Compile Data Set for Download or QSAR
Report error Found 124 Enz. Inhib. hit(s) with all data for entry = 50014918
TargetAdenosine receptor A3(Human)
Otsuka Pharmaceutical Factory

Curated by ChEMBL
LigandPNGBDBM50117232(5-Butyl-8-phenyl-3H-[1,2,4]triazolo[5,1-i]purine |...)
Affinity DataIC50: 0.25nMAssay Description:Displacement of specific [125I]AB-MECA binding at human adenosine A3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A3(Human)
Otsuka Pharmaceutical Factory

Curated by ChEMBL
LigandPNGBDBM50117238(5-Butyl-8-(4-chloro-phenyl)-3H-[1,2,4]triazolo[5,1...)
Affinity DataIC50: 0.410nMAssay Description:Displacement of specific [125I]AB-MECA binding at human adenosine A3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A3(Human)
Otsuka Pharmaceutical Factory

Curated by ChEMBL
LigandPNGBDBM50117215(5-Butyl-8-(4-trifluoromethyl-phenyl)-3H-[1,2,4]tri...)
Affinity DataIC50: 0.610nMAssay Description:Displacement of specific [125I]AB-MECA binding at human adenosine A3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A3(Human)
Otsuka Pharmaceutical Factory

Curated by ChEMBL
LigandPNGBDBM50149106(8-Biphenyl-4-yl-5-(2-methoxy-ethyl)-3H-[1,2,4]tria...)
Affinity DataIC50: 0.900nMAssay Description:Displacement of specific [125I]AB-MECA binding at human adenosine A3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A3(Human)
Otsuka Pharmaceutical Factory

Curated by ChEMBL
LigandPNGBDBM50149112(5-Butyl-2-(4-fluoro-phenyl)-7H-pyrazolo[4,3-e][1,2...)
Affinity DataIC50: 1.90nMAssay Description:Displacement of specific [125I]AB-MECA binding at human adenosine A3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A3(Human)
Otsuka Pharmaceutical Factory

Curated by ChEMBL
LigandPNGBDBM50145230(5-Butyl-2-phenyl-7H-pyrazolo[4,3-e][1,2,4]triazolo...)
Affinity DataIC50: 2.10nMAssay Description:Displacement of specific [125I]AB-MECA binding at human adenosine A3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A3(Human)
Otsuka Pharmaceutical Factory

Curated by ChEMBL
LigandPNGBDBM50149110(5-Butyl-2-p-tolyl-7H-pyrazolo[4,3-e][1,2,4]triazol...)
Affinity DataIC50: 4nMAssay Description:Displacement of specific [125I]AB-MECA binding at human adenosine A3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A3(Human)
Otsuka Pharmaceutical Factory

Curated by ChEMBL
LigandPNGBDBM50149105(2-Phenyl-5-propyl-7H-pyrazolo[4,3-e][1,2,4]triazol...)
Affinity DataIC50: 4.10nMAssay Description:Displacement of specific [125I]AB-MECA binding at human adenosine A3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A3(Human)
Otsuka Pharmaceutical Factory

Curated by ChEMBL
LigandPNGBDBM50149126(5-Butyl-2-(4-chloro-phenyl)-7H-pyrazolo[4,3-e][1,2...)
Affinity DataIC50: 4.90nMAssay Description:Displacement of specific [125I]AB-MECA binding at human adenosine A3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A3(Human)
Otsuka Pharmaceutical Factory

Curated by ChEMBL
LigandPNGBDBM50117219(8-Biphenyl-4-yl-5-butyl-3H-[1,2,4]triazolo[5,1-i]p...)
Affinity DataIC50: 5nMAssay Description:Displacement of specific [125I]AB-MECA binding at human adenosine A3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A3(Human)
Otsuka Pharmaceutical Factory

Curated by ChEMBL
LigandPNGBDBM50149124(4-[8-(4-Chloro-phenyl)-3H-[1,2,4]triazolo[5,1-i]pu...)
Affinity DataIC50: 5.40nMAssay Description:Displacement of specific [125I]AB-MECA binding at human adenosine A3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A3(Human)
Otsuka Pharmaceutical Factory

Curated by ChEMBL
LigandPNGBDBM50149118(5-Ethyl-2-phenyl-7H-pyrazolo[4,3-e][1,2,4]triazolo...)
Affinity DataIC50: 6.20nMAssay Description:Displacement of specific [125I]AB-MECA binding at human adenosine A3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A3(Human)
Otsuka Pharmaceutical Factory

Curated by ChEMBL
LigandPNGBDBM50149122(2-(4-Bromo-phenyl)-5-butyl-[1,2,4]triazolo[1,5-c]q...)
Affinity DataIC50: 8.20nMAssay Description:Displacement of specific [125I]AB-MECA binding at human adenosine A3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A3(Human)
Otsuka Pharmaceutical Factory

Curated by ChEMBL
LigandPNGBDBM50149129(4-(8-Biphenyl-4-yl-3H-[1,2,4]triazolo[5,1-i]purin-...)
Affinity DataIC50: 8.70nMAssay Description:Displacement of specific [125I]AB-MECA binding at human adenosine A3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A3(Human)
Otsuka Pharmaceutical Factory

Curated by ChEMBL
LigandPNGBDBM50149132(5-(8-Biphenyl-4-yl-3H-[1,2,4]triazolo[5,1-i]purin-...)
Affinity DataIC50: 9.10nMAssay Description:Displacement of specific [125I]AB-MECA binding at human adenosine A3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A3(Human)
Otsuka Pharmaceutical Factory

Curated by ChEMBL
LigandPNGBDBM50149116(4-(5-Butyl-[1,2,4]triazolo[1,5-c]quinazolin-2-yl)-...)
Affinity DataIC50: 10nMAssay Description:Displacement of specific [125I]AB-MECA binding at human adenosine A3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A3(Human)
Otsuka Pharmaceutical Factory

Curated by ChEMBL
LigandPNGBDBM50145227(5-Butyl-2-(4-methoxy-phenyl)-7H-pyrazolo[4,3-e][1,...)
Affinity DataIC50: 10nMAssay Description:Displacement of specific [125I]AB-MECA binding at human adenosine A3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A3(Human)
Otsuka Pharmaceutical Factory

Curated by ChEMBL
LigandPNGBDBM50149117(5-Butyl-2-(3-chloro-phenyl)-7H-pyrazolo[4,3-e][1,2...)
Affinity DataIC50: 10nMAssay Description:Displacement of specific [125I]AB-MECA binding at human adenosine A3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A3(Human)
Otsuka Pharmaceutical Factory

Curated by ChEMBL
LigandPNGBDBM50149136(5-Butyl-2-(4-ethoxy-phenyl)-7H-pyrazolo[4,3-e][1,2...)
Affinity DataIC50: 10nMAssay Description:Displacement of specific [125I]AB-MECA binding at human adenosine A3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A3(Human)
Otsuka Pharmaceutical Factory

Curated by ChEMBL
LigandPNGBDBM50149120(5-Butyl-2-(2-chloro-phenyl)-7H-pyrazolo[4,3-e][1,2...)
Affinity DataIC50: 10nMAssay Description:Displacement of specific [125I]AB-MECA binding at human adenosine A3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A3(Human)
Otsuka Pharmaceutical Factory

Curated by ChEMBL
LigandPNGBDBM50149121(5-Butyl-2-(4-ethyl-phenyl)-7H-pyrazolo[4,3-e][1,2,...)
Affinity DataIC50: 12nMAssay Description:Displacement of specific [125I]AB-MECA binding at human adenosine A3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A3(Human)
Otsuka Pharmaceutical Factory

Curated by ChEMBL
LigandPNGBDBM50149127(3-(8-Biphenyl-4-yl-3H-[1,2,4]triazolo[5,1-i]purin-...)
Affinity DataIC50: 15nMAssay Description:Displacement of specific [125I]AB-MECA binding at human adenosine A3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A3(Human)
Otsuka Pharmaceutical Factory

Curated by ChEMBL
LigandPNGBDBM50149128(2-(4-Bromo-phenyl)-5-butyl-7H-pyrazolo[4,3-e][1,2,...)
Affinity DataIC50: 19nMAssay Description:Displacement of specific [125I]AB-MECA binding at human adenosine A3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A3(Human)
Otsuka Pharmaceutical Factory

Curated by ChEMBL
LigandPNGBDBM50149130(2-(4-Bromo-phenyl)-5-butyl-9-chloro-[1,2,4]triazol...)
Affinity DataIC50: 22nMAssay Description:Displacement of specific [125I]AB-MECA binding at human adenosine A3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A3(Human)
Otsuka Pharmaceutical Factory

Curated by ChEMBL
LigandPNGBDBM50149111(5-Butyl-2-(4-chloro-phenyl)-[1,2,4]triazolo[1,5-c]...)
Affinity DataIC50: 26nMAssay Description:Displacement of specific [125I]AB-MECA binding at human adenosine A3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Human)
Otsuka Pharmaceutical Factory

