Compile Data Set for Download or QSAR
Report error Found 7 Enz. Inhib. hit(s) with all data for entry = 50015094
TargetRetinoic acid receptor RXR-alpha(Human)
Institute

Curated by ChEMBL
LigandPNGBDBM50151228(6-[Cyclopropylidene-(5,5,8,8-tetramethyl-3-propoxy...)
Affinity DataIC50: 6nMAssay Description:Inhibition of [3H]9-cis-retinoic acid binding to human retinoid X receptor alpha ligand-binding domain expressed in Escherichia coliMore data for this Ligand-Target Pair
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PubMed
TargetRetinoic acid receptor RXR-alpha(Human)
Institute

Curated by ChEMBL
LigandPNGBDBM50151230(6-[(3-Butoxy-5,5,8,8-tetramethyl-5,6,7,8-tetrahydr...)
Affinity DataIC50: 10nMAssay Description:Inhibition of [3H]9-cis-retinoic acid binding to human retinoid X receptor alpha ligand-binding domain expressed in Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRetinoic acid receptor RXR-alpha(Human)
Institute

Curated by ChEMBL
LigandPNGBDBM50151229(4-[Cyclopropylidene-(3,5,5,8,8-pentamethyl-5,6,7,8...)
Affinity DataIC50: 21nMAssay Description:Inhibition of [3H]9-cis-retinoic acid binding to human retinoid X receptor alpha ligand-binding domain expressed in Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRetinoic acid receptor RXR-alpha(Human)
Institute

Curated by ChEMBL
LigandPNGBDBM31892(CHEMBL705 | 9-cis retinoic acid | alitretinoin | P...)
Affinity DataIC50: 29nMAssay Description:Inhibition of [3H]9-cis-retinoic acid binding to human retinoid X receptor alpha ligand-binding domain expressed in Escherichia coliMore data for this Ligand-Target Pair
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PubMedPDB3D3D Structure (crystal)
TargetRetinoic acid receptor RXR-alpha(Human)
Institute

Curated by ChEMBL
LigandPNGBDBM50151231(4-[Cyclopropylidene-(5,5,8,8-tetramethyl-3-propoxy...)
Affinity DataIC50: 120nMAssay Description:Inhibition of [3H]9-cis-retinoic acid binding to human retinoid X receptor alpha ligand-binding domain expressed in Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRetinoic acid receptor RXR-alpha(Human)
Institute

Curated by ChEMBL
LigandPNGBDBM50151227(4-[(3-Butoxy-5,5,8,8-tetramethyl-5,6,7,8-tetrahydr...)
Affinity DataIC50: 270nMAssay Description:Inhibition of [3H]9-cis-retinoic acid binding to human retinoid X receptor alpha ligand-binding domain expressed in Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRetinoic acid receptor RXR-alpha(Human)
Institute

Curated by ChEMBL
LigandPNGBDBM50151226(4-[(3-Butyl-5,5,8,8-tetramethyl-5,6,7,8-tetrahydro...)
Affinity DataIC50: 500nMAssay Description:Inhibition of [3H]9-cis-retinoic acid binding to human retinoid X receptor alpha ligand-binding domain expressed in Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed