Compile Data Set for Download or QSAR
Report error Found 15 Enz. Inhib. hit(s) with all data for entry = 5478
TargetKappa-type opioid receptor(Human)
Temple University

Curated by PDSP Ki Database
LigandPNGBDBM86549(CAS_213055 | NSC_213055 | TRK-820)
Affinity DataKi:  0.0250nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2012
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
Temple University

Curated by PDSP Ki Database
LigandPNGBDBM86549(CAS_213055 | NSC_213055 | TRK-820)
Affinity DataKi:  0.0750nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2012
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
Temple University

Curated by PDSP Ki Database
LigandPNGBDBM86547(NSC_135349 | CAS_135349 | U50,488H)
Affinity DataKi:  2.20nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Temple University

Curated by PDSP Ki Database
LigandPNGBDBM86549(CAS_213055 | NSC_213055 | TRK-820)
Affinity DataKi:  3.20nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
Temple University

Curated by PDSP Ki Database
LigandPNGBDBM86546(NSC_104787 | CAS_88373-73-3 | DPDPE)
Affinity DataKi:  3.40nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2012
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
Temple University

Curated by PDSP Ki Database
LigandPNGBDBM86548(NSC_128563 | CAS_83729-01-5 | Salvinorin A)
Affinity DataKi:  4.60nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Temple University

Curated by PDSP Ki Database
LigandPNGBDBM86549(CAS_213055 | NSC_213055 | TRK-820)
Affinity DataKi:  5.20nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2012
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
Temple University

Curated by PDSP Ki Database
LigandPNGBDBM86548(NSC_128563 | CAS_83729-01-5 | Salvinorin A)
Affinity DataKi:  7.90nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Temple University

Curated by PDSP Ki Database
LigandPNGBDBM86253(CAS_100929-53-1 | NSC_104742 | DAMGO | US10836728,...)
Affinity DataKi:  8.90nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2012
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
Temple University

Curated by PDSP Ki Database
LigandPNGBDBM86547(NSC_135349 | CAS_135349 | U50,488H)
Affinity DataKi:  11nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2012
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
Temple University

Curated by PDSP Ki Database
LigandPNGBDBM50092521(CHEMBL447234 | 3FLB | 3-((3-Fluoro-phenyl)-{[(3-fl...)
Affinity DataKi:  73.6nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2012
Entry Details Article
PubMed
TargetNociceptin receptor(Human)
Temple University

Curated by PDSP Ki Database
LigandPNGBDBM86549(CAS_213055 | NSC_213055 | TRK-820)
Affinity DataKi:  147nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
Temple University

Curated by PDSP Ki Database
LigandPNGBDBM86549(CAS_213055 | NSC_213055 | TRK-820)
Affinity DataKi:  161nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2012
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
Temple University

Curated by PDSP Ki Database
LigandPNGBDBM50092521(CHEMBL447234 | 3FLB | 3-((3-Fluoro-phenyl)-{[(3-fl...)
Affinity DataKi:  248nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
Temple University

Curated by PDSP Ki Database
LigandPNGBDBM86549(CAS_213055 | NSC_213055 | TRK-820)
Affinity DataKi:  289nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2012
Entry Details Article
PubMed