Compile Data Set for Download or QSAR
Report error Found 99 Enz. Inhib. hit(s) with all data for entry = 50013711
TargetPeroxisome proliferator-activated receptor delta(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50133651(5-{3-[3-(2-Propyl-phenoxy)-propoxy]-phenyl}-oxazol...)
Affinity DataEC50: >3.00E+3nMAssay Description:In vitro activity in human Peroxisome proliferator activated receptor delta-transactivation assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50131503(CHEMBL1783066 | CHEMBL94306 | 5-{3-[3-(4-Phenoxy-2...)
Affinity DataEC50:  26nMAssay Description:In vitro activity in human Peroxisome proliferator activated receptor alpha-transactivation assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50133668(CHEMBL119066 | CHEMBL1783061 | 5-(3-{3-[4-(4,4-Dim...)
Affinity DataEC50: >3.00E+3nMAssay Description:In vitro activity in human Peroxisome proliferator activated receptor delta-transactivation assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50133659(CHEMBL332018 | CHEMBL1783060 | 5-(3-{3-[4-(4,4-Dif...)
Affinity DataEC50: >3.00E+3nMAssay Description:In vitro activity in human Peroxisome proliferator activated receptor delta-transactivation assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50133666(CHEMBL1783045 | CHEMBL122418 | 5-{3-[3-(4-Cyclohex...)
Affinity DataEC50:  76nMAssay Description:In vitro activity in human Peroxisome proliferator activated receptor alpha-transactivation assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50133654(CHEMBL119496 | CHEMBL1783041 | 5-{3-[3-(4-Cyclohex...)
Affinity DataEC50:  130nMAssay Description:In vitro activity in human Peroxisome proliferator activated receptor alpha-transactivation assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50133657(5-{3-[3-(4-Cyclohexylidenemethyl-2-propyl-phenoxy)...)
Affinity DataEC50: >3.00E+3nMAssay Description:In vitro activity in human Peroxisome proliferator activated receptor delta-transactivation assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50133659(CHEMBL332018 | CHEMBL1783060 | 5-(3-{3-[4-(4,4-Dif...)
Affinity DataEC50: >3.00E+3nMAssay Description:In vitro activity in human Peroxisome proliferator activated receptor alpha-transactivation assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50133654(CHEMBL119496 | CHEMBL1783041 | 5-{3-[3-(4-Cyclohex...)
Affinity DataEC50: >3.00E+3nMAssay Description:In vitro activity in human Peroxisome proliferator activated receptor delta-transactivation assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50133658(CHEMBL120570 | CHEMBL1783031 | 5-{3-[3-(4-Cyclohex...)
Affinity DataEC50: >3.00E+3nMAssay Description:In vitro activity in human Peroxisome proliferator activated receptor delta-transactivation assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50133652(CHEMBL280293 | CHEMBL1783052 | CHEMBL2037082 | 5-{...)
Affinity DataEC50:  90nMAssay Description:In vitro activity in human peroxisome proliferator activated receptor gamma-transactivation assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50133656(CHEMBL1782067 | CHEMBL117578 | 5-(3-{3-[4-(4-Chlor...)
Affinity DataEC50: >3.00E+3nMAssay Description:In vitro activity in human Peroxisome proliferator activated receptor alpha-transactivation assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50133659(CHEMBL332018 | CHEMBL1783060 | 5-(3-{3-[4-(4,4-Dif...)
Affinity DataEC50: >3.00E+3nMAssay Description:In vitro activity in human peroxisome proliferator activated receptor gamma-transactivation assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50133654(CHEMBL119496 | CHEMBL1783041 | 5-{3-[3-(4-Cyclohex...)
Affinity DataEC50:  110nMAssay Description:In vitro activity in human peroxisome proliferator activated receptor gamma-transactivation assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50133663(CHEMBL331071 | CHEMBL2037183 | 5-{3-[3-(4-Benzoyl-...)
Affinity DataEC50: >3.00E+3nMAssay Description:In vitro activity in human Peroxisome proliferator activated receptor alpha-transactivation assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50133657(5-{3-[3-(4-Cyclohexylidenemethyl-2-propyl-phenoxy)...)
Affinity DataEC50:  170nMAssay Description:In vitro activity in human Peroxisome proliferator activated receptor alpha-transactivation assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50133657(5-{3-[3-(4-Cyclohexylidenemethyl-2-propyl-phenoxy)...)
Affinity DataEC50:  210nMAssay Description:In vitro activity in human peroxisome proliferator activated receptor gamma-transactivation assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50133655(CHEMBL1783050 | CHEMBL118756 | 5-{3-[3-(4-Cyclohex...)
Affinity DataEC50:  55nMAssay Description:In vitro activity in human Peroxisome proliferator activated receptor alpha-transactivation assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50133651(5-{3-[3-(2-Propyl-phenoxy)-propoxy]-phenyl}-oxazol...)
Affinity DataEC50:  81nMAssay Description:In vitro activity in human peroxisome proliferator activated receptor gamma-transactivation assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50133666(CHEMBL1783045 | CHEMBL122418 | 5-{3-[3-(4-Cyclohex...)
Affinity DataEC50:  80nMAssay Description:In vitro activity in human peroxisome proliferator activated receptor gamma-transactivation assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50133668(CHEMBL119066 | CHEMBL1783061 | 5-(3-{3-[4-(4,4-Dim...)
Affinity DataEC50:  90nMAssay Description:In vitro activity in human peroxisome proliferator activated receptor gamma-transactivation assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50133658(CHEMBL120570 | CHEMBL1783031 | 5-{3-[3-(4-Cyclohex...)
Affinity DataEC50:  39nMAssay Description:In vitro activity in human peroxisome proliferator activated receptor gamma-transactivation assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50133668(CHEMBL119066 | CHEMBL1783061 | 5-(3-{3-[4-(4,4-Dim...)
Affinity DataEC50: >3.00E+3nMAssay Description:In vitro activity in human Peroxisome proliferator activated receptor alpha-transactivation assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50133655(CHEMBL1783050 | CHEMBL118756 | 5-{3-[3-(4-Cyclohex...)
Affinity DataEC50:  19nMAssay Description:In vitro activity in human peroxisome proliferator activated receptor gamma-transactivation assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50133663(CHEMBL331071 | CHEMBL2037183 | 5-{3-[3-(4-Benzoyl-...)
Affinity DataEC50: >3.00E+3nMAssay Description:In vitro activity in human Peroxisome proliferator activated receptor delta-transactivation assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50133660(CHEMBL118251 | CHEMBL1783054 | 5-{3-[3-(4-Cyclohep...)
Affinity DataEC50:  54nMAssay Description:In vitro activity in human Peroxisome proliferator activated receptor alpha-transactivation assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50131503(CHEMBL1783066 | CHEMBL94306 | 5-{3-[3-(4-Phenoxy-2...)
Affinity DataEC50: >3.00E+3nMAssay Description:In vitro activity in human Peroxisome proliferator activated receptor delta-transactivation assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50133660(CHEMBL118251 | CHEMBL1783054 | 5-{3-[3-(4-Cyclohep...)
Affinity DataEC50: >3.00E+3nMAssay Description:In vitro activity in human Peroxisome proliferator activated receptor delta-transactivation assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50133666(CHEMBL1783045 | CHEMBL122418 | 5-{3-[3-(4-Cyclohex...)
Affinity DataEC50: >3.00E+3nMAssay Description:In vitro activity in human Peroxisome proliferator activated receptor delta-transactivation assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50133652(CHEMBL280293 | CHEMBL1783052 | CHEMBL2037082 | 5-{...)
Affinity DataEC50:  2.00E+3nMAssay Description:In vitro activity in human Peroxisome proliferator activated receptor alpha-transactivation assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50133651(5-{3-[3-(2-Propyl-phenoxy)-propoxy]-phenyl}-oxazol...)
Affinity DataEC50:  53nMAssay Description:In vitro activity in human Peroxisome proliferator activated receptor alpha-transactivation assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50131503(CHEMBL1783066 | CHEMBL94306 | 5-{3-[3-(4-Phenoxy-2...)
Affinity DataEC50:  14nMAssay Description:In vitro activity in human peroxisome proliferator activated receptor gamma-transactivation assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50133655(CHEMBL1783050 | CHEMBL118756 | 5-{3-[3-(4-Cyclohex...)
Affinity DataEC50: >3.00E+3nMAssay Description:In vitro activity in human Peroxisome proliferator activated receptor delta-transactivation assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50133656(CHEMBL1782067 | CHEMBL117578 | 5-(3-{3-[4-(4-Chlor...)
Affinity DataEC50:  51nMAssay Description:In vitro activity in human peroxisome proliferator activated receptor gamma-transactivation assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50133660(CHEMBL118251 | CHEMBL1783054 | 5-{3-[3-(4-Cyclohep...)
Affinity DataEC50:  35nMAssay Description:In vitro activity in human peroxisome proliferator activated receptor gamma-transactivation assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50133652(CHEMBL280293 | CHEMBL1783052 | CHEMBL2037082 | 5-{...)
Affinity DataEC50: >3.00E+3nMAssay Description:In vitro activity in human Peroxisome proliferator activated receptor delta-transactivation assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50133663(CHEMBL331071 | CHEMBL2037183 | 5-{3-[3-(4-Benzoyl-...)
Affinity DataEC50:  167nMAssay Description:In vitro activity in human peroxisome proliferator activated receptor gamma-transactivation assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50133658(CHEMBL120570 | CHEMBL1783031 | 5-{3-[3-(4-Cyclohex...)
Affinity DataEC50:  35nMAssay Description:In vitro activity of compound in human Peroxisome proliferator activated receptor alpha-transactivation assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50133656(CHEMBL1782067 | CHEMBL117578 | 5-(3-{3-[4-(4-Chlor...)
Affinity DataEC50: >3.00E+3nMAssay Description:In vitro activity in human Peroxisome proliferator activated receptor delta-transactivation assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50133663(CHEMBL331071 | CHEMBL2037183 | 5-{3-[3-(4-Benzoyl-...)
Affinity DataIC50: 19nMAssay Description:In vitro binding affinity against human peroxisome proliferator activated receptor gammaMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50131503(CHEMBL1783066 | CHEMBL94306 | 5-{3-[3-(4-Phenoxy-2...)
Affinity DataIC50: 28nMAssay Description:In vitro binding affinity was tested towards human Peroxisome proliferator activated receptor alphaMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50133661(CHEMBL418874 | CHEMBL1783039 | CHEMBL2037182 | 5-{...)
Affinity DataIC50: 30nMAssay Description:In vitro binding affinity against human peroxisome proliferator activated receptor gammaMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50133661(CHEMBL418874 | CHEMBL1783039 | CHEMBL2037182 | 5-{...)
Affinity DataIC50: 37nMAssay Description:In vitro binding affinity was tested towards human Peroxisome proliferator activated receptor alphaMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50133658(CHEMBL120570 | CHEMBL1783031 | 5-{3-[3-(4-Cyclohex...)
Affinity DataIC50: 37nMAssay Description:In vitro binding affinity against human peroxisome proliferator activated receptor gammaMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50133667(CHEMBL1783035 | CHEMBL118169 | CHEMBL2037181 | 5-{...)
Affinity DataIC50: 42nMAssay Description:In vitro binding affinity was tested towards human Peroxisome proliferator activated receptor alphaMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50133666(CHEMBL1783045 | CHEMBL122418 | 5-{3-[3-(4-Cyclohex...)
Affinity DataIC50: 46nMAssay Description:In vitro binding affinity was tested towards human Peroxisome proliferator activated receptor alphaMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50131503(CHEMBL1783066 | CHEMBL94306 | 5-{3-[3-(4-Phenoxy-2...)
Affinity DataIC50: 57nMAssay Description:In vitro binding affinity against human peroxisome proliferator activated receptor gammaMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50133666(CHEMBL1783045 | CHEMBL122418 | 5-{3-[3-(4-Cyclohex...)
Affinity DataIC50: 59nMAssay Description:In vitro binding affinity against human peroxisome proliferator activated receptor gammaMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50133657(5-{3-[3-(4-Cyclohexylidenemethyl-2-propyl-phenoxy)...)
Affinity DataIC50: 62nMAssay Description:In vitro binding affinity was tested towards human Peroxisome proliferator activated receptor alphaMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50133667(CHEMBL1783035 | CHEMBL118169 | CHEMBL2037181 | 5-{...)
Affinity DataIC50: 63nMAssay Description:In vitro binding affinity against human peroxisome proliferator activated receptor gammaMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
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