Compile Data Set for Download or QSAR
Report error Found 40 Enz. Inhib. hit(s) with all data for entry = 50036032
TargetPlatelet-activating factor receptor(Guinea pig)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50004622(CHEMBL106908 | 4-(2-Chloro-phenyl)-2-methyl-6-[4-(...)
Affinity DataIC50: 0.5nMAssay Description:In vitro inhibition of PAF-induced aggregation of rabbit washed platelets.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Guinea pig)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50004615(CHEMBL318172 | 4-(2-Chloro-phenyl)-2-methyl-6-[4-(...)
Affinity DataIC50: 1.30nMAssay Description:In vitro inhibition of PAF-induced aggregation of rabbit washed platelets.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Guinea pig)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50004630(CHEMBL106350 | 4-(2-Chloro-phenyl)-2-methyl-6-[4-(...)
Affinity DataIC50: 1.60nMAssay Description:In vitro inhibition of PAF-induced aggregation of rabbit washed platelets.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Guinea pig)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50004617(CHEMBL106475 | 4-(2-Chloro-phenyl)-6-methyl-2-[4-(...)
Affinity DataIC50: 1.80nMAssay Description:In vitro inhibition of PAF-induced aggregation of rabbit washed platelets.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Guinea pig)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50004637(CHEMBL263022 | 4-(2-Chloro-phenyl)-6-methyl-2-[4-(...)
Affinity DataIC50: 2.10nMAssay Description:In vitro inhibition of PAF-induced aggregation of rabbit washed platelets.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Guinea pig)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50004650(CHEMBL323382 | 6-Methyl-2-[4-(2-methyl-imidazo[4,5...)
Affinity DataIC50: 2.30nMAssay Description:In vitro inhibition of PAF-induced aggregation of rabbit washed platelets.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Guinea pig)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50004616(CHEMBL106819 | 4-(2-Chloro-phenyl)-2-methyl-6-[4-(...)
Affinity DataIC50: 2.5nMAssay Description:In vitro inhibition of PAF-induced aggregation of rabbit washed platelets.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Guinea pig)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50004645(CHEMBL326039 | 4-Benzo[b]thiophen-3-yl-6-methyl-2-...)
Affinity DataIC50: 3.10nMAssay Description:In vitro inhibition of PAF-induced aggregation of rabbit washed platelets.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Guinea pig)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50004646(CHEMBL318348 | 4-Benzo[1,3]dioxol-4-yl-6-methyl-2-...)
Affinity DataIC50: 3.20nMAssay Description:In vitro inhibition of PAF-induced aggregation of rabbit washed platelets.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Guinea pig)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50004631(CHEMBL106526 | 5-tert-Butylcarbamoyl-4-(2-chloro-p...)
Affinity DataIC50: 3.20nMAssay Description:In vitro inhibition of PAF-induced aggregation of rabbit washed platelets.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Guinea pig)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50004632(CHEMBL323067 | 4-(2-Chloro-phenyl)-2-[4-(2-ethyl-i...)
Affinity DataIC50: 3.40nMAssay Description:In vitro inhibition of PAF-induced aggregation of rabbit washed platelets.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Guinea pig)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50004633(4-(2-Chloro-phenyl)-6-methyl-2-[4-(2-methyl-imidaz...)
Affinity DataIC50: 4.30nMAssay Description:In vitro inhibition of PAF-induced aggregation of rabbit washed platelets.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Guinea pig)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50004641(CHEMBL320900 | 4-(2-Chloro-phenyl)-6-methyl-2-[4-(...)
Affinity DataIC50: 5nMAssay Description:In vitro inhibition of PAF-induced aggregation of rabbit washed platelets.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Guinea pig)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50004625(CHEMBL323407 | 5-Carbamoyl-4-(2-chloro-phenyl)-6-m...)
Affinity DataIC50: 5.60nMAssay Description:In vitro inhibition of PAF-induced aggregation of rabbit washed platelets.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Guinea pig)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50004648(CHEMBL322772 | 4-(2-Chloro-phenyl)-6-methyl-5-(pyr...)
Affinity DataIC50: 5.90nMAssay Description:In vitro inhibition of PAF-induced aggregation of rabbit washed platelets.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Guinea pig)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50004642(CHEMBL323429 | 4-(2-Chloro-phenyl)-2-[4-(2,4-dimet...)
Affinity DataIC50: 10nMAssay Description:In vitro inhibition of PAF-induced aggregation of rabbit washed platelets.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Guinea pig)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50004636(CHEMBL107113 | 4-(2-Chloro-phenyl)-2-[4-(3,5-dimet...)
Affinity DataIC50: 12nMAssay Description:In vitro inhibition of PAF-induced aggregation of rabbit washed platelets.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Guinea pig)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50004643(CHEMBL106800 | 2-Chloro-6'-methyl-2'-[4-(2-methyl-...)
Affinity DataIC50: 13nMAssay Description:In vitro inhibition of PAF-induced aggregation of rabbit washed platelets.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Guinea pig)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50004644(CHEMBL107951 | 4-(2-Chloro-phenyl)-2-[4-(2,4-dimet...)
Affinity DataIC50: 13nMAssay Description:In vitro inhibition of PAF-induced aggregation of rabbit washed platelets.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Guinea pig)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50004628(CHEMBL108260 | 4-(2-Chloro-phenyl)-2-methyl-6-[4-(...)
Affinity DataIC50: 14nMAssay Description:In vitro inhibition of PAF-induced aggregation of rabbit washed platelets.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Guinea pig)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50004639(CHEMBL326201 | 6'-Methyl-2'-[4-(2-methyl-imidazo[4...)
Affinity DataIC50: 14nMAssay Description:In vitro inhibition of PAF-induced aggregation of rabbit washed platelets.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Guinea pig)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50004626(CHEMBL323290 | 4-(2-Chloro-phenyl)-6-methyl-5-(pyr...)
Affinity DataIC50: 15nMAssay Description:In vitro inhibition of PAF-induced aggregation of rabbit washed platelets.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Guinea pig)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50004618(CHEMBL107321 | 4-(2-Chloro-phenyl)-6-methyl-2-[4-(...)
Affinity DataIC50: 22nMAssay Description:In vitro inhibition of PAF-induced aggregation of rabbit washed platelets.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Guinea pig)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50004627(CHEMBL107159 | 4-(2-Chloro-phenyl)-6-methyl-2-[4-(...)
Affinity DataIC50: 23nMAssay Description:In vitro inhibition of PAF-induced aggregation of rabbit washed platelets.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Guinea pig)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50004634(CHEMBL321722 | 4-(4-Cyano-phenyl)-6-methyl-2-[4-(2...)
Affinity DataIC50: 25nMAssay Description:In vitro inhibition of PAF-induced aggregation of rabbit washed platelets.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Guinea pig)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50004651(CHEMBL326012 | 4-(2-Chloro-phenyl)-6-methyl-2-[4-(...)
Affinity DataIC50: 28nMAssay Description:In vitro inhibition of PAF-induced aggregation of rabbit washed platelets.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Guinea pig)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50004623(CHEMBL323023 | 4-(2-Chloro-phenyl)-6-methyl-5-(pyr...)
Affinity DataIC50: 30nMAssay Description:In vitro inhibition of PAF-induced aggregation of rabbit washed platelets.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Guinea pig)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50004638(CHEMBL107241 | 6'-Methyl-2'-[4-(2-methyl-imidazo[4...)
Affinity DataIC50: 33nMAssay Description:In vitro inhibition of PAF-induced aggregation of rabbit washed platelets.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Guinea pig)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50000714(3-[4-(2-Chloro-phenyl)-9-methyl-6H-1-thia-5,7,8,9a...)
Affinity DataIC50: 146nMAssay Description:In vitro inhibition of PAF-induced aggregation of rabbit washed platelets.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Guinea pig)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50004649(CHEMBL320226 | 2-[4-(2-Butyl-imidazo[4,5-c]pyridin...)
Affinity DataIC50: 190nMAssay Description:In vitro inhibition of PAF-induced aggregation of rabbit washed platelets.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Guinea pig)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50004624(CHEMBL105500 | 4-(2-Chloro-phenyl)-6-methyl-2-[4-(...)
Affinity DataIC50: 200nMAssay Description:In vitro inhibition of PAF-induced aggregation of rabbit washed platelets.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Guinea pig)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50004629(CHEMBL326474 | 4-(2-Chloro-phenyl)-2-[4-(6-methoxy...)
Affinity DataIC50: 270nMAssay Description:In vitro inhibition of PAF-induced aggregation of rabbit washed platelets.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Guinea pig)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50004640(CHEMBL106564 | 4-(2-Chloro-phenyl)-6-methyl-2-[4-(...)
Affinity DataIC50: 580nMAssay Description:In vitro inhibition of PAF-induced aggregation of rabbit washed platelets.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Guinea pig)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50004621(CHEMBL107198 | 4-(2-Chloro-phenyl)-6-methyl-2-[4-(...)
Affinity DataIC50: 1.40E+3nMAssay Description:In vitro inhibition of PAF-induced aggregation of rabbit washed platelets.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Guinea pig)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50004619(CHEMBL323151 | 4-(2-Chloro-phenyl)-2-[4-(3,5-dimet...)
Affinity DataIC50: 3.00E+3nMAssay Description:In vitro inhibition of PAF-induced aggregation of rabbit washed platelets.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
LigandPNGBDBM50004633(4-(2-Chloro-phenyl)-6-methyl-2-[4-(2-methyl-imidaz...)
Affinity DataIC50: 6.60E+3nMAssay Description:Displacement of [3H]nitrendipine from L-type calcium channel of bovine frontal cortex membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
LigandPNGBDBM50004633(4-(2-Chloro-phenyl)-6-methyl-2-[4-(2-methyl-imidaz...)
Affinity DataIC50: 6.80E+3nMAssay Description:Displacement of [3H]desmethoxy-verapamil from L-type calcium channel of bovine frontal cortex membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
LigandPNGBDBM50004633(4-(2-Chloro-phenyl)-6-methyl-2-[4-(2-methyl-imidaz...)
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of [3H]-diltiazem from L-type calcium channel of bovine frontal cortex membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Guinea pig)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50004620(CHEMBL431069 | 4-(2-Chloro-phenyl)-6-methyl-2-[4-(...)
Affinity DataIC50: 1.00E+4nMAssay Description:In vitro inhibition of PAF-induced aggregation of rabbit washed platelets.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Guinea pig)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50004635(CHEMBL320855 | 4-(2-Chloro-phenyl)-2-[4-(3,5-dimet...)
Affinity DataIC50: 1.00E+4nMAssay Description:In vitro inhibition of PAF-induced aggregation of rabbit washed platelets.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed