Compile Data Set for Download or QSAR
Report error Found 10 Enz. Inhib. hit(s) with all data for entry = 1250
TargetAcetylcholinesterase(Pacific electric ray)
Weizmann Institute of Science

LigandPNGBDBM10406((1S,12S,14R)-4-[8-(1,3-dioxo-2,3-dihydro-1H-isoind...)
Affinity DataIC50: 4nMpH: 8.0 T: 2°CAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. Enzyme activity was determined by measuring the absorbance at ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAcetylcholinesterase(Electric eel)
Weizmann Institute of Science

LigandPNGBDBM10406((1S,12S,14R)-4-[8-(1,3-dioxo-2,3-dihydro-1H-isoind...)
Affinity DataIC50: 11nMpH: 8.0 T: 2°CAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. Enzyme activity was determined by measuring the absorbance at ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAcetylcholinesterase(Pacific electric ray)
Weizmann Institute of Science

LigandPNGBDBM10405(galanthamine deriv. 3d | 2-{8-[(1S,12S,14R)-14-hyd...)
Affinity DataIC50: 38nMpH: 8.0 T: 2°CAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. Enzyme activity was determined by measuring the absorbance at ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAcetylcholinesterase(Electric eel)
Weizmann Institute of Science

LigandPNGBDBM10405(galanthamine deriv. 3d | 2-{8-[(1S,12S,14R)-14-hyd...)
Affinity DataIC50: 72nMpH: 8.0 T: 2°CAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. Enzyme activity was determined by measuring the absorbance at ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAcetylcholinesterase(Electric eel)
Weizmann Institute of Science

LigandPNGBDBM10407((1S,12S,14R)-9-{[8-(1,3-dioxo-2,3-dihydro-1H-isoin...)
Affinity DataIC50: 203nMpH: 8.0 T: 2°CAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. Enzyme activity was determined by measuring the absorbance at ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAcetylcholinesterase(Electric eel)
Weizmann Institute of Science

LigandPNGBDBM10408(galanthamine deriv. 14 | (1S,12S,14R)-14-hydroxy-9...)
Affinity DataIC50: 266nMpH: 8.0 T: 2°CAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. Enzyme activity was determined by measuring the absorbance at ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAcetylcholinesterase(Pacific electric ray)
Weizmann Institute of Science

LigandPNGBDBM10404(galantamine | (1S,12S,14R)-9-methoxy-4-methyl-11-o...)
Affinity DataIC50: 418nMpH: 8.0 T: 2°CAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. Enzyme activity was determined by measuring the absorbance at ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAcetylcholinesterase(Pacific electric ray)
Weizmann Institute of Science

LigandPNGBDBM10407((1S,12S,14R)-9-{[8-(1,3-dioxo-2,3-dihydro-1H-isoin...)
Affinity DataIC50: 499nMpH: 8.0 T: 2°CAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. Enzyme activity was determined by measuring the absorbance at ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAcetylcholinesterase(Electric eel)
Weizmann Institute of Science

LigandPNGBDBM10404(galantamine | (1S,12S,14R)-9-methoxy-4-methyl-11-o...)
Affinity DataIC50: 614nMpH: 8.0 T: 2°CAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. Enzyme activity was determined by measuring the absorbance at ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAcetylcholinesterase(Pacific electric ray)
Weizmann Institute of Science

LigandPNGBDBM10408(galanthamine deriv. 14 | (1S,12S,14R)-14-hydroxy-9...)
Affinity DataIC50: 702nMpH: 8.0 T: 2°CAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. Enzyme activity was determined by measuring the absorbance at ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed