Compile Data Set for Download or QSAR
Report error Found 54 Enz. Inhib. hit(s) with all data for entry = 50037198
TargetMelanocortin receptor 4(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50017181(CHEMBL441738)
Affinity DataEC50:  0.0170nMAssay Description:Effective concentration required for the biological activity against human Melanocortin 4 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50133264([(2S,3S)-TMT1]DPDPE | CHEMBL133719)
Affinity DataEC50:  170nMAssay Description:In vitro bioassay data to determine the effective concentration required for antagonistic activity against Opioid receptor delta 1 in functional assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50029747((4S)-4-{[(1S)-1-{[(1S)-1-{[(1S)-1-{[(1S)-1-[({[(2S...)
Affinity DataEC50:  0.0910nMAssay Description:Effective concentration required for the biological activity against human Melanocortin 1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50133273(Ac-Nle4-c[Asp5,D-Phe(pI)7,Lys10]R-MSH(4-10)-NH2 | ...)
Affinity DataEC50:  0.0550nMAssay Description:Effective concentration required for the biological activity against human Melanocortin 1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50029747((4S)-4-{[(1S)-1-{[(1S)-1-{[(1S)-1-{[(1S)-1-[({[(2S...)
Affinity DataEC50:  0.210nMAssay Description:Effective concentration required for the biological activity against human Melanocortin 4 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50133261([(2R,3R)-TMT1]DPDPE | CHEMBL134652)
Affinity DataEC50:  2.20E+3nMAssay Description:In vitro bioassay data to determine the effective concentration required for antagonistic activity against Opioid receptor delta 1 in functional assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50133257([(2S,3R)-TMT1]DPDPE | CHEMBL334369)
Affinity DataEC50:  1.80nMAssay Description:In vitro bioassay data to determine the effective concentration required for antagonistic activity against Opioid receptor delta 1 in functional assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetMelanocortin receptor 3(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50027084(Melatonan)
Affinity DataEC50:  0.270nMAssay Description:Effective concentration required for the biological activity against human Melanocortin 3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50017181(CHEMBL441738)
Affinity DataEC50:  0.0230nMAssay Description:Effective concentration required for the biological activity against human Melanocortin 1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50001683(CHEMBL294616 | 13-[2-Amino-3-(4-hydroxy-phenyl)-pr...)
Affinity DataEC50:  4.10nMAssay Description:In vitro bioassay data to determine the effective concentration required for antagonistic activity against Opioid receptor delta 1 in functional assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50133264([(2S,3S)-TMT1]DPDPE | CHEMBL133719)
Affinity DataEC50:  290nMAssay Description:In vitro bioassay data to determine the effective concentration required for antagonistic activity against Opioid receptor mu 1 in functional assay, ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50133261([(2R,3R)-TMT1]DPDPE | CHEMBL134652)
Affinity DataEC50:  5.00E+4nMAssay Description:In vitro bioassay data to determine the effective concentration required for antagonistic activity against Opioid receptor mu 1 in functional assay, ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50001683(CHEMBL294616 | 13-[2-Amino-3-(4-hydroxy-phenyl)-pr...)
Affinity DataEC50:  7.30E+3nMAssay Description:In vitro bioassay data to determine the effective concentration required for antagonistic activity against Opioid receptor mu 1 in functional assay, ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50121268(21-(2-Acetylamino-hexanoylamino)-7-[3-(diaminometh...)
Affinity DataEC50:  0.0360nMAssay Description:Effective concentration required for the biological activity against human Melanocortin 1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetMelanocortin receptor 3(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50017181(CHEMBL441738)
Affinity DataEC50:  0.130nMAssay Description:Effective concentration required for the biological activity against human Melanocortin 3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50027084(Melatonan)
Affinity DataEC50:  0.0570nMAssay Description:Effective concentration required for the biological activity against human Melanocortin 4 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetMelanocortin receptor 3(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50029747((4S)-4-{[(1S)-1-{[(1S)-1-{[(1S)-1-{[(1S)-1-[({[(2S...)
Affinity DataEC50:  0.670nMAssay Description:Effective concentration required for the biological activity against human Melanocortin 3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50001683(CHEMBL294616 | 13-[2-Amino-3-(4-hydroxy-phenyl)-pr...)
Affinity DataIC50: 1.60nMAssay Description:Binding affinity towards Opioid receptor delta 1 using [3H]- [p-CIPhe4] DPDPE as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50133257([(2S,3R)-TMT1]DPDPE | CHEMBL334369)
Affinity DataIC50: 5nMAssay Description:Binding affinity towards Opioid receptor delta 1 using [3H]- [p-CIPhe4] DPDPE as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetOxytocin receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50027070(CHEMBL2369136)
Affinity DataIC50: 8nMAssay Description:Binding affinity towards oxytocin receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetOxytocin receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50133272([D-Pen1,Glu4,Lys8]OT | CHEMBL406351)
Affinity DataIC50: 130nMAssay Description:Binding affinity towards oxytocin receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetOxytocin receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50133258([D-Pen1,(2S,3R)-p-MeOTMT2,Glu4,Lys8]OT | [D-Pen1,(...)
Affinity DataIC50: 160nMAssay Description:Binding affinity towards oxytocin receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50133264([(2S,3S)-TMT1]DPDPE | CHEMBL133719)
Affinity DataIC50: 210nMAssay Description:Binding affinity towards Opioid receptor delta 1 using [3H]- [p-CIPhe4] DPDPE as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50001683(CHEMBL294616 | 13-[2-Amino-3-(4-hydroxy-phenyl)-pr...)
Affinity DataIC50: 610nMAssay Description:Binding affinity towards Opioid receptor mu 1 using [3H]- CTOP as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50133264([(2S,3S)-TMT1]DPDPE | CHEMBL133719)
Affinity DataIC50: 720nMAssay Description:Binding affinity towards Opioid receptor mu 1 using [3H]- CTOP as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50133261([(2R,3R)-TMT1]DPDPE | CHEMBL134652)
Affinity DataIC50: 3.50E+3nMAssay Description:Binding affinity towards Opioid receptor delta 1 using [3H]- [p-CIPhe4] DPDPE as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50133257([(2S,3R)-TMT1]DPDPE | CHEMBL334369)
Affinity DataIC50: 4.30E+3nMAssay Description:Binding affinity towards Opioid receptor mu 1 using [3H]- CTOP as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetOxytocin receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50027082(CHEMBL2370761)
Affinity DataIC50: 1.90E+4nMAssay Description:Binding affinity towards oxytocin receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetOxytocin receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50027076(CHEMBL2370768)
Affinity DataIC50: 3.60E+4nMAssay Description:Binding affinity towards oxytocin receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50133261([(2R,3R)-TMT1]DPDPE | CHEMBL134652)
Affinity DataIC50: 7.70E+4nMAssay Description:Binding affinity towards Opioid receptor mu 1 using [3H]- CTOP as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50133259(H-Tyr-D-Phe-Gly-D-Trp-N-MeNle-Asp-Phe-NH2 | CHEMBL...)
Affinity DataKi:  0.5nMAssay Description:Binding affinity towards Opioid receptor delta 1 was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50133267(H-Tyr-D-Nle-Gly-Trp-N-MeNle-Asp-Phe-NH2 | CHEMBL13...)
Affinity DataKi:  0.600nMAssay Description:Binding affinity towards Cholecystokinin type B receptor (CCK-B) receptor was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM21136((3S)-3-[(2S)-2-[(2S)-2-(2-{2-[(2S)-2-amino-3-(4-hy...)
Affinity DataKi:  1.30nMAssay Description:Binding affinity towards Cholecystokinin type B receptor (CCK-B) receptor was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM21141((3S)-3-[(2S)-2-[(2R)-2-{2-[(2R)-2-[(2S)-2-amino-3-...)
Affinity DataKi:  1.30nMAssay Description:Binding affinity towards Cholecystokinin type B receptor (CCK-B) receptor was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50133259(H-Tyr-D-Phe-Gly-D-Trp-N-MeNle-Asp-Phe-NH2 | CHEMBL...)
Affinity DataKi:  1.60nMAssay Description:Binding affinity towards Cholecystokinin type B receptor (CCK-B) receptor was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50133267(H-Tyr-D-Nle-Gly-Trp-N-MeNle-Asp-Phe-NH2 | CHEMBL13...)
Affinity DataKi:  1.60nMAssay Description:Binding affinity towards Opioid receptor delta 1 was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM21141((3S)-3-[(2S)-2-[(2R)-2-{2-[(2R)-2-[(2S)-2-amino-3-...)
Affinity DataKi:  1.90nMAssay Description:Binding affinity towards Opioid receptor delta 1 was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50133268(H-Asp-Tyr-D-Phe-Gly-Trp-N-MeNle-Asp-Phe-NH2 | CHEM...)
Affinity DataKi:  2.10nMAssay Description:Binding affinity towards Cholecystokinin type B receptor (CCK-B) receptor was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50133265(H-Tyr-D-Phe-Glu-Trp-N-MeNle-Asp-Phe-NH2 | CHEMBL41...)
Affinity DataKi:  2.10nMAssay Description:Binding affinity towards Cholecystokinin type B receptor (CCK-B) receptor was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50133259(H-Tyr-D-Phe-Gly-D-Trp-N-MeNle-Asp-Phe-NH2 | CHEMBL...)
Affinity DataKi:  5.70nMAssay Description:Binding affinity towards Opioid receptor mu 1 using [3H]- CTOP as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50133265(H-Tyr-D-Phe-Glu-Trp-N-MeNle-Asp-Phe-NH2 | CHEMBL41...)
Affinity DataKi:  6.80nMAssay Description:Binding affinity towards Opioid receptor delta 1 was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM21141((3S)-3-[(2S)-2-[(2R)-2-{2-[(2R)-2-[(2S)-2-amino-3-...)
Affinity DataKi:  20nMAssay Description:Binding affinity towards Opioid receptor mu 1 was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50133267(H-Tyr-D-Nle-Gly-Trp-N-MeNle-Asp-Phe-NH2 | CHEMBL13...)
Affinity DataKi:  25nMAssay Description:Binding affinity towards Opioid receptor mu 1 using [3H]- CTOP as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM21141((3S)-3-[(2S)-2-[(2R)-2-{2-[(2R)-2-[(2S)-2-amino-3-...)
Affinity DataKi:  32nMAssay Description:Binding affinity towards Cholecystokinin type A receptor (CCK-A) receptor was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50133265(H-Tyr-D-Phe-Glu-Trp-N-MeNle-Asp-Phe-NH2 | CHEMBL41...)
Affinity DataKi:  136nMAssay Description:Binding affinity towards Opioid receptor mu 1 using [3H]- CTOP as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50133268(H-Asp-Tyr-D-Phe-Gly-Trp-N-MeNle-Asp-Phe-NH2 | CHEM...)
Affinity DataKi:  250nMAssay Description:Binding affinity towards Opioid receptor delta 1 was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM21136((3S)-3-[(2S)-2-[(2S)-2-(2-{2-[(2S)-2-amino-3-(4-hy...)
Affinity DataKi:  610nMAssay Description:Binding affinity towards Opioid receptor mu 1 using [3H]- CTOP as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM21136((3S)-3-[(2S)-2-[(2S)-2-(2-{2-[(2S)-2-amino-3-(4-hy...)
Affinity DataKi:  870nMAssay Description:Binding affinity towards Cholecystokinin type A receptor (CCK-A) receptor was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50133259(H-Tyr-D-Phe-Gly-D-Trp-N-MeNle-Asp-Phe-NH2 | CHEMBL...)
Affinity DataKi:  1.08E+3nMAssay Description:Binding affinity towards Cholecystokinin type A receptor (CCK-A) receptor was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM21136((3S)-3-[(2S)-2-[(2S)-2-(2-{2-[(2S)-2-amino-3-(4-hy...)
Affinity DataKi:  2.00E+3nMAssay Description:Binding affinity towards Opioid receptor delta 1 was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
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