Compile Data Set for Download or QSAR
Report error Found 108 Enz. Inhib. hit(s) with all data for entry = 50013815
TargetMelanocortin receptor 5(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50134950(H-Tyr-Val-Nle-Gly-His-D-Nal(2')-Arg-D-Nal(2')-Asp-...)
Affinity DataEC50: >1.00E+4nMAssay Description:Intracellular cAMP accumulation in human Melanocortin 5 receptor functional assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50134955(H-Tyr-Val-Nle-Gly-Pro-D-Nal(2')-Arg-Trp-Asp-Arg-Ph...)
Affinity DataEC50: >1.00E+4nMAssay Description:Intracellular cAMP accumulation in human Melanocortin 5 receptor functional assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50134957(H-Tyr-Val-Nle-Gly-MePhe-Phe-Arg-D-Nal(2)-Asp-Arg-P...)
Affinity DataEC50:  210nMAssay Description:Intracellular cAMP accumulation in human Melanocortin 5 receptor functional assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50134943(H-Tyr-Val-Nle-Gly-Aib-Phe-Arg-D-Nal(2')-Asp-Arg-Ph...)
Affinity DataEC50:  1.80nMAssay Description:Intracellular cAMP accumulation in human Melanocortin 5 receptor functional assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50134943(H-Tyr-Val-Nle-Gly-Aib-Phe-Arg-D-Nal(2')-Asp-Arg-Ph...)
Affinity DataEC50: >1.00E+4nMAssay Description:Intracellular cAMP accumulation in Melanocortin 4 receptor functional assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50134957(H-Tyr-Val-Nle-Gly-MePhe-Phe-Arg-D-Nal(2)-Asp-Arg-P...)
Affinity DataEC50:  53nMAssay Description:Intracellular cAMP accumulation in Melanocortin 4 receptor functional assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 3(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50134953(H-Tyr-Val-c[Cys-Gly-His-Phe-Arg-Trp-Cys]-Arg-Phe-G...)
Affinity DataEC50:  36nMAssay Description:Intracellular cAMP accumulation in human Melanocortin 3 receptor functional assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50134953(H-Tyr-Val-c[Cys-Gly-His-Phe-Arg-Trp-Cys]-Arg-Phe-G...)
Affinity DataEC50:  9nMAssay Description:Intracellular cAMP accumulation in Melanocortin 4 receptor functional assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50134951(H-Tyr-Val-Nle-c[Asp-His-Phe-Arg-Trp-Lys]-Arg-Phe-G...)
Affinity DataEC50:  340nMAssay Description:Intracellular cAMP accumulation in Melanocortin 4 receptor functional assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50134949(H-Tyr-Val-Nle-c[Cys-His-Phe-Arg-Trp-D-Cys]-Arg-Phe...)
Affinity DataEC50:  83nMAssay Description:Intracellular cAMP accumulation in Melanocortin 4 receptor functional assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50134942(H-Tyr-Val-c[Cys-Gly-His-Phe-Arg-Trp-D-Cys]-Arg-Phe...)
Affinity DataEC50: >1.00E+4nMAssay Description:Intracellular cAMP accumulation in Melanocortin 4 receptor functional assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 3(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50134942(H-Tyr-Val-c[Cys-Gly-His-Phe-Arg-Trp-D-Cys]-Arg-Phe...)
Affinity DataEC50: >1.00E+4nMAssay Description:Intracellular cAMP accumulation in human Melanocortin 3 receptor functional assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 3(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50134950(H-Tyr-Val-Nle-Gly-His-D-Nal(2')-Arg-D-Nal(2')-Asp-...)
Affinity DataEC50:  12nMAssay Description:Intracellular cAMP accumulation in human Melanocortin 3 receptor functional assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50134949(H-Tyr-Val-Nle-c[Cys-His-Phe-Arg-Trp-D-Cys]-Arg-Phe...)
Affinity DataEC50:  270nMAssay Description:Intracellular cAMP accumulation in human Melanocortin 5 receptor functional assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 3(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50134955(H-Tyr-Val-Nle-Gly-Pro-D-Nal(2')-Arg-Trp-Asp-Arg-Ph...)
Affinity DataEC50:  1.70E+3nMAssay Description:Intracellular cAMP accumulation in human Melanocortin 3 receptor functional assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50134951(H-Tyr-Val-Nle-c[Asp-His-Phe-Arg-Trp-Lys]-Arg-Phe-G...)
Affinity DataEC50:  200nMAssay Description:Intracellular cAMP accumulation in human Melanocortin 5 receptor functional assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 3(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50134947(H-Tyr-Val-Nle-Gly-His-Phe-Arg-D-Nal(2')-Asp-Arg-Ph...)
Affinity DataEC50:  2.40E+3nMAssay Description:Intracellular cAMP accumulation in human Melanocortin 3 receptor functional assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 3(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50134946(H-Tyr-Val-Nle-Gly-His-D-Nal(2')-Arg-Trp-Asp-Arg-Ph...)
Affinity DataEC50: >1.00E+4nMAssay Description:Intracellular cAMP accumulation in human Melanocortin 3 receptor functional assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 3(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50134957(H-Tyr-Val-Nle-Gly-MePhe-Phe-Arg-D-Nal(2)-Asp-Arg-P...)
Affinity DataEC50:  150nMAssay Description:Intracellular cAMP accumulation in human Melanocortin 3 receptor functional assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 3(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50134943(H-Tyr-Val-Nle-Gly-Aib-Phe-Arg-D-Nal(2')-Asp-Arg-Ph...)
Affinity DataEC50: >1.00E+4nMAssay Description:Intracellular cAMP accumulation in human Melanocortin 3 receptor functional assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 3(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50134949(H-Tyr-Val-Nle-c[Cys-His-Phe-Arg-Trp-D-Cys]-Arg-Phe...)
Affinity DataEC50:  39nMAssay Description:Intracellular cAMP accumulation in human Melanocortin 3 receptor functional assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 3(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50134954(H-Tyr-Val-Nle-c[Cys-His-Phe-Arg-Trp-Cys]-Arg-Phe-G...)
Affinity DataEC50:  4.20nMAssay Description:Intracellular cAMP accumulation in human Melanocortin 3 receptor functional assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 3(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50134958(H-Tyr-Val-Nle-c[D-Cys-His-Phe-Arg-Trp-Cys]-Arg-Phe...)
Affinity DataEC50:  210nMAssay Description:Intracellular cAMP accumulation in human Melanocortin 3 receptor functional assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 3(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50134959(H-Tyr-Val-Nle-c[Pen-His-Phe-Arg-Trp-Cys]-Arg-Phe-G...)
Affinity DataEC50:  19nMAssay Description:Intracellular cAMP accumulation in human Melanocortin 3 receptor functional assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 3(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50134945(H-Tyr-Val-Nle-Gly-His-Phe-Arg-Trp-Asp-Arg-Phe-Gly-...)
Affinity DataEC50:  1.60nMAssay Description:Intracellular cAMP accumulation in human Melanocortin 3 receptor functional assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 3(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50134948(H-Tyr-Val-Met-Gly-His-Phe-Arg-Trp-Asp-Arg-Phe-Gly-...)
Affinity DataEC50:  3.70nMAssay Description:Intracellular cAMP accumulation in human Melanocortin 3 receptor functional assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 3(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50134944(H-Tyr-Val-c[Pen-Gly-His-Phe-Arg-Trp-Cys]-Arg-Phe-G...)
Affinity DataEC50:  400nMAssay Description:Intracellular cAMP accumulation in human Melanocortin 3 receptor functional assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 3(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50134951(H-Tyr-Val-Nle-c[Asp-His-Phe-Arg-Trp-Lys]-Arg-Phe-G...)
Affinity DataEC50:  240nMAssay Description:Intracellular cAMP accumulation in human Melanocortin 3 receptor functional assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50134942(H-Tyr-Val-c[Cys-Gly-His-Phe-Arg-Trp-D-Cys]-Arg-Phe...)
Affinity DataEC50: >1.00E+4nMAssay Description:Intracellular cAMP accumulation in human Melanocortin 5 receptor functional assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 3(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50134956(H-Tyr-Val-c[Cys-Gly-His-Phe-Arg-Trp-Pen]-Arg-Phe-G...)
Affinity DataEC50: >1.00E+4nMAssay Description:Intracellular cAMP accumulation in human Melanocortin 3 receptor functional assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 3(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50134952(H-Tyr-Val-c[D-Cys-Gly-His-Phe-Arg-Trp-Cys]-Arg-Phe...)
Affinity DataEC50: >1.00E+4nMAssay Description:Intracellular cAMP accumulation in human Melanocortin 3 receptor functional assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50134948(H-Tyr-Val-Met-Gly-His-Phe-Arg-Trp-Asp-Arg-Phe-Gly-...)
Affinity DataEC50:  180nMAssay Description:Intracellular cAMP accumulation in Melanocortin 4 receptor functional assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50134947(H-Tyr-Val-Nle-Gly-His-Phe-Arg-D-Nal(2')-Asp-Arg-Ph...)
Affinity DataEC50: >1.00E+4nMAssay Description:Intracellular cAMP accumulation in Melanocortin 4 receptor functional assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50134944(H-Tyr-Val-c[Pen-Gly-His-Phe-Arg-Trp-Cys]-Arg-Phe-G...)
Affinity DataEC50: >1.00E+4nMAssay Description:Intracellular cAMP accumulation in human Melanocortin 5 receptor functional assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50134944(H-Tyr-Val-c[Pen-Gly-His-Phe-Arg-Trp-Cys]-Arg-Phe-G...)
Affinity DataEC50: >1.00E+4nMAssay Description:Intracellular cAMP accumulation in Melanocortin 4 receptor functional assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50134953(H-Tyr-Val-c[Cys-Gly-His-Phe-Arg-Trp-Cys]-Arg-Phe-G...)
Affinity DataEC50:  450nMAssay Description:Intracellular cAMP accumulation in human Melanocortin 5 receptor functional assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50134952(H-Tyr-Val-c[D-Cys-Gly-His-Phe-Arg-Trp-Cys]-Arg-Phe...)
Affinity DataEC50:  250nMAssay Description:Intracellular cAMP accumulation in Melanocortin 4 receptor functional assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50134945(H-Tyr-Val-Nle-Gly-His-Phe-Arg-Trp-Asp-Arg-Phe-Gly-...)
Affinity DataEC50:  99nMAssay Description:Intracellular cAMP accumulation in human Melanocortin 5 receptor functional assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50134950(H-Tyr-Val-Nle-Gly-His-D-Nal(2')-Arg-D-Nal(2')-Asp-...)
Affinity DataEC50:  12nMAssay Description:Intracellular cAMP accumulation in Melanocortin 4 receptor functional assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50134955(H-Tyr-Val-Nle-Gly-Pro-D-Nal(2')-Arg-Trp-Asp-Arg-Ph...)
Affinity DataEC50:  50nMAssay Description:Intracellular cAMP accumulation in Melanocortin 4 receptor functional assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50134946(H-Tyr-Val-Nle-Gly-His-D-Nal(2')-Arg-Trp-Asp-Arg-Ph...)
Affinity DataEC50:  24nMAssay Description:Intracellular cAMP accumulation in Melanocortin 4 receptor functional assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50134946(H-Tyr-Val-Nle-Gly-His-D-Nal(2')-Arg-Trp-Asp-Arg-Ph...)
Affinity DataEC50: >1.00E+4nMAssay Description:Intracellular cAMP accumulation in human Melanocortin 5 receptor functional assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50134956(H-Tyr-Val-c[Cys-Gly-His-Phe-Arg-Trp-Pen]-Arg-Phe-G...)
Affinity DataEC50: >1.00E+4nMAssay Description:Intracellular cAMP accumulation in Melanocortin 4 receptor functional assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50134948(H-Tyr-Val-Met-Gly-His-Phe-Arg-Trp-Asp-Arg-Phe-Gly-...)
Affinity DataEC50:  550nMAssay Description:Intracellular cAMP accumulation in human Melanocortin 5 receptor functional assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50134958(H-Tyr-Val-Nle-c[D-Cys-His-Phe-Arg-Trp-Cys]-Arg-Phe...)
Affinity DataEC50:  140nMAssay Description:Intracellular cAMP accumulation in human Melanocortin 5 receptor functional assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50134959(H-Tyr-Val-Nle-c[Pen-His-Phe-Arg-Trp-Cys]-Arg-Phe-G...)
Affinity DataEC50:  200nMAssay Description:Intracellular cAMP accumulation in Melanocortin 4 receptor functional assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50134958(H-Tyr-Val-Nle-c[D-Cys-His-Phe-Arg-Trp-Cys]-Arg-Phe...)
Affinity DataEC50:  360nMAssay Description:Intracellular cAMP accumulation in Melanocortin 4 receptor functional assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50134954(H-Tyr-Val-Nle-c[Cys-His-Phe-Arg-Trp-Cys]-Arg-Phe-G...)
Affinity DataEC50:  170nMAssay Description:Intracellular cAMP accumulation in Melanocortin 4 receptor functional assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50134947(H-Tyr-Val-Nle-Gly-His-Phe-Arg-D-Nal(2')-Asp-Arg-Ph...)
Affinity DataEC50:  2.40E+3nMAssay Description:Intracellular cAMP accumulation in human Melanocortin 5 receptor functional assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50134959(H-Tyr-Val-Nle-c[Pen-His-Phe-Arg-Trp-Cys]-Arg-Phe-G...)
Affinity DataEC50:  74nMAssay Description:Intracellular cAMP accumulation in human Melanocortin 5 receptor functional assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
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