Curated by ChEMBL
LigandPNGBDBM50149118(5-Ethyl-2-phenyl-7H-pyrazolo[4,3-e][1,2,4]triazolo...)
Affinity DataIC50: 27nMAssay Description:Displacement of specific [3H]DPCPX binding at human adenosine A1 receptor expressed in CHO cells.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Human)
Otsuka Pharmaceutical Factory

Curated by ChEMBL
LigandPNGBDBM50145230(5-Butyl-2-phenyl-7H-pyrazolo[4,3-e][1,2,4]triazolo...)
Affinity DataIC50: 27nMAssay Description:Displacement of specific [3H]DPCPX binding at human adenosine A1 receptor expressed in CHO cells.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A3(Human)
Otsuka Pharmaceutical Factory

Curated by ChEMBL
LigandPNGBDBM50149108(5-Butyl-2-(4-fluoro-phenyl)-[1,2,4]triazolo[1,5-c]...)
Affinity DataIC50: 28nMAssay Description:Displacement of specific [125I]AB-MECA binding at human adenosine A3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A3(Human)
Otsuka Pharmaceutical Factory

Curated by ChEMBL
LigandPNGBDBM50149104(5-Butyl-9-chloro-2-(4-chloro-phenyl)-[1,2,4]triazo...)
Affinity DataIC50: 28nMAssay Description:Displacement of specific [125I]AB-MECA binding at human adenosine A3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A3(Human)
Otsuka Pharmaceutical Factory

Curated by ChEMBL
LigandPNGBDBM50149103(5-Butyl-9-chloro-2-(4-methoxy-phenyl)-[1,2,4]triaz...)
Affinity DataIC50: 33nMAssay Description:Displacement of specific [125I]AB-MECA binding at human adenosine A3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A3(Human)
Otsuka Pharmaceutical Factory

Curated by ChEMBL
LigandPNGBDBM50149107(5-Butyl-2-p-tolyl-[1,2,4]triazolo[1,5-c]quinazolin...)
Affinity DataIC50: 34nMAssay Description:Displacement of specific [125I]AB-MECA binding at human adenosine A3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A3(Human)
Otsuka Pharmaceutical Factory

Curated by ChEMBL
LigandPNGBDBM50149133(5-Butyl-8-chloro-2-(4-methoxy-phenyl)-[1,2,4]triaz...)
Affinity DataIC50: 34nMAssay Description:Displacement of specific [125I]AB-MECA binding at human adenosine A3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A3(Human)
Otsuka Pharmaceutical Factory

Curated by ChEMBL
LigandPNGBDBM50149113(5-Butyl-2-(4-ethoxy-phenyl)-[1,2,4]triazolo[1,5-c]...)
Affinity DataIC50: 35nMAssay Description:Displacement of specific [125I]AB-MECA binding at human adenosine A3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Human)
Otsuka Pharmaceutical Factory

Curated by ChEMBL
LigandPNGBDBM50149105(2-Phenyl-5-propyl-7H-pyrazolo[4,3-e][1,2,4]triazol...)
Affinity DataIC50: 38nMAssay Description:Displacement of specific [3H]DPCPX binding at human adenosine A1 receptor expressed in CHO cells.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A3(Human)
Otsuka Pharmaceutical Factory

Curated by ChEMBL
LigandPNGBDBM50149134(5-Butyl-2-(4-propyl-phenyl)-7H-pyrazolo[4,3-e][1,2...)
Affinity DataIC50: 42nMAssay Description:Displacement of specific [125I]AB-MECA binding at human adenosine A3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A3(Human)
Otsuka Pharmaceutical Factory

Curated by ChEMBL
LigandPNGBDBM50149123(5-Butyl-9-chloro-2-phenyl-[1,2,4]triazolo[1,5-c]qu...)
Affinity DataIC50: 45nMAssay Description:Displacement of specific [125I]AB-MECA binding at human adenosine A3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A3(Human)
Otsuka Pharmaceutical Factory

Curated by ChEMBL
LigandPNGBDBM50149115(5-Butyl-8-chloro-2-phenyl-[1,2,4]triazolo[1,5-c]qu...)
Affinity DataIC50: 48nMAssay Description:Displacement of specific [125I]AB-MECA binding at human adenosine A3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A2a(Human)
Otsuka Pharmaceutical Factory

Curated by ChEMBL
LigandPNGBDBM50117232(5-Butyl-8-phenyl-3H-[1,2,4]triazolo[5,1-i]purine |...)
Affinity DataIC50: 71nMAssay Description:Displacement of specific [3H]-CGS- 21680 binding at human adenosine A2A receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A2b(Human)
Otsuka Pharmaceutical Factory

Curated by ChEMBL
LigandPNGBDBM50149118(5-Ethyl-2-phenyl-7H-pyrazolo[4,3-e][1,2,4]triazolo...)
Affinity DataIC50: 100nMAssay Description:Displacement of specific [3H]DPCPX binding at human adenosine A2B receptor expressed in HEK293 cells.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A3(Human)
Otsuka Pharmaceutical Factory

Curated by ChEMBL
LigandPNGBDBM50149119(5-Butyl-8-methyl-2-phenyl-[1,2,4]triazolo[1,5-c]qu...)
Affinity DataIC50: 110nMAssay Description:Displacement of specific [125I]AB-MECA binding at human adenosine A3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A2a(Human)
Otsuka Pharmaceutical Factory

Curated by ChEMBL
LigandPNGBDBM50149105(2-Phenyl-5-propyl-7H-pyrazolo[4,3-e][1,2,4]triazol...)
Affinity DataIC50: 120nMAssay Description:Displacement of specific [3H]-CGS- 21680 binding at human adenosine A2A receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A3(Human)
Otsuka Pharmaceutical Factory

Curated by ChEMBL
LigandPNGBDBM50149135(5-Butyl-2-furan-2-yl-[1,2,4]triazolo[1,5-c]quinazo...)
Affinity DataIC50: 120nMAssay Description:Displacement of specific [125I]AB-MECA binding at human adenosine A3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A3(Human)
Otsuka Pharmaceutical Factory

Curated by ChEMBL
LigandPNGBDBM50145228(5-Butyl-2-(4-trifluoromethyl-phenyl)-7H-pyrazolo[4...)
Affinity DataIC50: 130nMAssay Description:Displacement of specific [125I]AB-MECA binding at human adenosine A3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A2a(Human)
Otsuka Pharmaceutical Factory

Curated by ChEMBL
LigandPNGBDBM50149120(5-Butyl-2-(2-chloro-phenyl)-7H-pyrazolo[4,3-e][1,2...)
Affinity DataIC50: 130nMAssay Description:Displacement of specific [3H]-CGS- 21680 binding at human adenosine A2A receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A3(Human)
Otsuka Pharmaceutical Factory

Curated by ChEMBL
LigandPNGBDBM50149137(2-Biphenyl-4-yl-5-butyl-[1,2,4]triazolo[1,5-c]quin...)
Affinity DataIC50: 140nMAssay Description:Displacement of specific [125I]AB-MECA binding at human adenosine A3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A3(Human)
Otsuka Pharmaceutical Factory

Curated by ChEMBL
LigandPNGBDBM50149131(5-Butyl-2-(4-tert-butyl-phenyl)-7H-pyrazolo[4,3-e]...)
Affinity DataIC50: 150nMAssay Description:Displacement of specific [125I]AB-MECA binding at human adenosine A3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A3(Human)
Otsuka Pharmaceutical Factory

Curated by ChEMBL
LigandPNGBDBM50145231(5-Butyl-2-(4-methoxy-phenyl)-[1,2,4]triazolo[1,5-c...)
Affinity DataIC50: 160nMAssay Description:Displacement of specific [125I]AB-MECA binding at human adenosine A3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A2a(Human)
Otsuka Pharmaceutical Factory

Curated by ChEMBL
LigandPNGBDBM50145230(5-Butyl-2-phenyl-7H-pyrazolo[4,3-e][1,2,4]triazolo...)
Affinity DataIC50: 190nMAssay Description:Displacement of specific [3H]-CGS- 21680 binding at human adenosine A2A receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A3(Human)
Otsuka Pharmaceutical Factory

Curated by ChEMBL
LigandPNGBDBM50145226(5-Butyl-2-phenyl-[1,2,4]triazolo[1,5-c]quinazoline...)
Affinity DataIC50: 260nMAssay Description:Displacement of specific [125I]AB-MECA binding at human adenosine A3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A2a(Human)
Otsuka Pharmaceutical Factory

Curated by ChEMBL
LigandPNGBDBM50149118(5-Ethyl-2-phenyl-7H-pyrazolo[4,3-e][1,2,4]triazolo...)
Affinity DataIC50: 310nMAssay Description:Displacement of specific [3H]-CGS- 21680 binding at human adenosine A2A receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
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