Compile Data Set for Download or QSAR
Report error Found 82 Enz. Inhib. hit(s) with all data for entry = 50014517
TargetRetinoic acid receptor alpha(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50143835((E)-3-[4-(5,5,8,8-Tetramethyl-5,6,7,8-tetrahydro-n...)
Affinity DataEC50:  57nMAssay Description:Effective concentration for retinoic acid receptor alpha induced lipogenesis in C3H10T1/2 clone 8 fibroblast cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRetinoic acid receptor RXR-alpha(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50143826((E)-3-[4-(5,5,8,8-Tetramethyl-5,6,7,8-tetrahydro-n...)
Affinity DataEC50:  4nMAssay Description:Effective concentration for lipogenesis induced by retinoid X receptor alpha in C3H10T1/2 clone 8 fibroblast cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRetinoic acid receptor alpha(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50143833((E)-3-[4-(5,5,8,8-Tetramethyl-5,6,7,8-tetrahydro-n...)
Affinity DataEC50: >1.00E+4nMAssay Description:Effective concentration for Retinoic acid receptor alpha activity in CV-1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRetinoic acid receptor alpha(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50143827((E)-3-[4-(3-Methoxy-5,5,8,8-tetramethyl-5,6,7,8-te...)
Affinity DataEC50: >1.00E+4nMAssay Description:Effective concentration for retinoic acid receptor alpha induced lipogenesis in C3H10T1/2 clone 8 fibroblast cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRetinoic acid receptor RXR-alpha(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50143826((E)-3-[4-(5,5,8,8-Tetramethyl-5,6,7,8-tetrahydro-n...)
Affinity DataEC50:  660nMAssay Description:Effective concentration for lipogenesis induced by retinoid X receptor alpha in C3H10T1/2 clone 8 fibroblast cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRetinoic acid receptor RXR-alpha(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50143833((E)-3-[4-(5,5,8,8-Tetramethyl-5,6,7,8-tetrahydro-n...)
Affinity DataEC50:  20nMAssay Description:Effective concentration for Retinoid X receptor alpha activity in CV-1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRetinoic acid receptor alpha(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50143826((E)-3-[4-(5,5,8,8-Tetramethyl-5,6,7,8-tetrahydro-n...)
Affinity DataEC50: >1.00E+4nMAssay Description:Effective concentration for Retinoic acid receptor alpha activity in CV-1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRetinoic acid receptor RXR-alpha(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50143821((E)-3-[4-(5,5,8,8-Tetramethyl-3-propoxy-5,6,7,8-te...)
Affinity DataEC50:  40nMAssay Description:Effective concentration for lipogenesis induced by retinoid X receptor alpha in C3H10T1/2 clone 8 fibroblast cells; Partial agonistMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRetinoic acid receptor RXR-alpha(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50143825(5-[1-[4-(5,5,8,8-Tetramethyl-5,6,7,8-tetrahydro-na...)
Affinity DataEC50:  5nMAssay Description:Effective concentration for lipogenesis induced by retinoid X receptor alpha in C3H10T1/2 clone 8 fibroblast cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRetinoic acid receptor RXR-alpha(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50143827((E)-3-[4-(3-Methoxy-5,5,8,8-tetramethyl-5,6,7,8-te...)
Affinity DataEC50:  48nMAssay Description:Effective concentration for Retinoid X receptor alpha activity in CV-1 cells; Partial agonistMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRetinoic acid receptor RXR-alpha(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50143826((E)-3-[4-(5,5,8,8-Tetramethyl-5,6,7,8-tetrahydro-n...)
Affinity DataEC50:  3nMAssay Description:Effective concentration for Retinoid X receptor alpha activity in CV-1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRetinoic acid receptor RXR-alpha(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50143826((E)-3-[4-(5,5,8,8-Tetramethyl-5,6,7,8-tetrahydro-n...)
Affinity DataEC50:  5nMAssay Description:Effective concentration for Retinoid X receptor alpha activity in CV-1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRetinoic acid receptor RXR-alpha(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50143832((E)-3-[4-(3,5,5,8,8-Pentamethyl-5,6,7,8-tetrahydro...)
Affinity DataEC50:  29nMAssay Description:Effective concentration for Retinoid X receptor alpha activity in CV-1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRetinoic acid receptor alpha(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50143833((E)-3-[4-(5,5,8,8-Tetramethyl-5,6,7,8-tetrahydro-n...)
Affinity DataEC50: >1.00E+4nMAssay Description:Effective concentration for retinoic acid receptor alpha induced lipogenesis in C3H10T1/2 clone 8 fibroblast cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRetinoic acid receptor RXR-alpha(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50143823((E)-3-[5-Methyl-4-(5,5,8,8-tetramethyl-5,6,7,8-tet...)
Affinity DataEC50:  106nMAssay Description:Effective concentration for Retinoid X receptor alpha activity in CV-1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRetinoic acid receptor alpha(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50143826((E)-3-[4-(5,5,8,8-Tetramethyl-5,6,7,8-tetrahydro-n...)
Affinity DataEC50: >1.00E+4nMAssay Description:Effective concentration for retinoic acid receptor alpha induced lipogenesis in C3H10T1/2 clone 8 fibroblast cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRetinoic acid receptor RXR-alpha(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50143828(3-[4-(5,5,8,8-Tetramethyl-5,6,7,8-tetrahydro-napht...)
Affinity DataEC50:  97nMAssay Description:Effective concentration for Retinoid X receptor alpha activity in CV-1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRetinoic acid receptor RXR-alpha(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50143831((E)-3-[4-(5,5,8,8-Tetramethyl-5,6,7,8-tetrahydro-n...)
Affinity DataEC50:  42nMAssay Description:Effective concentration for Retinoid X receptor alpha activity in CV-1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRetinoic acid receptor RXR-alpha(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50143833((E)-3-[4-(5,5,8,8-Tetramethyl-5,6,7,8-tetrahydro-n...)
Affinity DataEC50:  72nMAssay Description:Effective concentration for lipogenesis induced by retinoid X receptor alpha in C3H10T1/2 clone 8 fibroblast cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRetinoic acid receptor RXR-alpha(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50143826((E)-3-[4-(5,5,8,8-Tetramethyl-5,6,7,8-tetrahydro-n...)
Affinity DataEC50:  97nMAssay Description:Effective concentration for Retinoid X receptor alpha activity in CV-1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRetinoic acid receptor alpha(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50143826((E)-3-[4-(5,5,8,8-Tetramethyl-5,6,7,8-tetrahydro-n...)
Affinity DataEC50: >1.00E+4nMAssay Description:Effective concentration for Retinoic acid receptor alpha activity in CV-1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRetinoic acid receptor alpha(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50409929(CHEMBL2113736)
Affinity DataEC50: >1.00E+4nMAssay Description:Effective concentration for retinoic acid receptor alpha induced lipogenesis in C3H10T1/2 clone 8 fibroblast cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRetinoic acid receptor alpha(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50409928(CHEMBL2113737)
Affinity DataEC50: >1.00E+4nMAssay Description:Effective concentration for retinoic acid receptor alpha induced lipogenesis in C3H10T1/2 clone 8 fibroblast cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRetinoic acid receptor RXR-alpha(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50409928(CHEMBL2113737)
Affinity DataEC50:  10nMAssay Description:Effective concentration for lipogenesis induced by retinoid X receptor alpha in C3H10T1/2 clone 8 fibroblast cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRetinoic acid receptor RXR-alpha(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50409928(CHEMBL2113737)
Affinity DataEC50:  60nMAssay Description:Effective concentration for Retinoid X receptor alpha activity in CV-1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRetinoic acid receptor alpha(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50409928(CHEMBL2113737)
Affinity DataEC50: >1.00E+4nMAssay Description:Effective concentration for Retinoic acid receptor alpha activity in CV-1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRetinoic acid receptor RXR-alpha(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50409929(CHEMBL2113736)
Affinity DataEC50:  22nMAssay Description:Effective concentration for lipogenesis induced by retinoid X receptor alpha in C3H10T1/2 clone 8 fibroblast cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRetinoic acid receptor RXR-alpha(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50409929(CHEMBL2113736)
Affinity DataEC50:  70nMAssay Description:Effective concentration for Retinoid X receptor alpha activity in CV-1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRetinoic acid receptor RXR-alpha(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50143823((E)-3-[5-Methyl-4-(5,5,8,8-tetramethyl-5,6,7,8-tet...)
Affinity DataEC50:  1.00E+3nMAssay Description:Effective concentration for lipogenesis induced by retinoid X receptor alpha in C3H10T1/2 clone 8 fibroblast cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRetinoic acid receptor alpha(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50143832((E)-3-[4-(3,5,5,8,8-Pentamethyl-5,6,7,8-tetrahydro...)
Affinity DataEC50: >1.00E+4nMAssay Description:Effective concentration for retinoic acid receptor alpha induced lipogenesis in C3H10T1/2 clone 8 fibroblast cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRetinoic acid receptor RXR-alpha(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50143826((E)-3-[4-(5,5,8,8-Tetramethyl-5,6,7,8-tetrahydro-n...)
Affinity DataEC50:  3nMAssay Description:Effective concentration for Retinoid X receptor alpha activity in CV-1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRetinoic acid receptor alpha(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50143832((E)-3-[4-(3,5,5,8,8-Pentamethyl-5,6,7,8-tetrahydro...)
Affinity DataEC50: >1.00E+4nMAssay Description:Effective concentration for Retinoic acid receptor alpha activity in CV-1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRetinoic acid receptor alpha(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50143831((E)-3-[4-(5,5,8,8-Tetramethyl-5,6,7,8-tetrahydro-n...)
Affinity DataEC50: >1.00E+4nMAssay Description:Effective concentration for retinoic acid receptor alpha induced lipogenesis in C3H10T1/2 clone 8 fibroblast cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRetinoic acid receptor alpha(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50143821((E)-3-[4-(5,5,8,8-Tetramethyl-3-propoxy-5,6,7,8-te...)
Affinity DataEC50: >1.00E+4nMAssay Description:Effective concentration for Retinoic acid receptor alpha activity in CV-1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRetinoic acid receptor alpha(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50143823((E)-3-[5-Methyl-4-(5,5,8,8-tetramethyl-5,6,7,8-tet...)
Affinity DataEC50: >1.00E+4nMAssay Description:Effective concentration for Retinoic acid receptor alpha activity in CV-1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRetinoic acid receptor alpha(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50143823((E)-3-[5-Methyl-4-(5,5,8,8-tetramethyl-5,6,7,8-tet...)
Affinity DataEC50: >1.00E+3nMAssay Description:Effective concentration for retinoic acid receptor alpha induced lipogenesis in C3H10T1/2 clone 8 fibroblast cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRetinoic acid receptor alpha(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50143827((E)-3-[4-(3-Methoxy-5,5,8,8-tetramethyl-5,6,7,8-te...)
Affinity DataEC50: >1.00E+4nMAssay Description:Effective concentration for Retinoic acid receptor alpha activity in CV-1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRetinoic acid receptor RXR-alpha(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50143832((E)-3-[4-(3,5,5,8,8-Pentamethyl-5,6,7,8-tetrahydro...)
Affinity DataEC50:  3.00E+3nMAssay Description:Effective concentration for lipogenesis induced by retinoid X receptor alpha in C3H10T1/2 clone 8 fibroblast cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRetinoic acid receptor RXR-alpha(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50143831((E)-3-[4-(5,5,8,8-Tetramethyl-5,6,7,8-tetrahydro-n...)
Affinity DataEC50:  749nMAssay Description:Effective concentration for lipogenesis induced by retinoid X receptor alpha in C3H10T1/2 clone 8 fibroblast cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRetinoic acid receptor RXR-alpha(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50143825(5-[1-[4-(5,5,8,8-Tetramethyl-5,6,7,8-tetrahydro-na...)
Affinity DataEC50:  4nMAssay Description:Effective concentration for Retinoid X receptor alpha activity in CV-1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRetinoic acid receptor alpha(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50143825(5-[1-[4-(5,5,8,8-Tetramethyl-5,6,7,8-tetrahydro-na...)
Affinity DataEC50: >1.00E+4nMAssay Description:Effective concentration for Retinoic acid receptor alpha activity in CV-1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRetinoic acid receptor alpha(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50143826((E)-3-[4-(5,5,8,8-Tetramethyl-5,6,7,8-tetrahydro-n...)
Affinity DataEC50: >1.00E+4nMAssay Description:Effective concentration for retinoic acid receptor alpha induced lipogenesis in C3H10T1/2 clone 8 fibroblast cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRetinoic acid receptor RXR-alpha(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50143830(4-(5,5,8,8-Tetramethyl-5,6,7,8-tetrahydro-naphthal...)
Affinity DataEC50: >1.00E+4nMAssay Description:Effective concentration for Retinoid X receptor alpha activity in CV-1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRetinoic acid receptor alpha(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50143825(5-[1-[4-(5,5,8,8-Tetramethyl-5,6,7,8-tetrahydro-na...)
Affinity DataEC50: >1.00E+4nMAssay Description:Effective concentration for retinoic acid receptor alpha induced lipogenesis in C3H10T1/2 clone 8 fibroblast cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRetinoic acid receptor RXR-alpha(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50143827((E)-3-[4-(3-Methoxy-5,5,8,8-tetramethyl-5,6,7,8-te...)
Affinity DataEC50:  123nMAssay Description:Effective concentration for lipogenesis induced by retinoid X receptor alpha in C3H10T1/2 clone 8 fibroblast cells; Partial agonistMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRetinoic acid receptor RXR-alpha(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50143821((E)-3-[4-(5,5,8,8-Tetramethyl-3-propoxy-5,6,7,8-te...)
Affinity DataEC50:  137nMAssay Description:Effective concentration for Retinoid X receptor alpha activity in CV-1 cells; Partial agonistMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRetinoic acid receptor RXR-alpha(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50143826((E)-3-[4-(5,5,8,8-Tetramethyl-5,6,7,8-tetrahydro-n...)
Affinity DataEC50:  4nMAssay Description:Effective concentration for lipogenesis induced by retinoid X receptor alpha in C3H10T1/2 clone 8 fibroblast cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRetinoic acid receptor alpha(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50143828(3-[4-(5,5,8,8-Tetramethyl-5,6,7,8-tetrahydro-napht...)
Affinity DataEC50: >1.00E+4nMAssay Description:Effective concentration for Retinoic acid receptor alpha activity in CV-1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRetinoic acid receptor alpha(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50143821((E)-3-[4-(5,5,8,8-Tetramethyl-3-propoxy-5,6,7,8-te...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibitory concentration for lipogenesis induced by retinoic acid receptor alpha in C3H10T1/2 clone 8 fibroblast cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRetinoic acid receptor RXR-alpha(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50143826((E)-3-[4-(5,5,8,8-Tetramethyl-5,6,7,8-tetrahydro-n...)
Affinity DataKi:  5nMAssay Description:Binding affinity for retinoid X receptor alpha (RXRalpha), using 9-cis-[3H]-retinoic acidMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
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