Compile Data Set for Download or QSAR
Report error Found 35 Enz. Inhib. hit(s) with all data for entry = 50048564
TargetHistone deacetylase(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50005711(GNF-Pf-1011 | CHEBI:46024 | TRICHOSTATIN | Trichos...)
Affinity DataIC50: 3.40nMAssay Description:Inhibitory activity against Histone deacetylase (HDAC) in K 562 erythroleukemia cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2018
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM19149(Zolinza | suberoylanilide hydroxamic acid | CHEMBL...)
Affinity DataIC50: 10nMAssay Description:Inhibitory activity against Histone deacetylase (HDAC) in K 562 erythroleukemia cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2018
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetHistone deacetylase(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50222391(CHEMBL127953)
Affinity DataIC50: 30nMAssay Description:In vitro inhibition of Histone deacetylase in K 562 erythroleukemia cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2018
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50222389(CHEMBL125416)
Affinity DataIC50: 60nMAssay Description:In vitro inhibition of Histone deacetylase in K 562 erythroleukemia cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2018
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50222393(CHEMBL340725)
Affinity DataIC50: 90nMAssay Description:In vitro inhibition of Histone deacetylase in K 562 erythroleukemia cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2018
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50221965(CHEMBL113303)
Affinity DataIC50: 110nMAssay Description:Inhibitory activity against Histone deacetylase (HDAC) in K 562 erythroleukemia cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2018
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50222378(CHEMBL127627)
Affinity DataIC50: 250nMAssay Description:Inhibitory activity against Histone deacetylase (HDAC) in K 562 erythroleukemia cells (Radioactivity based HDAC assay)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2018
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50222370(CHEMBL126289)
Affinity DataIC50: 310nMAssay Description:In vitro inhibition of Histone deacetylase in K 562 erythroleukemia cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2018
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50222374(CHEMBL423515)
Affinity DataIC50: 320nMAssay Description:In vitro inhibition of Histone deacetylase in K 562 erythroleukemia cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2018
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50222396(CHEMBL338816)
Affinity DataIC50: 340nMAssay Description:In vitro inhibition of Histone deacetylase in K 562 erythroleukemia cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2018
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50222385(CHEMBL127179)
Affinity DataIC50: 430nMAssay Description:In vitro inhibition of Histone deacetylase in K 562 erythroleukemia cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2018
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50222369(CHEMBL127328)
Affinity DataIC50: 520nMAssay Description:In vitro inhibition of Histone deacetylase in K 562 erythroleukemia cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2018
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50222390(CHEMBL127606)
Affinity DataIC50: 540nMAssay Description:In vitro inhibition of Histone deacetylase in K 562 erythroleukemia cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2018
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50222371(CHEMBL126777)
Affinity DataIC50: 580nMAssay Description:In vitro inhibition of Histone deacetylase in K 562 erythroleukemia cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2018
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50222392(CHEMBL340721)
Affinity DataIC50: 610nMAssay Description:In vitro inhibition of Histone deacetylase in K 562 erythroleukemia cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2018
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50222367(CHEMBL127351)
Affinity DataIC50: 620nMAssay Description:In vitro inhibition of Histone deacetylase in K 562 erythroleukemia cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2018
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50222381(CHEMBL126465)
Affinity DataIC50: 990nMAssay Description:In vitro inhibition of Histone deacetylase in K 562 erythroleukemia cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2018
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50222394(CHEMBL126355)
Affinity DataIC50: 1.10E+3nMAssay Description:In vitro inhibition of Histone deacetylase in K 562 erythroleukemia cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2018
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50222375(CHEMBL126947)
Affinity DataIC50: 1.50E+3nMAssay Description:In vitro inhibition of Histone deacetylase in K 562 erythroleukemia cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2018
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50222373(CHEMBL338141)
Affinity DataIC50: 1.80E+3nMAssay Description:In vitro inhibition of Histone deacetylase in K 562 erythroleukemia cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2018
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50222382(CHEMBL126874)
Affinity DataIC50: 1.83E+3nMAssay Description:Inhibitory activity against Histone deacetylase (HDAC) in K 562 erythroleukemia cells (Radioactivity based HDAC assay)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2018
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM19410(benzamide-type inhibitor, 3 | CHEMBL27759 | pyridi...)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibitory activity against Histone deacetylase (HDAC) in K 562 erythroleukemia cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2018
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50222377(CHEMBL272294)
Affinity DataIC50: 2.00E+3nMAssay Description:In vitro inhibition of Histone deacetylase in K 562 erythroleukemia cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2018
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50218532(CHEMBL112148)
Affinity DataIC50: 2.90E+3nMAssay Description:Inhibitory activity against Histone deacetylase (HDAC) in K 562 erythroleukemia cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2018
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50222376(CHEMBL127949)
Affinity DataIC50: 6.40E+3nMAssay Description:In vitro inhibition of Histone deacetylase in K 562 erythroleukemia cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2018
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50222380(CHEMBL126675)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibitory activity against Histone deacetylase (HDAC) in K 562 erythroleukemia cells (Radioactivity based HDAC assay)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2018
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50222388(CHEMBL129419)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibitory activity against Histone deacetylase (HDAC) in K 562 erythroleukemia cells (Radioactivity based HDAC assay)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2018
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50222387(CHEMBL126478)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibitory activity against Histone deacetylase (HDAC) in K 562 erythroleukemia cells (Radioactivity based HDAC assay)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2018
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50222386(CHEMBL126828)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibitory activity against Histone deacetylase (HDAC) in K 562 erythroleukemia cells (Radioactivity based HDAC assay)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2018
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50222372(CHEMBL126815)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibitory activity against Histone deacetylase (HDAC) in K 562 erythroleukemia cells (Radioactivity based HDAC assay)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2018
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50222379(CHEMBL129641)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibitory activity against Histone deacetylase (HDAC) in K 562 erythroleukemia cells (Radioactivity based HDAC assay)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2018
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50222384(CHEMBL129739)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibitory activity against Histone deacetylase (HDAC) in K 562 erythroleukemia cells (Radioactivity based HDAC assay)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2018
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50222383(CHEMBL127401)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibitory activity against Histone deacetylase (HDAC) in K 562 erythroleukemia cells (Radioactivity based HDAC assay)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2018
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50222395(CHEMBL125919)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibitory activity against Histone deacetylase (HDAC) in K 562 erythroleukemia cells (Radioactivity based HDAC assay)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2018
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50222368(CHEMBL127964)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibitory activity against Histone deacetylase (HDAC) in K 562 erythroleukemia cells (Radioactivity based HDAC assay)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2018
Entry Details Article
PubMed