Compile Data Set for Download or QSAR
Report error Found 4 Enz. Inhib. hit(s) with all data for entry = 5741
TargetFarnesyl pyrophosphate synthase(Human)
Merck Research Laboratories

LigandPNGBDBM50059860(CHEMBL26180 | Hydroxy phosphonate, 1 | ((2E,6E)-1-...)
Affinity DataKi:  4.70nMAssay Description:Assay using farnesyl-ras-CVLS as the protein acceptor substrate.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetFarnesyl pyrophosphate synthase(Human)
Merck Research Laboratories

LigandPNGBDBM50059860(CHEMBL26180 | Hydroxy phosphonate, 1 | ((2E,6E)-1-...)
Affinity DataKi:  5.20nMAssay Description:FPTase activity was assayed in the biosynthetically forward direction at 30C.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetFarnesyl pyrophosphate synthase(Human)
Merck Research Laboratories

LigandPNGBDBM50059865([Hydroxy-(4,8,12-trimethyl-trideca-3,7,11-trienyl)...)
Affinity DataKi:  830nMAssay Description:FPTase activity was assayed in the biosynthetically forward direction at 30C.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetFarnesyl pyrophosphate synthase(Human)
Merck Research Laboratories

LigandPNGBDBM50059865([Hydroxy-(4,8,12-trimethyl-trideca-3,7,11-trienyl)...)
Affinity DataKi:  1.30E+3nMAssay Description:Assay using farnesyl-ras-CVLS as the protein acceptor substrate.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed