Compile Data Set for Download or QSAR
Report error Found 8 Enz. Inhib. hit(s) with all data for entry = 50014241
TargetSolute carrier family 15 member 1(Human)
University of Tromsø

Curated by ChEMBL
LigandPNGBDBM50139892((S)-2-((S)-2-Amino-3-phenyl-propionylamino)-propio...)
Affinity DataIC50: 180nMAssay Description:Concentration required to inhibit the maximum [14C]Gly-Sar uptake by human Intestinal peptide transporter PepT1 in Caco-2 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSolute carrier family 15 member 1(Human)
University of Tromsø

Curated by ChEMBL
LigandPNGBDBM50139894(Phe-Gly | ((S)-3-Amino-2-oxo-4-phenyl-butylamino)-...)
Affinity DataIC50: 200nMAssay Description:Concentration required to inhibit the maximum [14C]Gly-Sar uptake by human Intestinal peptide transporter PepT1 in Caco-2 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSolute carrier family 15 member 1(Human)
University of Tromsø

Curated by ChEMBL
LigandPNGBDBM50139890((S)-5-Amino-4-oxo-6-phenyl-hexanoic acid | CHEMBL1...)
Affinity DataIC50: 400nMAssay Description:Concentration required to inhibit the maximum [14C]Gly-Sar uptake by human Intestinal peptide transporter PepT1 in Caco-2 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSolute carrier family 15 member 1(Human)
University of Tromsø

Curated by ChEMBL
LigandPNGBDBM50139893((E)-(S)-5-Amino-4-(S)-hydroxy-6-phenyl-hex-2-enoic...)
Affinity DataIC50: 4.05E+4nMAssay Description:Concentration required to inhibit the maximum [14C]Gly-Sar uptake by human Intestinal peptide transporter PepT1 in Caco-2 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSolute carrier family 15 member 1(Human)
University of Tromsø

Curated by ChEMBL
LigandPNGBDBM50139892((S)-2-((S)-2-Amino-3-phenyl-propionylamino)-propio...)
Affinity DataKi:  180nMAssay Description:Affinity fo the compound against human Intestinal peptide transporter PepT1 in Caco-2 cells was measured as inhibition of [14C]Gly-Sar uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSolute carrier family 15 member 1(Human)
University of Tromsø

Curated by ChEMBL
LigandPNGBDBM50139894(Phe-Gly | ((S)-3-Amino-2-oxo-4-phenyl-butylamino)-...)
Affinity DataKi:  200nMAssay Description:Affinity fo the compound against human Intestinal peptide transporter PepT1 in Caco-2 cells was measured as inhibition of [14C]Gly-Sar uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSolute carrier family 15 member 1(Human)
University of Tromsø

Curated by ChEMBL
LigandPNGBDBM50139890((S)-5-Amino-4-oxo-6-phenyl-hexanoic acid | CHEMBL1...)
Affinity DataKi:  400nMAssay Description:Affinity fo the compound against human Intestinal peptide transporter PepT1 in Caco-2 cells was measured as inhibition of [14C]Gly-Sar uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSolute carrier family 15 member 1(Human)
University of Tromsø

Curated by ChEMBL
LigandPNGBDBM50139893((E)-(S)-5-Amino-4-(S)-hydroxy-6-phenyl-hex-2-enoic...)
Affinity DataKi:  3.98E+4nMAssay Description:Affinity fo the compound against human Intestinal peptide transporter PepT1 in Caco-2 cells was measured as inhibition of [14C]Gly-Sar uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed