Compile Data Set for Download or QSAR
Report error Found 9 Enz. Inhib. hit(s) with all data for entry = 50037275
TargetDelta-type opioid receptor(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50138632(1-Phenyl-cyclopentanecarboxylic acid [(S)-5-(3-hyd...)
Affinity DataIC50: 1.80nMAssay Description:Inverse agonist potency at cloned human delta-opioid receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50138633(1-Phenyl-cyclopentanecarboxylic acid [5-(3-hydroxy...)
Affinity DataIC50: 2.40nMAssay Description:Inverse agonist potency at cloned human delta-opioid receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50064515(RTI-5989-25 | 3-[3,4-Dimethyl-1-(3-o-tolyl-allyl)-...)
Affinity DataIC50: 2.80nMAssay Description:Inverse agonist potency at cloned human opioid receptor delta 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50138634(1-Phenyl-cyclopentanecarboxylic acid [(R)-5-(3-hyd...)
Affinity DataIC50: 15nMAssay Description:Inverse agonist potency at cloned human opioid receptor delta 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM21864(NALTRINDOLE | (8R)-7-(cyclopropylmethyl)-5,6,7,8,1...)
Affinity DataKi:  0.0700nMAssay Description:[3H]-Cl-DPDPE competition binding assay using human cloned opioid receptor delta 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50138632(1-Phenyl-cyclopentanecarboxylic acid [(S)-5-(3-hyd...)
Affinity DataKi:  0.960nMAssay Description:[3H]-Cl-DPDPE competition binding assay using human cloned opioid receptor delta 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50138633(1-Phenyl-cyclopentanecarboxylic acid [5-(3-hydroxy...)
Affinity DataKi:  2.10nMAssay Description:[3H]-Cl-DPDPE competition binding assay using human cloned opioid receptor delta 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50138634(1-Phenyl-cyclopentanecarboxylic acid [(R)-5-(3-hyd...)
Affinity DataKi:  9.30nMAssay Description:[3H]-Cl-DPDPE competition binding assay using human cloned opioid receptor delta 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50006946(ICI-174864 | CHEMBL47545 | 2-[2-(2-{2-[2-Diallylam...)
Affinity DataKi:  19nMAssay Description:Binding affinity towards opioid receptor delta 1 expressed in CHO cells was determined by using [3H]DPDPE as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed