Compile Data Set for Download or QSAR
Report error Found 13 Enz. Inhib. hit(s) with all data for entry = 50013765
TargetTubulin alpha-1A chain(Pig)
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50070107((E)-3-(3''-Hydroxy-4''-methoxyphenyl)-2-methyl-1-(...)
Affinity DataIC50: 500nMAssay Description:Concentration that cause a 50% inhibition in tubulin assembly as measured by an increase in turbidity using microtubule assembly assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTubulin alpha-1A chain(Pig)
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50134450(2-[1-(3-Hydroxy-4-methoxy-phenyl)-meth-(Z)-ylidene...)
Affinity DataIC50: 2.20E+4nMAssay Description:Concentration that cause a 50% inhibition in tubulin assembly as measured by an increase in turbidity using microtubule assembly assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTubulin alpha-1A chain(Pig)
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50134459(2-(3-Hydroxy-4-methoxy-phenyl)-6,7,8-trimethoxy-ch...)
Affinity DataIC50: 2.50E+4nMAssay Description:Concentration that cause a 50% inhibition in tubulin assembly as measured by an increase in turbidity using microtubule assembly assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTubulin alpha-1A/beta chain(Pig)
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50134459(2-(3-Hydroxy-4-methoxy-phenyl)-6,7,8-trimethoxy-ch...)
Affinity DataIC50: 4.00E+4nMAssay Description:Ability to inhibit the binding of [3H]colchicine to porcine tubulinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTubulin alpha-1A chain(Pig)
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50134451(2-[1-(3-Fluoro-4-methoxy-phenyl)-meth-(Z)-ylidene]...)
Affinity DataIC50: 5.00E+4nMAssay Description:Concentration that cause a 50% inhibition in tubulin assembly as measured by an increase in turbidity using microtubule assembly assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTubulin alpha-1A chain(Pig)
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50134456(2-[1-(3,4-Dihydroxy-phenyl)-meth-(Z)-ylidene]-5,6,...)
Affinity DataIC50: 5.00E+4nMAssay Description:Concentration that cause a 50% inhibition in tubulin assembly as measured by an increase in turbidity using microtubule assembly assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTubulin alpha-1A chain(Pig)
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50134452(2-[1-(3-Hydroxy-4-methoxy-phenyl)-meth-(Z)-ylidene...)
Affinity DataIC50: 5.00E+4nMAssay Description:Concentration that cause a 50% inhibition in tubulin assembly as measured by an increase in turbidity using microtubule assembly assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTubulin alpha-1A chain(Pig)
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50134460(3',4',-dihydroxy4,5,6-trimethoxyaurone | 2-[1-(3,4...)
Affinity DataIC50: 5.00E+4nMAssay Description:Concentration that cause a 50% inhibition in tubulin assembly as measured by an increase in turbidity using microtubule assembly assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTubulin alpha-1A chain(Pig)
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50134461(2-(3-Hydroxy-4-methoxy-phenyl)-5,6,7-trimethoxy-ch...)
Affinity DataIC50: 5.00E+4nMAssay Description:Concentration that cause a 50% inhibition in tubulin assembly as measured by an increase in turbidity using microtubule assembly assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTubulin alpha-1A chain(Pig)
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50134462(2-(3-Fluoro-4-methoxy-phenyl)-5,6,7-trimethoxy-chr...)
Affinity DataIC50: 5.00E+4nMAssay Description:Concentration that cause a 50% inhibition in tubulin assembly as measured by an increase in turbidity using microtubule assembly assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTubulin alpha-1A chain(Pig)
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50134458(2-(3-Fluoro-4-methoxy-phenyl)-6,7,8-trimethoxy-chr...)
Affinity DataIC50: 5.00E+4nMAssay Description:Concentration that cause a 50% inhibition in tubulin assembly as measured by an increase in turbidity using microtubule assembly assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTubulin alpha-1A chain(Pig)
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50134454(2-[1-(3-Fluoro-4-methoxy-phenyl)-meth-(Z)-ylidene]...)
Affinity DataIC50: 5.00E+4nMAssay Description:Concentration that cause a 50% inhibition in tubulin assembly as measured by an increase in turbidity using microtubule assembly assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTubulin alpha-1A/beta chain(Pig)
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50134450(2-[1-(3-Hydroxy-4-methoxy-phenyl)-meth-(Z)-ylidene...)
Affinity DataIC50: 6.00E+4nMAssay Description:Ability to inhibit the binding of [3H]colchicine to porcine tubulinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed