histamine-H1 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50160934(2-{2-[4-(1-Butyl-1H-indol-3-yl)-piperidin-1-yl]-et...)
Affinity DataIC50: 215nMAssay Description:Inhibitory concentration against histamine-H1 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50160941(2-{2-[4-(1-Furan-3-ylmethyl-1H-indol-3-yl)-piperid...)
Affinity DataIC50: 225nMAssay Description:Inhibitory concentration against histamine-H1 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50156873(2-{2-[4-(1-butyl-1H-indol-3-yl)piperidin-1-yl]etho...)
Affinity DataIC50: 235nMAssay Description:Inhibitory concentration against histamine-H1 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50160933(2-(2-{4-[1-(5-Chloro-thiophen-2-ylmethyl)-1H-indol...)
Affinity DataIC50: 240nMAssay Description:Inhibitory concentration against histamine-H1 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50160936(3-[4-(1-Butyl-1H-indol-3-yl)-piperidin-1-ylmethyl]...)
Affinity DataIC50: 275nMAssay Description:Inhibitory concentration against histamine-H1 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50156882(2-(2-(4-(1-((5-chlorothiophen-2-yl)methyl)-1H-indo...)
Affinity DataIC50: 295nMAssay Description:Inhibitory concentration against histamine-H1 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50156880(3-{4-[1-(5-chlorothiophen-2-ylmethyl)-1H-indol-3-y...)
Affinity DataIC50: 330nMAssay Description:Inhibitory concentration against histamine-H1 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50160932(5-{4-[1-(5-Chloro-thiophen-2-ylmethyl)-1H-indol-3-...)
Affinity DataIC50: 365nMAssay Description:Inhibitory concentration against histamine-H1 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50156871(4-{4-[1-(2-ethoxyethyl)-1H-indol-3-yl]piperidin-1-...)
Affinity DataIC50: 403nMAssay Description:Inhibitory concentration against histamine-H1 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50160940(5-[4-(1-Butyl-1H-indol-3-yl)-piperidin-1-ylmethyl]...)
Affinity DataIC50: 475nMAssay Description:Inhibitory concentration against histamine-H1 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50160931(3-[4-(1-Furan-3-ylmethyl-1H-indol-3-yl)-piperidin-...)
Affinity DataIC50: 560nMAssay Description:Inhibitory concentration against histamine-H1 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50156898(5-{4-[1-(2-Ethoxy-ethyl)-1H-indol-3-yl]-piperidin-...)
Affinity DataIC50: 690nMAssay Description:Inhibitory concentration against histamine-H1 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed